日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Piperidine CD4-Mimetic Compounds Expose Vulnerable Env Epitopes Sensitizing HIV-1-Infected Cells to ADCC

哌啶 CD4 模拟化合物暴露易受攻击的 Env 表位,使 HIV-1 感染细胞对 ADCC 敏感

Shilei Ding, William D Tolbert, Huile Zhu, Daniel Lee, Lorie Marchitto, Tyler Higgins, Xuchen Zhao, Dung Nguyen, Rebekah Sherburn, Jonathan Richard, Gabrielle Gendron-Lepage, Halima Medjahed, Mohammadjavad Mohammadi, Cameron Abrams, Marzena Pazgier, Amos B Smith 3rd, Andrés Finzi

Indoline CD4-mimetic compounds mediate potent and broad HIV-1 inhibition and sensitization to antibody-dependent cellular cytotoxicity

二氢吲哚 CD4 模拟化合物介导强效和广泛的 HIV-1 抑制以及对抗体依赖性细胞毒性的敏化

Christopher J Fritschi, Saumya Anang, Zhen Gong, Mohammadjavad Mohammadi, Jonathan Richard, Catherine Bourassa, Kenny T Severino, Hannah Richter, Derek Yang, Hung-Ching Chen, Ta-Jung Chiu, Michael S Seaman, Navid Madani, Cameron Abrams, Andrés Finzi, Wayne A Hendrickson, Joseph G Sodroski, Amos B Sm

Piperidine CD4-mimetic compounds expose vulnerable Env epitopes sensitizing HIV-1-infected cells to ADCC

哌啶 CD4 模拟化合物暴露易受攻击的 Env 表位,使 HIV-1 感染细胞对 ADCC 敏感

Shilei Ding, William D Tolbert, Huile Zhu, Daniel Lee, Tyler Higgins, Xuchen Zhao, Dung Nguyen, Rebekah Sherburn, Jonathan Richard, Gabrielle-Gendron Lepage, Halima Medjahed, Mohammadjavad Mohammadi, Cameron Abrams, Marzena Pazgier, Amos B Smith 3rd, Andrés Finzi

VE607 stabilizes SARS-CoV-2 Spike in the "RBD-up" conformation and inhibits viral entry

VE607 可稳定 SARS-CoV-2 刺突蛋白的“RBD 上调”构象,从而抑制病毒入侵。

Shilei Ding ,Irfan Ullah ,Shang Yu Gong ,Jonathan R Grover ,Mohammadjavad Mohammadi ,Yaozong Chen ,Dani Vézina ,Guillaume Beaudoin-Bussières ,Vijay Tailor Verma ,Guillaume Goyette ,Fleur Gaudette ,Jonathan Richard ,Derek Yang ,Amos B Smith 3rd ,Marzena Pazgier ,Marceline Côté ,Cameron Abrams ,Priti Kumar ,Walther Mothes ,Pradeep D Uchil ,Andrés Finzi ,Christian Baron

A New Family of Small-Molecule CD4-Mimetic Compounds Contacts Highly Conserved Aspartic Acid 368 of HIV-1 gp120 and Mediates Antibody-Dependent Cellular Cytotoxicity

一类新的小分子 CD4 模拟化合物与 HIV-1 gp120 高度保守的天冬氨酸 368 接触并介导抗体依赖性细胞毒作用

Shilei Ding #, Melissa C Grenier #, William D Tolbert, Dani Vézina, Rebekah Sherburn, Jonathan Richard, Jérémie Prévost, Jean-Philippe Chapleau, Gabrielle Gendron-Lepage, Halima Medjahed, Cameron Abrams, Joseph Sodroski, Marzena Pazgier, Amos B Smith 3rd, Andrés Finzi

The β20-β21 of gp120 is a regulatory switch for HIV-1 Env conformational transitions

gp120 的 β20-β21 是 HIV-1 Env 构象转变的调节开关

Alon Herschhorn, Christopher Gu, Francesca Moraca, Xiaochu Ma, Mark Farrell, Amos B Smith 3rd, Marie Pancera, Peter D Kwong, Arne Schön, Ernesto Freire, Cameron Abrams, Scott C Blanchard, Walther Mothes, Joseph G Sodroski

Recognition of HIV-inactivating peptide triazoles by the recombinant soluble Env trimer, BG505 SOSIP.664

重组可溶性 Env 三聚体 BG505 SOSIP.664 对 HIV 灭活肽三唑的识别

Kriti Acharya, Adel A Rashad, Francesca Moraca, Per Johan Klasse, John P Moore, Cameron Abrams, Irwin Chaiken

Impact of HIV-1 Membrane Cholesterol on Cell-Independent Lytic Inactivation and Cellular Infectivity

HIV-1 膜胆固醇对细胞独立溶解失活和细胞传染性的影响

Ramalingam Venkat Kalyana Sundaram, Huiyuan Li, Lauren Bailey, Adel A Rashad, Rachna Aneja, Karl Weiss, James Huynh, Arangaserry Rosemary Bastian, Elisabeth Papazoglou, Cameron Abrams, Steven Wrenn, Irwin Chaiken

Mechanism of multivalent nanoparticle encounter with HIV-1 for potency enhancement of peptide triazole virus inactivation

多价纳米粒子与 HIV-1 相遇增强肽三唑病毒灭活效力的机制

Arangassery Rosemary Bastian, Aakansha Nangarlia, Lauren D Bailey, Andrew Holmes, R Venkat Kalyana Sundaram, Charles Ang, Diogo R M Moreira, Kevin Freedman, Caitlin Duffy, Mark Contarino, Cameron Abrams, Michael Root, Irwin Chaiken