The compound millepachine and its derivatives inhibit tubulin polymerization by irreversibly binding to the colchicine-binding site in β-tubulin
化合物米帕金及其衍生物通过不可逆地结合β-微管蛋白中的秋水仙碱结合位点来抑制微管蛋白聚合
期刊:Journal of Biological Chemistry
影响因子:4
doi:10.1074/jbc.RA117.001658
Jianhong Yang, Wei Yan, Yamei Yu, Yuxi Wang, Tao Yang, Linlin Xue, Xue Yuan, Caofeng Long, Zuowei Liu, Xiaoxin Chen, Mengshi Hu, Li Zheng, Qiang Qiu, Heying Pei, Dan Li, Fang Wang, Peng Bai, Jiaolin Wen, Haoyu Ye, Lijuan Chen