日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules

胖还是扁?偶极矩矢量对芳香标签与大分子间非共价相互作用的影响

Holub, Josef; Jílková, Adéla; Lemke, Carina; Cianni, Lorenzo; Spiwoková, Petra; Horn, Martin; Breuer, Christian; Leontovyč, Adrian; Brynda, Jiří; Mertlíková-Kaiserová, Helena; Chanová, Marta; Dos Reis Rocho, Fernanda; Montanari, Carlos A; El-Sakkary, Nelly; Caffrey, Conor R; Gütschow, Michael; Hnyk, Drahomír; Mareš, Michael; Fanfrlík, Jindřich

Discovery of benzyl carbamate inhibitors of coronavirus M(pro) enzymes from a legacy collection of cysteine protease inhibitors

从一系列已知的半胱氨酸蛋白酶抑制剂中发现冠状病毒M(pro)酶的苄基氨基甲酸酯抑制剂

Sá Magalhães Serafim, Mateus; Kronenberger, Thales; Francisco, Karol R; de Sousa Reis, Erik Vinicius; Gonçalves de Oliveira, Ellen; Marcelino E Oliveira, Fernanda Kelly; Serraglio Fortes, Isadora; Maciel Fernandes, Thaís Helena; Barbosa da Silva, Elany; Fajtova, Pavla; Skinner, Danielle E; Syed, Rafay O; Lage de Siqueira-Neto, Jair; Poso, Antti; Fernandes Mota, Bruno Eduardo; Alves Coelho-Dos-Reis, Jordana Grazziela; Santos Abrahão, Jônatas; Gonçalves Maltarollo, Vinícius; O'Donoghue, Anthony J; Caffrey, Conor R

Enhancing schistosomiasis drug discovery approaches with optimized proteasome substrates.

利用优化的蛋白酶体底物增强血吸虫病药物发现方法

Silva Elany B, Jiang Zhenze, Liu Chenxi, Fajtová Pavla, Teixeira Thaiz R, de Castro Fiorini Maia Giovana, Liu Lawrence J, El-Sakkary Nelly, Skinner Danielle E, Syed Ali, Wang Steven C, Caffrey Conor R, O'Donoghue Anthony J

Chalcogen Derivatives for the Treatment of African Trypanosomiasis: Biological Evaluation of Thio- and Seleno-Semicarbazones and Their Azole Derivatives.

硫族元素衍生物治疗非洲锥虫病:硫代和硒代氨基脲及其唑类衍生物的生物学评价

Rubio-Hernández Mercedes, Teixeira Thaiz R, Nguyen Tina P, Shingyoji Mai, da Silva Elany Barbosa, O'Donoghue Anthony J, Caffrey Conor R, Pérez-Silanes Silvia, Martínez-Sáez Nuria

Nitroquinolones and nitroquinolines: syntheses and antitrypanosomal activity

硝基喹诺酮类和硝基喹啉类:合成及抗锥虫活性

Dube, Phelelisiwe S; Francisco, Karol R; Legoabe, Lesetja J; Sun, Yujie Uli; Kaur, Yashpreet; Nguyen, Tina P; Caffrey, Conor R; Beteck, Richard M

Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents

鉴定取代的4-氨基喹啉类化合物作为广谱抗寄生虫药物

Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A; Hoffman, Benjamin; Bernatchez, Jean A; McCall, Laura-Isobel; Calvet, Claudia M; Ackermann, Jasmin; Souza, Julia M; Thomas, Diane; Millard, Caroline C; Devine, William G; Singh, Baljinder; Silva, Everton M; Leed, Susan E; Roncal, Norma E; Penn, Erica C; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J; Campbell, Robert F; Momper, Jeremiah D; McKerrow, James H; Caffrey, Conor R; Siqueira-Neto, Jair L; Pollastri, Michael P; Mensa-Wilmot, Kojo; Ferrins, Lori

Aza-peptide aldehydes and ketones: synthesis and evaluation as human 20S proteasome inhibitors

氮杂肽醛和酮:合成及作为人20S蛋白酶体抑制剂的评价

Corrigan, Thomas S; Border, Sarah E; Lotti Diaz, Leilani M; Kasper, Kayla Q; Noonchester, Abigail M; Amer, Rasmiah; Kucway, Kayla S; Fleisher, Michael; Fernandez, Joseph P; Lovins, Alex R; Serrano, Ana K; Caffrey, Conor R; O'Donoghue, Anthony J; Benson, Don M Jr; Hadad, Christopher M; Ekici, Özlem Doğan

Discovery of small molecules with anthelmintic potential in the Medicines for Malaria Venture's COVID and Global Health Priority Boxes using an infrared-based assay for Caenorhabditis elegans motility

利用基于红外光谱的秀丽隐杆线虫运动性检测方法,在疟疾药物研发联盟的COVID-19和全球健康优先项目箱中发现具有抗蠕虫潜力的分子。

Sun, Yujie Uli; Liu, Lawrence J; Caffrey, Conor R

Photoaffinity labeling of protein targets in a complex metazoan: proof-of-concept using a probe for Schistosoma mansoni tubulin

利用光亲和标记技术对复杂后生动物中的蛋白质靶标进行标记:以曼氏血吸虫微管蛋白探针为例的概念验证

Lucero, Bobby; Alle, Thibault; Bufano, Marianna; Yao, Yuemang; Brunden, Kurt R; Brancale, Andrea; Ballatore, Carlo; Francisco, Karol R; Caffrey, Conor R

Structure-Activity Relationship and Target Investigation of Thiophen-2-yl-Pyrimidines against Schistosoma species

噻吩-2-基嘧啶类化合物对血吸虫的构效关系及靶点研究

Francisco, Karol R; Lucero, Bobby; Yohannan, Darius; Varricchio, Carmine; Lam, Anny; Sebastiani, Jessica; Liu, Lawrence J; Sun, Yujie Uli; Jacinto, Jorge; Renzulli, Michele; Monti, Ludovica; Brancale, Andrea; Ballatore, Carlo; Alle, Thibault; Caffrey, Conor R