日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Building Confidence in Physiologically Based Pharmacokinetic Modeling of CYP3A Induction Mediated by Rifampin: An Industry Perspective

建立对利福平介导的CYP3A诱导的生理药代动力学模型的信心:行业视角

Reddy, Micaela B; Cabalu, Tamara D; de Zwart, Loeckie; Ramsden, Diane; Dowty, Martin E; Taskar, Kunal S; Badée, Justine; Bolleddula, Jayaprakasam; Boulu, Laurent; Fu, Qiang; Kotsuma, Masakatsu; Leblanc, Alix F; Lewis, Gareth; Liang, Guiqing; Parrott, Neil; Pilla Reddy, Venkatesh; Prakash, Chandra; Shah, Kushal; Umehara, Kenichi; Mukherjee, Dwaipayan; Rehmel, Jessica; Hariparsad, Niresh

Application of a Rat Liver Drug Bioactivation Transcriptional Response Assay Early in Drug Development That Informs Chemically Reactive Metabolite Formation and Potential for Drug-induced Liver Injury

在药物研发早期应用大鼠肝脏药物生物活化转录反应分析,以了解化学活性代谢物的形成和药物引起肝损伤的可能性

Monroe, James J; Tanis, Keith Q; Podtelezhnikov, Alexei A; Nguyen, Truyen; Machotka, Sam V; Lynch, Donna; Evers, Raymond; Palamanda, Jairam; Miller, Randy R; Pippert, Todd; Cabalu, Tamara D; Johnson, Timothy E; Aslamkhan, Amy G; Kang, Wen; Tamburino, Alex M; Mitra, Kaushik; Agrawal, Nancy G B; Sistare, Frank D

Application of Physiologically Based Pharmacokinetic Modeling to Predict Pharmacokinetics in Healthy Japanese Subjects

应用生理药代动力学模型预测健康日本受试者的药代动力学

Matsumoto, Yuki; Cabalu, Tamara; Sandhu, Punam; Hartmann, Georgy; Iwasa, Takashi; Yoshitsugu, Hiroyuki; Gibson, Christopher; Uemura, Naoto

Recommendations for the Design of Clinical Drug-Drug Interaction Studies With Itraconazole Using a Mechanistic Physiologically-Based Pharmacokinetic Model

基于机制生理药代动力学模型的伊曲康唑临床药物相互作用研究设计建议

Chen, Yuan; Cabalu, Tamara D; Callegari, Ernesto; Einolf, Heidi; Liu, Lichuan; Parrott, Neil; Peters, Sheila Annie; Schuck, Edgar; Sharma, Pradeep; Tracey, Helen; Upreti, Vijay V; Zheng, Ming; Zhu, Andy Z X; Hall, Stephen D

Drug-drug interaction studies: regulatory guidance and an industry perspective

药物相互作用研究:监管指导和行业视角

Prueksaritanont, Thomayant; Chu, Xiaoyan; Gibson, Christopher; Cui, Donghui; Yee, Ka Lai; Ballard, Jeanine; Cabalu, Tamara; Hochman, Jerome