日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pan-tumor activity of olomorasib, a next-generation KRAS G12C inhibitor in KRAS G12C-mutant advanced solid tumors: a first-in-human study

奥洛莫拉西布(一种新一代 KRAS G12C 抑制剂)在 KRAS G12C 突变型晚期实体瘤中的泛肿瘤活性:一项首次人体研究

Murciano-Goroff, Yonina R; Hollebecque, Antoine; Heist, Rebecca S; Cassier, Philippe A; Han, Ji-Youn; Kim, So Yeon; Sabari, Joshua K; Tosi, Diego; Sacher, Adrian; Burns, Timothy F; Shimizu, Toshio; Reddy Ammakkanavar, Natraj; Spira, Alexander; Gomez-Roca, Carlos; Patnaik, Amita; Cosman, Rasha; Bodor, J Nicholas; Nagasaka, Misako; You, Arthur Xintian; McNeely, Samuel C; Peter, Raimund; Fink, Aaron; Chen, Aaron; Oxnard, Geoffrey R; Willard, Melinda D; Kuboki, Yasutoshi; Koyama, Takafumi

MET alterations are enriched in lung adenocarcinoma brain metastases, defining a distinct biologic subtype

MET基因改变在肺腺癌脑转移瘤中富集,定义了一种独特的生物学亚型。

Burns, Timothy F; Dacic, Sanja; Chakka, Anish; Miller, Ethan; Velez, Maria A; Somasundaram, Ashwin; Bhattacharya, Saveri; Gaither-Davis, Autumn; Devadassan, Princey; Jin, Jingxiao; Kumar, Vinod; Pennathur, Arjun; Xiu, Joanne; Oberley, Matthew; Glantz, Michael J; Aulakh, Sonikpreet; Chandran, Uma R; Bao, Riyue; Tatsuoka, Curtis; Stabile, Laura P

SUNRAY-01 trial protocol: an innovative study design of olomorasib and pembrolizumab with or without chemotherapy in KRAS G12C NSCLC

SUNRAY-01试验方案:一项创新性的研究设计,旨在评估奥洛莫拉西布和帕博利珠单抗联合或不联合化疗治疗KRAS G12C非小细胞肺癌的疗效。

Peters, Solange; Hochmair, Maximilian; Arbour, Kathryn C; Rodriguez, Luis Paz-Ares; Reck, Martin; Leal, Ticiana; R Lindsay, Colin; Shun, Lu; William, William Nassib; Spira, Alexander I; Sabari, Joshua K; Henning Grønberg, Bjørn; Nishio, Makoto; Burns, Timothy F; Girard, Nicolas; Capuzzo, Frederico; Merced, Alyson; Fasnacht, Nicolas; Visseren-Grul, Carla; Negrao, Marcelo V

Advanced hierarchical computational modeling-based rational development of platinum (II) nanocomplex to improve lung cancer therapy.

基于先进分层计算建模的铂(II)纳米复合物合理开发,以改善肺癌治疗

Huang Haozhe, Ji Beihong, Huang Yixian, Li Shichen, Luo Zhangyi, Chen Shangyu, Li Sihan, Chen Yuang, Bain Daniel J, Sun Jingjing, Yang Da, Burns Timothy F, Wang Junmei, Li Song

Phase I/II Trial of Exportin 1 Inhibitor Selinexor plus Docetaxel in Previously Treated, Advanced KRAS-Mutant Non-Small Cell Lung Cancer.

Exportin 1 抑制剂 Selinexor 联合多西他赛治疗既往接受过治疗的晚期 KRAS 突变型非小细胞肺癌的 I/II 期试验

von Itzstein Mitchell S, Burns Timothy F, Dowell Jonathan E, Horn Leora, Camidge D Ross, York Sally J, Eaton Keith D, Kyle Kelly, Fattah Farjana, Liu Jialiang, Mu-Mosley Hong, Gupta Arjun, Nadeem Urooba, Gao Ang, Zhang Song, Gerber David E

Advances in the treatment of KRAS(G12C) mutant non-small cell lung cancer

KRAS(G12C)突变型非小细胞肺癌治疗进展

Shaverdashvili, Khvaramze; Burns, Timothy F

Phase 1 clinical trial of the ataxia telangiectasia and Rad3-related inhibitor berzosertib with irinotecan in patients with advanced solid tumors (ETCTN 9938)

共济失调毛细血管扩张症和 Rad3 相关抑制剂 berzosertib 与伊立替康联合治疗晚期实体瘤患者的 1 期临床试验 (ETCTN 9938)

Villaruz, Liza C; Jin, Jingxiao; Wang, Hong; Lee, James J; Luke, Jason J; Rhee, John C; Waqar, Saiama N; Shapiro, Geoffrey I; Cleary, James; Davar, Diwakar; Burns, Timothy F; Verma, Rashmi; Amin, Manik; Appleman, Leonard; Ciombor, Kristen K; Davis, Elizabeth J; Riess, Jonathan W; Dees, E Claire; Kim, Edward J; Cardin, Dana; Guo, Jianxia; Christner, Susan M; Deppas, Joshua; Parise, Angelina M; Schmitz, John C; Guerrouahen, Bella S; Suchko, Michael; Contreras, Alejandro; Li, Li; Ferry-Galow, Katherine V; Chang, Ting-Chia; Jiwani, Shahanawaz; Bakkenist, Christopher J; Chu, Edward; Gore, Steven D; Beumer, Jan H

Time-Resolved Crystallography Reveals the Mechanisms of GTP hydrolysis for N-RAS and the Oncogenic Mutants G12C, G12V and Q61L

时间分辨晶体学揭示了N-RAS及其致癌突变体G12C、G12V和Q61L的GTP水解机制

Lin, Guowu; Zinser-Peniche, Paola; Zhou, Xiaohong; Santiago, Ulises; Kurnikov, Igor; Russi, Silvia; Chagas, Brisa; Sharpe, May E; Stegmann, Dennis P; Heinig, Shannon A; Goyal, Rohan K; Nagarajan, V; Calero, Daniel; Vergara, Sandra; Deiters, Alexander; Kurnikova, Maria G; Burns, Timothy F; Cohen, Aina; Calero, Guillermo

Corrigendum to "Structure-function studies of the bHLH phosphorylation domain of TWIST1 in prostate cancer cells" [Neoplasia 17 (2014) 85]

对“前列腺癌细胞中 TWIST1 的 bHLH 磷酸化结构域的结构功能研究”的更正[Neoplasia 17 (2014) 85]

Gajula, Rajendra P; Chettiar, Sivarajan T; Williams, Russell D; Nugent, Katriana; Kato, Yoshinori; Wang, Hailun; Malek, Reem; Taparra, Kekoa; Cades, Jessica; Annadanam, Anvesh; Yoon, A-Rum; Fertig, Elana; Firulli, Beth A; Mazzacurati, Lucia; Burns, Timothy F; Firulli, Anthony B; An, Steven S; Tran, Phuoc T

CASTOR1 phosphorylation predicts poor survival in male patients with KRAS-mutated lung adenocarcinoma

CASTOR1磷酸化预示着KRAS突变型肺腺癌男性患者的预后不良

Loo, Suet Kee; Sica, Gabriel; Wang, Xian; Li, Tingting; Chen, Luping; Gaither-Davis, Autumn; Huang, Yufei; Burns, Timothy F; Stabile, Laura P; Gao, Shou-Jiang