日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule targeting Na V 1.7 via inhibition of CRMP2-Ubc9 interaction reduces pain-related outcomes in a rodent osteoarthritic model.

通过抑制 CRMP2-Ubc9 相互作用靶向 Na V 1.7 的小分子可减轻啮齿动物骨关节炎模型中的疼痛相关结果

Hestehave Sara, Allen Heather N, Gomez Kimberly, Duran Paz, Calderon-Rivera Aida, Loya-López Santiago, Rodríguez-Palma Erick J, Khanna Rajesh

Quinoline-Based Neuropilin‑1 Antagonists Exhibit a Pure Antagonist Profile and Block Vascular Endothelial Growth Factor-Induced Pain

基于喹啉的神经纤毛蛋白-1拮抗剂表现出纯拮抗剂特性,并能阻断血管内皮生长因子诱导的疼痛。

Hestehave, Sara; Dragoni, Silvia; Fallon, Philip; Mota, Filipa; Calderon-Rivera, Aida; Gomez, Kimberly; Powell, Jonathan; Patsiarika, Anastasia; Reisinger, Tifelle; Crosby, Stuart; Chan, A W Edith; Steadman, David; Winfield, Natalie; Jarvis, Ashley; Martin, John; Zachary, Ian C; Frankel, Paul; Djordjevic, Snezana; Ruhrberg, Christiana; Khanna, Rajesh; Selwood, David L

Targeting Na(v)1.7 and Na(v)1.8 with a PIKfyve inhibitor to reverse inflammatory and neuropathic pain.

使用 PIKfyve 抑制剂靶向 Na(v)1.7 和 Na(v)1.8 来逆转炎症性和神经性疼痛

Rodríguez-Palma Erick J, Loya-Lopez Santiago, Min Sophia M, Calderon-Rivera Aida, Gomez Kimberly, Khanna Rajesh, Axtman Alison D

Enabling wider access to human molecular neuroscience research in pain: A simple preservation method for human dorsal root ganglion neurons in Hibernate A media.

使人类疼痛分子神经科学研究能够更广泛地进行:一种在 Hibernate A 培养基中保存人类背根神经节神经元的简单方法。

Lesnak Joseph B, Schaub Mandee K, Gomez Kimberly, Calderon-Rivera Aida, Loya-Lopez Santiago, Stewart Robert, Jo Sooyeon, Fujita Akie, Osorno Tomás, Desai Marisa, Natarajan Keerthana, Schackmuth Morgan K, Moreno Marisol Mancilla, Shiers Stephanie I, Cervantes Anna, Funk Geoffrey, Horton Peter, Vines Erin, Yousuf Muhammad Saad, Sadler Katelyn E, Bean Bruce P, Khanna Rajesh, Dussor Gregory, Price Theodore J

Neuropilin-1 inhibition suppresses nerve growth factor signaling and nociception in pain models

神经纤毛蛋白-1抑制剂可抑制疼痛模型中的神经生长因子信号传导和伤害感受。

Peach, Chloe J; Tonello, Raquel; Damo, Elisa; Gomez, Kimberly; Calderon-Rivera, Aida; Bruni, Renato; Bansia, Harsh; Maile, Laura; Manu, Ana-Maria; Hahn, Hyunggu; Thomsen, Alex Rb; Schmidt, Brian L; Davidson, Steve; des Georges, Amedee; Khanna, Rajesh; Bunnett, Nigel W

C2230, a preferential use- and state-dependent CaV2.2 channel blocker, mitigates pain behaviors across multiple pain models.

C2230 是一种优先使用和状态依赖的 CaV2.2 通道阻滞剂,可减轻多种疼痛模型中的疼痛行为

Tang Cheng, Gomez Kimberly, Chen Yan, Allen Heather N, Hestehave Sara, Rodríguez-Palma Erick J, Loya-Lopez Santiago, Calderon-Rivera Aida, Duran Paz, Nelson Tyler S, Kanumuri Siva Rama Raju, Shah Bijal, Panigrahi Nihar R, Perez-Miller Samantha, Schackmuth Morgan K, Ruparel Shivani, Patwardhan Amol, Price Theodore J, Arora Paramjit S, Sharma Ravindra K, Sharma Abhisheak, Yu Jie, Korczeniewska Olga A, Khanna Rajesh

Effect of Crude Extract from the Sea Anemone Bunodeopsis globulifera on Voltage-Gated Ion Channels from Central and Peripheral Murine Nervous Systems.

海葵 Bunodeopsis globulifera 粗提物对小鼠中枢和外周神经系统电压门控离子通道的影响

Flores-Pérez Aleida Jeannette, Loya-López Santiago, Ávalos-Fuentes Arturo, Calderon-Rivera Aida, Damo Elisa, Lazcano-Pérez Fernando, Khanna Rajesh, Florán-Garduño Benjamin, Sánchez-Rodríguez Judith

Regulating neuronal excitability: The role of S-palmitoylation in Na(V)1.7 activity and voltage sensitivity

调节神经元兴奋性:S-棕榈酰化在Na(V)1.7活性和电压敏感性中的作用

Tang, Cheng; Duran, Paz; Calderon-Rivera, Aida; Loya-Lopez, Santiago; Gomez, Kimberly; Perez-Miller, Samantha; Khanna, Rajesh

A peptidomimetic modulator of the Ca(V)2.2 N-type calcium channel for chronic pain

一种用于治疗慢性疼痛的 Ca(V)2.2 N 型钙通道的肽模拟调节剂

Gomez, Kimberly; Santiago, Ulises; Nelson, Tyler S; Allen, Heather N; Calderon-Rivera, Aida; Hestehave, Sara; Rodríguez Palma, Erick J; Zhou, Yuan; Duran, Paz; Loya-Lopez, Santiago; Zhu, Elaine; Kumar, Upasana; Shields, Rory; Koseli, Eda; McKiver, Bryan; Giuvelis, Denise; Zuo, Wanhong; Inyang, Kufreobong E; Dorame, Angie; Chefdeville, Aude; Ran, Dongzhi; Perez-Miller, Samantha; Lu, Yi; Liu, Xia; Handoko; Arora, Paramjit S; Patek, Marcel; Moutal, Aubin; Khanna, May; Hu, Huijuan; Laumet, Geoffroy; King, Tamara; Wang, Jing; Damaj, M Imad; Korczeniewska, Olga A; Camacho, Carlos J; Khanna, Rajesh

Identification and targeting of a unique Na(V)1.7 domain driving chronic pain

识别并靶向驱动慢性疼痛的独特Na(V)1.7结构域

Gomez, Kimberly; Stratton, Harrison J; Duran, Paz; Loya, Santiago; Tang, Cheng; Calderon-Rivera, Aida; François-Moutal, Liberty; Khanna, May; Madura, Cynthia L; Luo, Shizhen; McKiver, Bryan; Choi, Edward; Ran, Dongzhi; Boinon, Lisa; Perez-Miller, Samantha; Damaj, M Imad; Moutal, Aubin; Khanna, Rajesh