Discovery of VU6024578/BI02982816: An mGlu(1) Positive Allosteric Modulator with Efficacy in Preclinical Antipsychotic and Cognition Models
VU6024578/BI02982816 的发现:一种 mGlu(1) 正向变构调节剂,在临床前抗精神病和认知模型中具有疗效
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c02554
Reed, Carson W; Kalbfleisch, Jacob F; Turkett, Jeremy A; Trombley, Trevor A; Nastase, Anthony F; Spearing, Paul K; Haymer, Daniel H; Sarwar, Mohammad Moshin; Quitalig, Marc; Dickerson, Jonathan W; Blobaum, Annie L; Boutaud, Olivier; Voehringer, Patrizia; Schuelert, Niklas; Cho, Hyekyung P; Niswender, Colleen M; Rook, Jerri M; Priepke, Henning; Ursu, Daniel; Conn, P Jeffrey; Melancon, Bruce J; Lindsley, Craig W