日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemical optimization of the exercise mimetic SLU-PP-332 enables insight into estrogen-related receptor signaling

对运动模拟剂SLU-PP-332进行化学优化,有助于深入了解雌激素相关受体信号传导。

Okda, Hazem Essam; Zhao, Puhan; Hayes, Matt; Duvall, Colten; Quillin, Elsa; Fang, Hong; Mohammed, Bassem M; Hegazy, Lamees; Burris, Thomas P; Elgendy, Bahaa

Cold exposure induces the constitutively active thermogenic receptor, GPR3, via ERRα and ERRγ.

寒冷暴露通过 ERRα 和 ERRγ 诱导组成型活性产热受体 GPR3。

Sveidahl Johansen Olivia, McIntyre Rebecca L, Rahbani Janane F, Zhang Qiaoqiao, Scholtes Charlotte, Lagarde Damien Marc, Billon Cyrielle, Côté Isabelle, Delgado-Martin Maria, Tandio David, Basse Astrid Linde, Eury Elodie, Kralli Anastasia, Burris Thomas P, Giguère Vincent, Kazak Lawrence, Gerhart-Hines Zachary

STL1267 inhibits myofibroblast differentiation in a TGFβ1-driven human lung fibroblast model.

STL1267 在 TGFβ1 驱动的人类肺成纤维细胞模型中抑制肌成纤维细胞分化。

Prasad Chandrashekhar, Huang Steven K, Burris Thomas P, Sundar Isaac Kirubakaran

Limited effects of the REV-ERB agonist SR9009 after mouse spinal cord contusion: Reduced acute pathology with unaffected functional recovery and chronic white matter loss

REV-ERB激动剂SR9009对小鼠脊髓挫伤的影响有限:减轻急性病理损伤,功能恢复不受影响,但慢性白质丢失也未受影响。

Slomnicki, Lukasz P; Hodges, Emily; Armstrong, Christine; Morehouse, Johnny; Burke, Darlene; Ohri, Sujata Saraswat; Burris, Thomas P; Hetman, Michal

From Functional Fatty Acids to Potent and Selective Natural-Product-Inspired Mimetics via Conformational Profiling

从功能性脂肪酸到高效选择性天然产物仿生化合物的构象分析

Markham, Lauren E; Koelblen, Thomas; Chobanian, Harry R; Follis, Ariele Viacava; Burris, Thomas P; Micalizio, Glenn C

Merging Natural Product Structures with Pharmaceutical Leads: Unnatural Enantiomers of Estranes as Glucocorticoid Receptor Modulators That Suppress TNF-α and IL-6 Release

将天然产物结构与先导化合物相结合:雌烷的非天然对映异构体作为糖皮质激素受体调节剂,可抑制TNF-α和IL-6的释放

Nicholson, Joshua M; Yang, Dexi; Koelblen, Thomas; Hu, Eric L; Coss, Christopher C; Burris, Thomas P; Hu, Xiao; Micalizio, Glenn C

A Synthetic ERR Agonist Alleviates Metabolic Syndrome

合成的ERR激动剂可缓解代谢综合征

Billon, Cyrielle; Schoepke, Emmalie; Avdagic, Amer; Chatterjee, Arindam; Butler, Andrew A; Elgendy, Bahaa; Walker, John K; Burris, Thomas P

The Estrogen Receptor-Related Orphan Receptors Regulate Autophagy through TFEB.

雌激素受体相关孤儿受体通过 TFEB 调节自噬

Losby McKenna, Hayes Matthew, Valfort Aurore, Sopariwala Danesh H, Sanders Ryan, Walker John K, Xu Weiyi, Narkar Vihang A, Zhang Lilei, Billon Cyrielle, Burris Thomas P

International Union of Basic and Clinical Pharmacology CXIII: Nuclear Receptor Superfamily-Update 2023

国际基础与临床药理学联合会第113届会议:核受体超家族——2023年最新进展

Burris, Thomas P; de Vera, Ian Mitchelle S; Cote, Isabelle; Flaveny, Colin A; Wanninayake, Udayanga S; Chatterjee, Arindam; Walker, John K; Steinauer, Nickolas; Zhang, Jinsong; Coons, Laurel A; Korach, Kenneth S; Cain, Derek W; Hollenberg, Anthony N; Webb, Paul; Forrest, Douglas; Jetten, Anton M; Edwards, Dean P; Grimm, Sandra L; Hartig, Sean; Lange, Carol A; Richer, Jennifer K; Sartorius, Carol A; Tetel, Marc; Billon, Cyrielle; Elgendy, Bahaa; Hegazy, Lamees; Griffett, Kristine; Peinetti, Nahuel; Burnstein, Kerry L; Hughes, Travis S; Sitaula, Sadichha; Stayrook, Keitch R; Culver, Alexander; Murray, Meghan H; Finck, Brian N; Cidlowski, John A

Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915

开发和药理学评价一系列新型强效泛ERR激动剂,并鉴定出SLU-PP-915

Hampton, Carissa S; Sitaula, Sadichha; Billon, Cyrielle; Haynes, Keith; Avdagic, Amer; Wanninayake, Udayanga; Adeyemi, Christiana M; Chatterjee, Arindam; Griffett, Kristine; Banerjee, Subhashis; Burris, Sheryl L; Schoepke, Emmalie; Boehm, Terri; Bess, Alex; de Vera, Ian Mitchelle S; Burris, Thomas P; Walker, John K