日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Species-Selective Reversible Proteasome Inhibitors for the Treatment of Malaria

优化物种选择性可逆蛋白酶体抑制剂以治疗疟疾

Gahalawat, Suraksha; Ray, Sneha; Zhang, Xiaoyu; Deng, Xiaoyi; Han, Yan; Chen, Zhe; Lawong, Aloysus; Shackleford, David M; Katneni, Kasiram; Chen, Gong; Li, Peng; Ng, Alice; Zhong, Longjin; Hu, Meiyu; McInerney, Mitchell; Wang, Wen; Saunders, Jessica; Collins, Daniel; Jayaseelan, Jaya; Noack, Cassandra L; C Maity, Bikash; De, Nirupam; Laleu, Benoît; Campbell, Simon F; Phillips, Margaret A; Charman, Susan A; Ready, Joseph M

Identification of potent and reversible piperidine carboxamides that are species-selective orally active proteasome inhibitors to treat malaria.

鉴定出强效且可逆的哌啶甲酰胺类化合物,它们是具有物种选择性的口服活性蛋白酶体抑制剂,可用于治疗疟疾

Lawong Aloysus, Gahalawat Suraksha, Ray Sneha, Ho Nhi, Han Yan, Ward Kurt E, Deng Xiaoyi, Chen Zhe, Kumar Ashwani, Xing Chao, Hosangadi Varun, Fairhurst Kate J, Tashiro Kyuto, Liszczak Glen, Shackleford David M, Katneni Kasiram, Chen Gong, Saunders Jessica, Crighton Elly, Casas Arturo, Robinson Joshua J, Imlay Leah S, Zhang Xiaoyu, Lemoff Andrew, Zhao Zhiyu, Angulo-Barturen Iñigo, Jiménez-Díaz María Belén, Wittlin Sergio, Campbell Simon F, Fidock David A, Laleu Benoît, Charman Susan A, Ready Joseph M, Phillips Margaret A

Substituted Aminoacetamides as Novel Leads for Malaria Treatment

取代氨基乙酰胺作为疟疾治疗的新型先导化合物

Norcross, Neil R; Wilson, Caroline; Baragaña, Beatriz; Hallyburton, Irene; Osuna-Cabello, Maria; Norval, Suzanne; Riley, Jennifer; Fletcher, Daniel; Sinden, Robert; Delves, Michael; Ruecker, Andrea; Duffy, Sandra; Meister, Stephan; Antonova-Koch, Yevgeniya; Crespo, Benigno; de Cózar, Cristina; Sanz, Laura M; Gamo, Francisco Javier; Avery, Vicky M; Frearson, Julie A; Gray, David W; Fairlamb, Alan H; Winzeler, Elizabeth A; Waterson, David; Campbell, Simon F; Willis, Paul A; Read, Kevin D; Gilbert, Ian H