日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Prodiginines as Single-Dose Curative Antimalarials

优化灵菌红素类药物作为单剂量治愈性抗疟药

Kumar, Amrendra; Li, Yuexin; Zhang, Xiaowei; Gaddam, Mahesh; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; DeLuca, Jesse; Vuong, Chau; Kudyba, Karl; Roncal, Norma; Ashraf, Kutub; Lee, Patricia J; Pannone, Kristina; Leed, Susan; Dinh, Hieu T; Mdaki, Kennedy; Navarrete, Kimberly; Charlton, Jordan; Binauhan, Angely J; Qahash, Tarrick; Kibe, Kevin Mugambi; Shoue, Douglas A; Checkley, Lisa; Ferdig, Michael T; Chim-Ong, Anongruk; Cui, Liwang; Orena, Stephen; Byaruhanga, Oswald; Assimwe, Jackson; Tibagambirwa, Innocent; Chithanna, Sivanna; Dodean, Rozalia A; Legac, Jennifer; Kreutzfeld, Oriana; Rosenthal, Philip J; Cooper, Roland A; Reynolds, Kevin A; Roth, Alison; Kelly, Jane X; Kancharla, Papireddy

Preclinical in vitro and in vivo evaluation of omadacycline against multidrug-resistant Acinetobacter baumannii

奥马环素对多重耐药鲍曼不动杆菌的临床前体外和体内评价

Vanachayangkul, Pattaraporn; Ruamsap, Nattaya; Caridha, Diana; Imerbsin, Rawiwan; Ball, Erin; Chattagul, Supaksorn; Tungtang, Anchalee; Gonwong, Siriphan; Kodchakorn, Chanikarn; Lertsethtakarn, Paphavee; Silapong, Sasikorn; Chaisatit, Chaiyaporn; Khemnu, Nuanpan; Boudreaux, Daniel; Boonyalai, Nonlawat; Demons, Samandra; Pierce, Jessica V; Martin, Monica; Anastasiou, Diane; Serio, Alisa W; Vesely, Brian; Lanteri, Charlotte Anne

In vitro activity and in vivo efficacy of omadacycline against Plasmodium species.

奥马环素对疟原虫的体外活性和体内疗效

Madejczyk Michael S, Leed Susan E, Kudyba Karl, Roth Alison, Martin Monica L, Lee Patricia, Anastasiou Diane, Pierce Jessica V, Serio Alisa W, Caridha Diana

Potent Acridone Antimalarial against All Three Life Stages of Plasmodium

强效抗疟药吖啶酮,可对抗疟原虫所有三个生命阶段

Kancharla, Papireddy; Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kelly, Sean; Charlton, Jordan; Binauhan, Angley; Garcia, Laurize; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Kudyba, Karl; McEnearney, Sharon; Lee, Partricia J; Blount, Cameron; DeLuca, Jesse; Vuong, Chua; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Martin, Monica L; Pybus, Brandon S; Chimong, Anongruk; Cui, Liwang; Vega-Rodriguez, Joel; Okitwi, Martin; Kreutzfeld, Oriana; Docan, Christina; Green, Carol; Liu, Ying; Agulay, Aaron; Mirsalis, Jon; Farrell, Sarah N; McFadden, Geoffrey I; Goodman, Christopher D; Probst, Alexandra S; Nilsen, Aaron; Catteruccia, Flaminia; Rosenthal, Philip J; Riscoe, Michael; Cooper, Roland; Roth, Alison; Kelly, Jane

Discovery and Optimization of Tambjamines as a Novel Class of Antileishmanial Agents

发现和优化 Tambjamines 作为一类新型抗利什曼原虫药物

Papireddy Kancharla, Diana Ortiz, Corinne M Fargo, Xiaowei Zhang, Yuexin Li, Marco Sanchez, Amrendra Kumar, Monish Yeluguri, Rozalia A Dodean, Diana Caridha, Michael S Madejczyk, Monica Martin, Xiannu Jin, Cameron Blount, Ravi Chetree, Kristina Pannone, Hieu T Dinh, Jesse DeLuca, Martin Evans, Rober

DDDR-05. SPATIALLY RESOLVED DRUG SENSITIVITY PROFILING IN GLIOBLASTOMA

DDDR-05. 胶质母细胞瘤的空间分辨药物敏感性分析

Kumar, Amrendra; Li, Yuexin; Dodean, Rozalia A; Roth, Alison; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Lee, Patricia J; Pybus, Brandon S; Martin, Monica; Pannone, Kristina; Dinh, Hieu T; Blount, Cameron; Chetree, Ravi; DeLuca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G; Rasmussen, Stephanie A; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A; Delves, Michael J; Matthews, Holly; Baum, Jake; Kirby, Robert W; Burrows, Jeremy N; Duffy, James; Peyton, David H; Reynolds, Kevin A; Kelly, Jane X; Kancharla, Papireddy; Buck, Alicia; Lee, Sohyon; Wegmann, Rebekka; Mena, Julien; Vasella, Flavio; Friesen, Julia; Regli, Luca; Le Rhun, Emilie; Zeitlberger, Anna Maria; Neidert, Marian Christoph; Tatari, Nazanin; Hutter, Gregor; Weller, Michael; Snijder, Berend; Weiss, Tobias

Animal Models in Regulatory Breakpoint Determination: Review of New Drug Applications of Approved Antibiotics from 2014-2022

动物模型在监管断点确定中的应用:2014-2022年已批准抗生素新药申请的回顾

Selig, Daniel; Caridha, Diana; Evans, Martin; Kress, Adrian; Lanteri, Charlotte; Ressner, Roseanne; DeLuca, Jesse

Dual stop codon suppression in mammalian cells with genomically integrated genetic code expansion machinery

具有基因组整合遗传密码扩展机制的哺乳动物细胞中的双终止密码子抑制

Birthe Meineke, Johannes Heimgärtner, Rozina Caridha, Matthias F Block, Kyle J Kimler, Maria F Pires, Michael Landreh, Simon J Elsässer

An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections

迭代方法指导FabI抑制剂法比霉素的发现,法比霉素是一种后期抗生素候选药物,对耐药革兰氏阴性菌感染具有体内疗效。

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J

Correction to "An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections"

对“迭代方法指导发现FabI抑制剂法比霉素,一种对耐药革兰氏阴性菌感染具有体内疗效的后期抗生素候选药物”一文的更正

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Rohde, Jason M; Zak, Mark; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J