Design, Synthesis and Biological Evaluation of 2-Phenyl Indole Analogues of OXi8006 as Colchicine Site Inhibitors of Tubulin Polymerization and Vascular Disrupting Agents
OXi8006 的 2-苯基吲哚类似物作为秋水仙碱位点抑制剂抑制微管蛋白聚合和血管破坏剂的设计、合成和生物学评价
期刊:Bioorganic & Medicinal Chemistry
影响因子:3
doi:10.1016/j.bmc.2024.117981
Vairin, Rebecca; Tamminga, Caleb; Shi, Zhe; Borchardt, Christian; Jambulapati, Jayaram; Bai, Ruoli; Wanniarachchi, Hashini; Bueno, Lorena; Hamel, Ernest; Mason, Ralph P; Trawick, Mary Lynn; Pinney, Kevin G