日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An AKR1C3-activated kinase inhibitor prodrug.

AKR1C3激活激酶抑制剂前药。

Li Zhengnian, Martinez Michael, Byun Woong Sub, Thathireddy Anuradha, Qiu Tian, Wang Yaning, Katzengruber Leon, Chouldjian Ani, Lu Wenchao, Ji Wenzhi, Che Jianwei, Zhang Tinghu, Hinshaw Stephen M, Gray Nathanael S

Rational Design of CDK12/13 and BRD4 Molecular Glue Degraders

CDK12/13 和 BRD4 分子胶降解剂的合理设计

Zhuang, Zhe; Byun, Woong Sub; Kozicka, Zuzanna; Donovan, Katherine A; Dwyer, Brendan G; Thornhill, Abby M; Jones, Hannah M; Jiang, Zixuan; Zhu, Xijun; Fischer, Eric S; Thomä, Nicolas H; Gray, Nathanael S

Development of Potent and Selective CK1α Molecular Glue Degraders.

高效选择性CK1α分子胶降解剂的开发。

Geng Qixiang, Jiang Zixuan, Byun Woong Sub, Donovan Katherine A, Zhuang Zhe, Jiang Fen, Jones Hannah M, Razumkov Hlib, Tang Michelle T, Sarott Roman C, Fischer Eric S, Corsello Steven M, Hinshaw Stephen M, Gray Nathanael S

Development of Degraders and 2-pyridinecarboxyaldehyde (2-PCA) as a recruitment Ligand for FBXO22.

开发降解剂和 2-吡啶甲醛 (2-PCA) 作为 FBXO22 的募集配体

Qiu Tian, Zhuang Zhe, Byun Woong Sub, Kozicka Zuzanna, Baek Kheewoong, Zhong Jianing, Thornhill Abby M, Ryan Julia K, Donovan Katherine A, Fischer Eric S, Ebert Benjamin L, Gray Nathanael S

Discovery of CRBN-Dependent WEE1 Molecular Glue Degraders from a Multicomponent Combinatorial Library

从多组分组合库中发现 CRBN 依赖性 WEE1 分子胶降解剂

Razumkov, Hlib; Jiang, Zixuan; Baek, Kheewoong; You, Inchul; Geng, Qixiang; Donovan, Katherine A; Tang, Michelle T; Metivier, Rebecca J; Mageed, Nada; Seo, Pooreum; Li, Zhengnian; Byun, Woong Sub; Hinshaw, Stephen M; Sarott, Roman C; Fischer, Eric S; Gray, Nathanael S

Exploration of the tunability of BRD4 degradation by DCAF16 trans-labelling covalent glues

利用DCAF16反式标记共价胶探索BRD4降解的可调控性

Hassan, Muhammad Murtaza; Li, Yen-Der; Ma, Michelle W; Teng, Mingxing; Byun, Woong Sub; Puvar, Kedar; Lumpkin, Ryan; Sandoval, Brittany; Rutter, Justine C; Jin, Cyrus Y; Wang, Michelle Y; Xu, Shawn; Schmoker, Anna M; Cheong, Hakyung; Groendyke, Brian J; Qi, Jun; Fischer, Eric S; Ebert, Benjamin L; Gray, Nathanael S

Discovery of bivalent small molecule degraders of cyclin-dependent kinase 7 (CDK7).

发现细胞周期蛋白依赖性激酶 7 (CDK7) 的二价小分子降解剂

Ji Wenzhi, Du Guangyan, Jiang Jie, Lu Wenchao, Mills Caitlin E, Yuan Linjie, Jiang Fen, He Zhixiang, Bradshaw Gary A, Chung Mirra, Jiang Zixuan, Byun Woong Sub, Hinshaw Stephen M, Zhang Tinghu, Gray Nathanael S

Activating p53(Y220C) with a Mutant-Specific Small Molecule.

用突变体特异性小分子激活p53(Y220C)

Zhu Xijun, Byun Woong Sub, Pieńkowska Dominika Ewa, Nguyen Kha The, Gerhartz Jan, Geng Qixiang, Qiu Tian, Zhong Jianing, Jiang Zixuan, Wang Mengxiong, Sarott Roman C, Hinshaw Stephen M, Zhang Tinghu, Attardi Laura D, Nowak Radosław P, Gray Nathanael S

Proteomics-Based Discovery of First-in-Class Chemical Probes for Programmed Cell Death Protein 2 (PDCD2)

基于蛋白质组学的程序性细胞死亡蛋白2 (PDCD2) 首创化学探针的发现

Ji, Wenzhi; Byun, Woong Sub; Lu, Wenchao; Zhu, Xijun; Donovan, Katherine A; Dwyer, Brendan G; Che, Jianwei; Yuan, Linjie; Abulaiti, Xianmixinuer; Corsello, Steven M; Fischer, Eric S; Zhang, Tinghu; Gray, Nathanael S

Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A(2A)/A(3) Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity.

截短的 2,8-二取代腺苷衍生物作为双重 A(2A)/A(3) 腺苷受体拮抗剂的构效关系及其癌症免疫治疗活性

Kim Gibae, Hou Xiyan, Byun Woong Sub, Kim Gyudong, Jarhad Dnyandev B, Lee Grim, Hyun Young Eum, Yu Jinha, Lee Chang Soo, Qu Shuhao, Warnick Eugene, Gao Zhan-Guo, Kim Ji Yong, Ji Seunghee, Shin Hyunwoo, Choi Jong-Ryoul, Jacobson Kenneth A, Lee Hyuk Woo, Lee Sang Kook, Jeong Lak Shin