Discovery of Pyridopyrimidinones that Selectively Inhibit the H1047R PI3Kα Mutant Protein
发现能选择性抑制H1047R PI3Kα突变蛋白的吡啶并嘧啶酮类化合物
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c00078
Ketcham, John M; Harwood, Stephen J; Aranda, Ruth; Aloiau, Athenea N; Bobek, Briana M; Briere, David M; Burns, Aaron C; Caddell Haatveit, Kersti; Calinisan, Andrew; Clarine, Jeffery; Elliott, Adam; Engstrom, Lars D; Gunn, Robin J; Ivetac, Anthony; Jones, Benjamin; Kuehler, Jon; Lawson, J David; Nguyen, Natalie; Parker, Cody; Pearson, Kelly E; Rahbaek, Lisa; Saechao, Barbara; Wang, Xiaolun; Waters, Anna; Waters, Laura; Watkins, Ashlee H; Olson, Peter; Smith, Christopher R; Christensen, James G; Marx, Matthew A