日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Arrestin-biased allosteric modulator of neurotensin receptor 1 alleviates acute and chronic pain.

神经降压素受体 1 的 Arrestin 偏向性变构调节剂可缓解急性和慢性疼痛

Guo Ran, Chen Ouyang, Zhou Yang, Bang Sangsu, Chandra Sharat, Li Yize, Chen Gang, Xie Rou-Gang, He Wei, Xu Jing, Zhou Richard, Song Shaoyong, Person Kelsey L, Moore Madelyn N, Alwin Abigail R, Spasojevic Ivan, Jackson Michael R, Olson Steven H, Caron Marc G, Slosky Lauren M, Wetsel William C, Barak Lawrence S, Ji Ru-Rong

Combination of Haloperidol With UNC9994, β-arrestin-Biased Analog of Aripiprazole, Ameliorates Schizophrenia-Related Phenotypes Induced by NMDAR Deficit in Mice.

氟哌啶醇与 UNC9994(阿立哌唑的β-arrestin偏向类似物)的组合可改善小鼠NMDAR缺陷引起的精神分裂症相关表型

Lipina Tatiana V, Giang Huy, Thacker Jonathan S, Wetsel William C, Caron Marc G, Beaulieu Jean Martin, Salahpour Ali, Ramsey Amy J

Ghrelin receptor signaling in health and disease: a biased view

胃饥饿素受体信号传导在健康和疾病中的作用:一种有偏见的观点

Gross, Joshua D; Zhou, Yang; Barak, Lawrence S; Caron, Marc G

Neurotensin receptor 1-biased ligand attenuates neurotensin-mediated excitation of ventral tegmental area dopamine neurons and dopamine release in the nucleus accumbens

神经降压素受体1偏向性配体减弱神经降压素介导的腹侧被盖区多巴胺神经元的兴奋以及伏隔核中的多巴胺释放

Singhal, Sarthak M; Zell, Vivien; Faget, Lauren; Slosky, Lauren M; Barak, Lawrence S; Caron, Marc G; Pinkerton, Anthony B; Hnasko, Thomas S

Prenatal heroin exposure alters brain morphology and connectivity in adolescent mice

产前接触海洛因会改变青春期小鼠的大脑形态和连接性。

Hornburg, Kathryn J; Slosky, Lauren M; Cofer, Gary; Cook, James; Qi, Yi; Porkka, Fiona; Clark, Nicholas B; Pires, Andrea; Petrella, Jeffrey R; White, Leonard E; Wetsel, William C; Barak, Lawrence; Caron, Marc G; Johnson, G Allan

Biased agonists of the chemokine receptor CXCR3 differentially signal through Gα(i):β-arrestin complexes

趋化因子受体CXCR3的偏向性激动剂通过Gα(i):β-arrestin复合物差异性地传递信号

Zheng, Kevin; Smith, Jeffrey S; Eiger, Dylan S; Warman, Anmol; Choi, Issac; Honeycutt, Christopher C; Boldizsar, Noelia; Gundry, Jaimee N; Pack, Thomas F; Inoue, Asuka; Caron, Marc G; Rajagopal, Sudarshan

Establishment of multi-stage intravenous self-administration paradigms in mice

建立小鼠多阶段静脉注射自我给药模型

Slosky, Lauren M; Pires, Andrea; Bai, Yushi; Clark, Nicholas B; Hauser, Elizabeth R; Gross, Joshua D; Porkka, Fiona; Zhou, Yang; Chen, Xiaoxiao; Pogorelov, Vladimir M; Toth, Krisztian; Wetsel, William C; Barak, Lawrence S; Caron, Marc G

Biased Allosteric Modulators: New Frontiers in GPCR Drug Discovery

偏向性变构调节剂:GPCR药物发现的新前沿

Slosky, Lauren M; Caron, Marc G; Barak, Lawrence S

Cholinergic dysfunction in the dorsal striatum promotes habit formation and maladaptive eating

背侧纹状体胆碱能功能障碍会促进习惯形成和适应不良的饮食行为。

Favier, Mathieu; Janickova, Helena; Justo, Damian; Kljakic, Ornela; Runtz, Léonie; Natsheh, Joman Y; Pascoal, Tharick A; Germann, Jurgen; Gallino, Daniel; Kang, Jun-Ii; Meng, Xiang Qi; Antinora, Christina; Raulic, Sanda; Jacobsen, Jacob Pr; Moquin, Luc; Vigneault, Erika; Gratton, Alain; Caron, Marc G; Duriez, Philibert; Brandon, Mark P; Neto, Pedro Rosa; Chakravarty, M Mallar; Herzallah, Mohammad M; Gorwood, Philip; Prado, Marco Am; Prado, Vania F; El Mestikawy, Salah

Deletion of Glycogen Synthase Kinase-3β in D(2) Receptor-Positive Neurons Ameliorates Cognitive Impairment via NMDA Receptor-Dependent Synaptic Plasticity

糖原合成酶激酶-3β在D(2)受体阳性神经元中的缺失可通过NMDA受体依赖性突触可塑性改善认知障碍

Li, Yan-Chun; Panikker, Priyalakshmi; Xing, Bo; Yang, Sha-Sha; Alexandropoulos, Cassandra; McEachern, Erin P; Akumuo, Rita; Zhao, Elise; Gulchina, Yelena; Pletnikov, Mikhail V; Urs, Nikhil M; Caron, Marc G; Elefant, Felice; Gao, Wen-Jun