CYX-5, a G-protein biassed MOP receptor agonist, DOP receptor antagonist and KOP receptor agonist, evokes constipation but not respiratory depression relative to morphine in rats
CYX-5 是一种 G 蛋白偏向性 MOP 受体激动剂、DOP 受体拮抗剂和 KOP 受体激动剂,与吗啡相比,它能引起大鼠便秘,但不会引起呼吸抑制。
期刊:Pharmacological Reports
影响因子:3.8
doi:10.1007/s43440-023-00446-8
Imam, Mohammad Zafar; Kuo, Andy; Ghassabian, Sussan; Cai, Yunxin; Qin, Yajuan; Li, Tingyou; Smith, Maree T