日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pyrimidine Azepine Targets the Plasmodium bc 1 Complex and Displays Multistage Antimalarial Activity

嘧啶氮杂卓靶向疟原虫 bc 1 复合物并显示多级抗疟活性

Juliana Calit, Surendra K Prajapati, Ernest D Benavente, Jessica E Araújo, Bingbing Deng, Kazutoyo Miura, Yasmin Annunciato, Igor M R Moura, Miho Usui, Jansen F Medeiros, Carolina H Andrade, Sabrina Silva-Mendonça, Anton Simeonov, Richard T Eastman, Carole A Long, Maisa da Silva Araujo, Kim C Willia

A novel 4-aminoquinoline chemotype with multistage antimalarial activity and lack of cross-resistance with PfCRT and PfMDR1 mutants

一种新型的4-氨基喹啉化学类型,具有多阶段抗疟活性,且与PfCRT和PfMDR1突变体无交叉耐药性。

Ferreira, Letícia Tiburcio; Cassiano, Gustavo Capatti; Alvarez, Luis Carlos Salazar; Okombo, John; Calit, Juliana; Fontinha, Diana; Gil-Iturbe, Eva; Coyle, Rachael; Andrade, Carolina Horta; Sunnerhagen, Per; Bargieri, Daniel Youssef; Prudêncio, Miguel; Quick, Matthias; Cravo, Pedro V; Lee, Marcus C S; Fidock, David A; Costa, Fabio Trindade Maranhão

Innovative Multistage ML-QSAR Models for Malaria: From Data to Discovery

疟疾创新型多阶段机器学习-定量构效关系模型:从数据到发现

Borba, Joyce V B; Salazar-Alvarez, Luis Carlos; Ferreira, Letícia Tiburcio; Silva-Mendonça, Sabrina; Silva, Meryck Felipe Brito da; Sanches, Igor H; Clementino, Leandro da Costa; Magalhães, Marcela Lucas; Rimoldi, Aline; Calit, Juliana; Santana, Sofia; Prudêncio, Miguel; Cravo, Pedro V; Bargieri, Daniel Y; Cassiano, Gustavo C; Costa, Fabio T M; Andrade, Carolina Horta

Characterisation of the merozoite thrombospondin related anonymous protein (MTRAP) of Plasmodium berghei as a transmission-blocking antigen

伯氏疟原虫裂殖子血小板反应蛋白相关匿名蛋白(MTRAP)作为一种阻断传播抗原的特性鉴定

Gaitán, Xiomara Alexandra; Calit, Juliana; Dobrescu, Irina; Ramos, Marisé Solórzano; Gimenez, Alba Marina; Bargieri, Daniel Youssef

Novel Transmission-Blocking Antimalarials Identified by High-Throughput Screening of Plasmodium berghei Ookluc

通过伯氏疟原虫的高通量筛选鉴定出新型阻断传播的抗疟药

Juliana Calit, Jessica E Araújo, Bingbing Deng, Kazutoyo Miura, Xiomara A Gaitán, Maisa da Silva Araújo, Jansen F Medeiros, Carole A Long, Anton Simeonov, Richard T Eastman, Daniel Y Bargieri

Computational Chemogenomics Drug Repositioning Strategy Enables the Discovery of Epirubicin as a New Repurposed Hit for Plasmodium falciparum and P. vivax

计算化学基因组学药物重定位策略促成了表柔比星作为一种新的可用于治疗恶性疟原虫和间日疟原虫的先导化合物的发现

Ferreira, Letícia Tiburcio; Rodrigues, Juliana; Cassiano, Gustavo Capatti; Tavella, Tatyana Almeida; Tomaz, Kaira Cristina Peralis; Baia-da-Silva, Djane Clarys; Souza, Macejane Ferreira; Lima, Marilia Nunes do Nascimento; Mottin, Melina; Almeida, Ludimila Dias; Calit, Juliana; Puça, Maria Carolina Silva de Barros; Melo, Gisely Cardoso; Bargieri, Daniel Youssef; Lopes, Stefanie Costa Pinto; Lacerda, Marcus Vinicius Guimarães; Bilsland, Elizabeth; Sunnerhagen, Per; Neves, Bruno Junior; Andrade, Carolina Horta; Cravo, Pedro Vitor Lemos; Costa, Fabio Trindade Maranhão

Correction for Ferreira et al., "Computational Chemogenomics Drug Repositioning Strategy Enables the Discovery of Epirubicin as a New Repurposed Hit for Plasmodium falciparum and P. vivax"

对 Ferreira 等人的论文“计算化学基因组学药物重定位策略促成了表柔比星作为恶性疟原虫和间日疟原虫新用途先导化合物的发现”的更正

Ferreira, Letícia Tiburcio; Rodrigues, Juliana; Cassiano, Gustavo Capatti; Tavella, Tatyana Almeida; Tomaz, Kaira Cristina Peralis; Baia-da-Silva, Djane Clarys; Souza, Macejane Ferreira; Lima, Marilia Nunes do Nascimento; Mottin, Melina; Almeida, Ludimila Dias; Calit, Juliana; Puça, Maria Carolina Silva de Barros; Melo, Gisely Cardoso; Bargieri, Daniel Youssef; Lopes, Stefanie Costa Pinto; Lacerda, Marcus Vinicius Guimarães; Bilsland, Elizabeth; Sunnerhagen, Per; Neves, Bruno Junior; Andrade, Carolina Horta; Cravo, Pedro Vitor Lemos; Costa, Fabio Trindade Maranhão

Integrative Multi-Kinase Approach for the Identification of Potent Antiplasmodial Hits

整合多激酶方法筛选高效抗疟原虫先导化合物

Lima, Marilia N N; Cassiano, Gustavo C; Tomaz, Kaira C P; Silva, Arthur C; Sousa, Bruna K P; Ferreira, Leticia T; Tavella, Tatyana A; Calit, Juliana; Bargieri, Daniel Y; Neves, Bruno J; Costa, Fabio T M; Andrade, Carolina Horta

Screening the Pathogen Box for Molecules Active against Plasmodium Sexual Stages Using a New Nanoluciferase-Based Transgenic Line of P. berghei Identifies Transmission-Blocking Compounds

使用基于纳米荧光素酶的新型伯氏疟原虫转基因系筛选病原体盒中针对疟原虫有性阶段具有活性的分子,从而识别出阻断传播的化合物

Juliana Calit #, Irina Dobrescu #, Xiomara A Gaitán, Miriam H Borges, Marisé S Ramos, Richard T Eastman, Daniel Y Bargieri