日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Covalent adduct Grob fragmentation underlies LSD1 demethylase-specific inhibitor mechanism of action and resistance.

共价加合物 Grob 断裂是 LSD1 去甲基酶特异性抑制剂作用机制和耐药性的基础

Waterbury Amanda L, Caroli Jonatan, Zhang Olivia, Tuttle Paloma R, Liu Chao, Li Jiaming, Park Ji Sung, Hoenig Samuel M, Barone Marco, Furui Airi, Mattevi Andrea, Liau Brian B

Uncoupling histone modification crosstalk by engineering lysine demethylase LSD1.

通过改造赖氨酸去甲基酶 LSD1 来解耦组蛋白修饰串扰

Lee Kwangwoon, Barone Marco, Waterbury Amanda L, Jiang Hanjie, Nam Eunju, DuBois-Coyne Sarah E, Whedon Samuel D, Wang Zhipeng A, Caroli Jonatan, Neal Katherine, Ibeabuchi Brian, Dhoondia Zuzer, Kuroda Mitzi I, Liau Brian B, Beck Samuel, Mattevi Andrea, Cole Philip A

Tranylcypromine-Based LSD1 Inhibitors as Useful Agents to Reduce Viability of Schistosoma mansoni

基于反式环丙胺的LSD1抑制剂可有效降低曼氏血吸虫的存活率

Fabbrizi, Emanuele; Hailu, Gebremedhin Solomon; Ganesan, A; Fioravanti, Rossella; Zwergel, Clemens; Lambona, Chiara; Valente, Sergio; Fianco, Giulia; Iuzzolino, Angela; Trisciuoglio, Daniela; Caroli, Jonatan; Mattevi, Andrea; Häberli, Cécile; Keiser, Jennifer; Rotili, Dante; Mai, Antonello