日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-class multifunctional TYMS nonclassical antifolate inhibitor with potent in vivo activity that prolongs survival

首创的多功能 TYMS 非经典抗叶酸抑制剂,具有强效体内活性,可延长生存期

Maria V Guijarro, Patrick C Kellish, Peter E Dib, Nicholas G Paciaroni, Akbar Nawab, Jacob Andring, Lidia Kulemina, Nicholas V Borrero, Carlos Modenutti, Michael Feely, Elham Nasri, Robert P Seifert, Xiaoping Luo, Richard L Bennett, Daniil Shabashvili, Jonathan D Licht, Robert McKenna, Adrian Roitbe

A Remote Secondary Binding Pocket Promotes Heteromultivalent Targeting of DC-SIGN

远程二级结合口袋促进 DC-SIGN 的异多价靶向

Robert Wawrzinek, Eike-Christian Wamhoff, Jonathan Lefebre, Mareike Rentzsch, Gunnar Bachem, Gary Domeniconi, Jessica Schulze, Felix F Fuchsberger, Hengxi Zhang, Carlos Modenutti, Lennart Schnirch, Marcelo A Marti, Oliver Schwardt, Maria Bräutigam, Mónica Guberman, Dirk Hauck, Peter H Seeberger, Oli