日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identifying a next-generation antimalarial trioxolane in a landscape of artemisinin partial resistance

在青蒿素部分耐药性的背景下,寻找下一代抗疟疾三氧杂环戊烷类药物。

Klope, Matthew T; Talukder, Poulami; Blank, Brian R; Chelebieva, Sevil; Chen, Jun; Fontaine, Shaun D; Gonciarz, Ryan L; Jaishankar, Priyadarshini; Lee, Grace J; Legac, Jennifer; Mathur, Vineet; Narayan, Avani; Okitwi, Martin; Orena, Stephen; Settineri, Nicholas S; Tapia, Juan A; Taremwa, Yoweri; Tumwebaze, Patrick K; Vinod, Aswathy; Burrows, Jeremy N; Rosenthal, Philip J; Cooper, Roland A; Renslo, Adam R

Characterizing the quick-killing mechanism of action of azithromycin analogs against malaria parasites

阐明阿奇霉素类似物对疟原虫的快速杀灭机制

Mao, Emma Y; Nguyen, William; Jana, Gouranga P; Maity, Bikash C; Pazicky, Samuel; Giannangelo, Carlo; Reader, Janette; Famodimu, Mufuliat T; Birkholtz, Lyn-Marie; Delves, Michael J; Creek, Darren J; Bozdech, Zbynek; Laleu, Benoît; Burrows, Jeremy N; Sleebs, Brad E; Gancheva, Maria R; Wilson, Danny W

Screening of Medicines for Malaria Venture Open Boxes Identifies Potent SARS-CoV‑2 Papain-like Protease (PL(pro)) Inhibitors

疟疾药物筛选项目“开放盒子”发现了强效的SARS-CoV-2木瓜蛋白酶样蛋白酶(PL(pro))抑制剂

Gawriljuk, Victor Oliveira; Noske, Gabriela Dias; Fernandes, Rafaela Sachetto; Nakamura, Aline Minalli; Freire, Marjorie C L C; Godoy, Mariana Ortiz; Bonatto, Vinicius; Chelucci, Rafael; Andricopulo, Adriano; Bakowski, Malina A; Wolff, Karen C; Riva, Laura; Burrows, Jeremy N; Wells, Timothy N C; Laleu, Benoît; Martins, Ronaldo; Souza, Juliano Paula; Arruda, Eurico; Samby, Kirandeep; Laskar, Sujay; Guido, Rafael Victorio Carvalho; Oliva, Glaucius; Godoy, Andre Schutzer

Inhibitors of malaria parasite cyclic nucleotide phosphodiesterases block asexual blood-stage development and mosquito transmission.

疟原虫环核苷酸磷酸二酯酶抑制剂可阻断无性血液期发育和蚊子传播

Gomez-Gonzalez Paula-Josefina, Gupta Antima, Drought Laura G, Patel Avnish, Okombo John, van der Watt Mariëtte, Walker-Gray Ryan, Schindler Kyra A, Burkhard Anna Y, Yeo Tomas, Narwal Sunil K, Bloxham Talia S, Flueck Christian, Walker Eloise M, Rey Joshua A, Fairhurst Kate J, Reader Janette, Park Heekuk, Pollard Harry G, Stewart Lindsay B, Brandner-Garrod Luke, Kristan Mojca, Sterk Geert-Jan, van Nuland Youri M, Manko Emilia, van Schalkwyk Donelly A, Zheng Yang, Leurs Rob, Dechering Koen J, Aguiar Anna Caroline C, Guido Rafael V C, Pereira Dhelio B, Tumwebaze Patrick K, Nosbya Samuel L, Rosenthal Philip J, Cooper Roland A, Palmer Mike, Parkinson Tanya, Burrows Jeremy N, Uhlemann Anne-Catrin, Birkholtz Lyn-Marié, Small-Saunders Jennifer L, Duffy James, Fidock David A, Brown Alan, Gardner Mark, Baker David A

Optimization of diastereomeric dihydropyridines as antimalarials

优化非对映异构二氢吡啶类化合物作为抗疟药

Van Horn, Kurt S; Zhao, Yingzhao; Parvatkar, Prakash T; Maier, Julie; Mutka, Tina; Lacrue, Alexis; Brockmeier, Fabian; Ebert, Daniel; Wu, Wesley; Casandra, Debora R; Namelikonda, Niranjan; Yacoub, Jeanine; Sigal, Martina; Knapp, Spencer; Floyd, David; Waterson, David; Burrows, Jeremy N; Duffy, James; DeRisi, Joseph L; Kyle, Dennis E; Guy, R Kiplin; Manetsch, Roman

Protein target similarity is positive predictor of in vitro antipathogenic activity: a drug repurposing strategy for Plasmodium falciparum

蛋白质靶标相似性是体外抗病原体活性的正向预测因子:恶性疟原虫药物再利用策略

Mogire, Reagan M; Miruka, Silviane A; Juma, Dennis W; McNamara, Case W; Andagalu, Ben; Burrows, Jeremy N; Chenu, Elodie; Duffy, James; Ogutu, Bernhards R; Akala, Hoseah M

Oxidative stress changes the effectiveness of artemisinin in Plasmodium falciparum

氧化应激会改变青蒿素对恶性疟原虫的疗效

Pires, Camilla Valente; Cassandra, Debora; Xu, Shulin; Laleu, Benoit; Burrows, Jeremy N; Adams, John H

Global Health Priority Box─Proactive Pandemic Preparedness

全球卫生优先事项栏目——主动应对大流行病

Adam, Anna; Besson, Dominique; Bryant, Rob; Rees, Sarah; Willis, Paul A; Burrows, Jeremy N; Hooft van Huisjduijnen, Rob; Laleu, Benoît; Norton, Larry; Canan, Stacie; Hawryluk, Natalie; Robinson, Dale; Palmer, Mike; Samby, Kirandeep Kaur

Combating antimicrobial resistance in malaria, HIV and tuberculosis

对抗疟疾、艾滋病和结核病中的抗菌素耐药性

Duffey, Maëlle; Shafer, Robert W; Timm, Juliano; Burrows, Jeremy N; Fotouhi, Nader; Cockett, Mark; Leroy, Didier

Antimalarial drug discovery: progress and approaches

抗疟药物研发:进展与方法

Siqueira-Neto, Jair L; Wicht, Kathryn J; Chibale, Kelly; Burrows, Jeremy N; Fidock, David A; Winzeler, Elizabeth A