日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Elucidating molecularly stratified single agent, and combination, therapeutic strategies targeting MCL1 for lethal prostate cancer.

阐明针对致命性前列腺癌的 MCL1 分子分层单药和联合治疗策略。

Jiménez-Vacas Juan M, Westaby Daniel, Figueiredo Ines, De Haven Brandon Alexis, Padilha Ana, Yuan Wei, Seed George, Bogdan Denisa, Gurel Bora, Bertan Claudia, Miranda Susana, Lambros Maryou, Montero-Hidalgo Antonio J, Coleman Ilsa, Yu Ivan Pak Lok, Buroni Lorenzo, Zeng Wanting, Neeb Antje J, Welti Jon, Rekowski Jan, Paravati Roberta, Gabel Florian, Pandell Nicole, Ferreira Ana, Crespo Mateus, Riisnaes Ruth, Das Souvik, Taylor Joe, Waldron Nick, Hobern Emily, Valenti Melanie, Ning Jian, Bernett Ilona, Liodaki Kate, Persse Thomas, Galipeau Patricia, Wilkinson Scott, Trostel Shana Y, Karzai Fatima, Chau Cindy H, Beatson Erica L, Zhang Xiaohu, Klumpp-Thomas Carleen, Varkaris Andreas, Luque Raul M, Swain Amanda, Raynaud Florence, Lack Nathan A, Thomas Craig J, Ha Gavin, Figg William D, Bezzi Marco, Sowalsky Adam G, Nelson Peter S, Carreira Suzanne, Balk Steven P, de Bono Johann S, Sharp Adam

BH3 mimetics targeting BCL-XL have efficacy in solid tumors with RB1 loss and replication stress.

靶向 BCL-XL 的 BH3 模拟物对 RB1 缺失和复制压力的实体瘤有效

Varkaris Andreas, Wang Keshan, Nouri Mannan, Kozlova Nina, Schmidt Daniel R, Stavridi Anastasia, Arai Seiji, Ambrosio Nicholas, Poluben Larysa, Jimenez-Vacas Juan M, Westaby Daniel, Carmichael Juliet, Xie Fang, Figueiredo Ines, Buroni Lorenzo, Neeb Antje, Gurel Bora, Chevalier Nicholas, Brown Lisha, Voznesensky Olga, Chen Shao-Yong, Russo Joshua W, Yuan Xin, Juric Dejan, Beltran Himisha, De Bono Johann S, Vander Heiden Matthew G, Einstein David J, Muranen Taru, Corey Eva, Sharp Adam, Balk Steven P

The Evolution of Antimicrobial Resistance in Acinetobacter baumannii and New Strategies to Fight It

鲍曼不动杆菌抗菌素耐药性的演变及其新的应对策略

Scoffone, Viola Camilla; Trespidi, Gabriele; Barbieri, Giulia; Arshad, Arooba; Israyilova, Aygun; Buroni, Silvia

Identification of a New FtsZ Inhibitor by Virtual Screening, Mechanistic Insights, and Structure-Activity Relationship Analyses

通过虚拟筛选、机制研究和构效关系分析鉴定一种新的FtsZ抑制剂

Sciò, Pietro; Scoffone, Viola Camilla; Parisi, Anastasia; Bufano, Marianna; Caneva, Martina; Trespidi, Gabriele; Irudal, Samuele; Barbieri, Giulia; Cariani, Lisa; Orena, Beatrice Silvia; Daccò, Valeria; Imperi, Francesco; Buroni, Silvia; Coluccia, Antonio

BCL2 expression is enriched in advanced prostate cancer with features of lineage plasticity

BCL2表达在具有谱系可塑性特征的晚期前列腺癌中富集

Westaby, Daniel; Jiménez-Vacas, Juan M; Figueiredo, Ines; Rekowski, Jan; Pettinger, Claire; Gurel, Bora; Lundberg, Arian; Bogdan, Denisa; Buroni, Lorenzo; Neeb, Antje; Padilha, Ana; Taylor, Joe; Zeng, Wanting; Das, Souvik; Hobern, Emily; Riisnaes, Ruth; Crespo, Mateus; Miranda, Susana; Ferreira, Ana; Hanratty, Brian P; Nava Rodrigues, Daniel; Bertan, Claudia; Seed, George; Fenor de La Maza, Maria de Los Dolores; Guo, Christina; Carmichael, Juliet; Grochot, Rafael; Chandran, Khobe; Stavridi, Anastasia; Varkaris, Andreas; Stylianou, Nataly; Hollier, Brett G; Tunariu, Nina; Balk, Steven P; Carreira, Suzanne; Yuan, Wei; Nelson, Peter S; Corey, Eva; Haffner, Michael; de Bono, Johann; Sharp, Adam

New Antimicrobial Strategies to Treat Multi-Drug Resistant Infections Caused by Gram-Negatives in Cystic Fibrosis

治疗囊性纤维化中革兰氏阴性菌引起的多重耐药感染的新型抗菌策略

Scoffone, Viola Camilla; Barbieri, Giulia; Irudal, Samuele; Trespidi, Gabriele; Buroni, Silvia

Characterization of the dispirotripiperazine derivative PDSTP as antibiotic adjuvant and antivirulence compound against Pseudomonas aeruginosa

对二螺三哌嗪衍生物PDSTP作为抗生素佐剂和抗铜绿假单胞菌毒力化合物的特性进行表征

Bonacorsi, Andrea; Trespidi, Gabriele; Scoffone, Viola C; Irudal, Samuele; Barbieri, Giulia; Riabova, Olga; Monakhova, Natalia; Makarov, Vadim; Buroni, Silvia

B7-H3 as a Therapeutic Target in Advanced Prostate Cancer.

B7-H3 作为晚期前列腺癌的治疗靶点

Guo Christina, Figueiredo Ines, Gurel Bora, Neeb Antje, Seed George, Crespo Mateus, Carreira Suzanne, Rekowski Jan, Buroni Lorenzo, Welti Jon, Bogdan Denisa, Gallagher Lewis, Sharp Adam, Fenor de la Maza Maria D, Rescigno Pasquale, Westaby Daniel, Chandran Khobe, Riisnaes Ruth, Ferreira Ana, Miranda Susana, Calì Bianca, Alimonti Andrea, Bressan Silvia, Nguyen Alana H T, Shen Michael M, Hawley Jessica E, Obradovic Aleksandar, Drake Charles G, Bertan Claudia, Baker Chloe, Tunariu Nina, Yuan Wei, de Bono Johann S

Critical role of antioxidant programs in enzalutamide-resistant prostate cancer

抗氧化剂在恩杂鲁胺耐药前列腺癌中的关键作用

Eliot B Blatt, Karla Parra, Antje Neeb, Lorenzo Buroni, Denisa Bogdan, Wei Yuan, Yunpeng Gao, Collin Gilbreath, Alec Paschalis, Suzanne Carreira, Ralph J DeBerardinis, Ram S Mani, Johann S de Bono, Ganesh V Raj

Editorial: Burkholderia spp.-transmission, pathogenesis, host-pathogen interaction, prevention and treatment

社论:伯克霍尔德菌属——传播、致病机制、宿主-病原体相互作用、预防和治疗

Buroni, Silvia; Samy, Ramar Perumal