日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combined crystallographic fragment screening and deep mutational scanning enable discovery of Zika virus NS2B-NS3 protease inhibitors

结合晶体学片段筛选和深度突变扫描,可以发现寨卡病毒NS2B-NS3蛋白酶抑制剂。

Ni, Xiaomin; Richardson, R Blake; Godoy, Andre Schutzer; Ferla, Matteo P; Kikawa, Caroline; Scheen, Jenke; Hannon, William W; Capkin, Eda; Lahav, Noa; Balcomb, Blake H; Marples, Peter G; Fairhead, Michael; Wang, SiYi; Williams, Eleanor P; Tomlinson, Charles W E; Aschenbrenner, Jasmin C; Lithgo, Ryan M; Winokan, Max; Giroud, Charline; Dolci, Isabela; Fernandes, Rafaela Sachetto; Oliva, Glaucius; Chandran, Anu V; Xavier, Mary-Ann; Walsh, Martin A; Thompson, Warren; Bloom, Jesse D; Kenton, Nathaniel T; Lee, Alpha A; von Delft, Annette; Barr, Haim; Kirkegaard, Karla; Koekemoer, Lizbé; Fearon, Daren; Evans, Matthew J; von Delft, Frank

Therapeutic effects of cinnamic acid in a rat model of collagenase-induced Achilles tendinopathy

肉桂酸对胶原酶诱导的大鼠跟腱病模型的治疗作用

Capkin, Sercan; Kilic, Ali Ihsan; Dizakar, Saadet Ozen Akarca; Isin, Yagmur

Machine learning models for predicting tibial intramedullary nail length

用于预测胫骨髓内钉长度的机器学习模型

Capkin, Sercan; Kilic, Ali Ihsan; Cici, Hakan; Akdemir, Mehmet; Marasli, Mert Kahraman

A framework for countermeasures design to support professional drivers' fitness-to-drive

为保障职业驾驶员的驾驶能力而设计的应对措施框架

Filtness, Ashleigh; Pilkington-Cheney, Fran; Motnikar, Lenart; Talbot, Rachel; Capkin, Sevket Oguz Kagan; Touliou, Katerina; Delgrado, Beatriz; Anund, Anna

Crystallographic fragment screening and deep mutational scanning of Zika virus NS2B-NS3 protease enable development of resistance-resilient inhibitors

对寨卡病毒NS2B-NS3蛋白酶进行晶体学片段筛选和深度突变扫描,可以开发出抗耐药性抑制剂。

Ni, Xiaomin; Richardson, R Blake; Godoy, Andre Schutzer; Ferla, Matteo P; Kikawa, Caroline; Scheen, Jenke; Hannon, William W; Capkin, Eda; Lahav, Noa; Balcomb, Blake H; Marples, Peter G; Fairhead, Michael; Wang, Siyi; Williams, Eleanor P; Tomlinson, Charlie W E; Aschenbrenner, Jasmin Cara; Lithgo, Ryan M; Winokan, Max; Giroud, Charline; Chandran, Anu V; Walsh, Martin; Thompson, Warren; Bloom, Jesse D; Barr, Haim; Kirkegaard, Karla; Koekemoer, Lizbé; Fearon, Daren; Evans, Matthew J; von Delft, Frank

Crystallographic fragment screening and deep mutational scanning of Zika virus NS2B-NS3 protease enable development of resistance-resilient inhibitors

对寨卡病毒NS2B-NS3蛋白酶进行晶体学片段筛选和深度突变扫描,可以开发出抗耐药性抑制剂。

von Delft, Frank; Ni, Xiaomin; Richardson, R; Godoy, Andre; Ferla, Matteo; Kikawa, Caroline; Scheen, Jenke; Hannon, William; Capkin, Eda; Lahav, Noa; Balcomb, Blake; Marples, Peter; Fairhead, Michael; Wang, SiYi; Williams, Eleanor; Tomlinson, Charles; Aschenbrenner, Jasmin; Lithgo, Ryan; Winokan, Max; Giroud, Charline; Chandran, Anu; Walsh, Martin; Thompson, Warren; Bloom, Jesse; Barr, Haim; Kirkegaard, Karla; Koekemoer, Lizbé; Fearon, Daren; Evans, Matthew

Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening

通过晶体学片段筛选鉴定针对基孔肯雅病毒nsP3宏结构域的新型化学物质

Aschenbrenner, Jasmin C; de Godoy, Andre Schutzer; Fairhead, Michael; Tomlinson, Charles W E; Winokan, Max; Balcomb, Blake H; Capkin, Eda; Chandran, Anu V; Golding, Mathew; Koekemoer, Lizbe; Lithgo, Ryan M; Marples, Peter G; Ni, Xiaomin; Thompson, Warren; Wild, Conor; Xavier, Mary-Ann E; Fearon, Daren; von Delft, Frank

The effect of biceps tenotomy on superior humeral migration in arthroscopic repaired full-thickness supraspinatus tears

肱二头肌腱切断术对关节镜下修复全层冈上肌撕裂后肱骨上移的影响

Aydin, Mahmud; Capkin, Sercan; Surucu, Serkan; Karahasanoglu, Ridvan; Yilmaz, Murat

Structural and Functional Analysis of CEX Fractions Collected from a Novel Avastin® Biosimilar Candidate and Its Innovator: A Comparative Study

从新型 Avastin® 生物仿制药候选药物及其创新药物中收集的 CEX 馏分的结构和功能分析:一项比较研究

Busra Gurel, Melike Berksoz, Eda Capkin, Ayhan Parlar, Meltem Corbacioglu Pala, Aylin Ozkan, Yılmaz Capan, Duygu Emine Daglikoca, Meral Yuce

Characterization of FcγRIa (CD64) as a Ligand Molecule for Site-Specific IgG1 Capture: A Side-By-Side Comparison with Protein A

FcγRIa (CD64) 作为位点特异性 IgG1 捕获配体分子的表征:与 Protein A 的并排比较

Eda Capkin, Hasan Kurt, Busra Gurel, Dilan Bicak, Sibel Akgun Bas, Duygu Emine Daglikoca, Meral Yuce