日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of diastereomeric dihydropyridines as antimalarials

优化非对映异构二氢吡啶类化合物作为抗疟药

Van Horn, Kurt S; Zhao, Yingzhao; Parvatkar, Prakash T; Maier, Julie; Mutka, Tina; Lacrue, Alexis; Brockmeier, Fabian; Ebert, Daniel; Wu, Wesley; Casandra, Debora R; Namelikonda, Niranjan; Yacoub, Jeanine; Sigal, Martina; Knapp, Spencer; Floyd, David; Waterson, David; Burrows, Jeremy N; Duffy, James; DeRisi, Joseph L; Kyle, Dennis E; Guy, R Kiplin; Manetsch, Roman

Protein KIC5 is a novel regulator of artemisinin stress response in the malaria parasite Plasmodium falciparum

蛋白质KIC5是疟原虫(恶性疟原虫)中青蒿素应激反应的一种新型调节因子。

Simmons, Caroline F; Gibbons, Justin; Zhang, Min; Oberstaller, Jenna; Pires, Camilla Valente; Casandra, Debora; Wang, Chengqi; Seyfang, Andreas; Otto, Thomas D; Rayner, Julian C; Adams, John H

Chemogenomic Profiling of a Plasmodium falciparum Transposon Mutant Library Reveals Shared Effects of Dihydroartemisinin and Bortezomib on Lipid Metabolism and Exported Proteins.

对恶性疟原虫转座子突变体库的化学基因组分析揭示了双氢青蒿素和硼替佐米对脂质代谢和输出蛋白的共同影响

Pires Camilla Valente, Oberstaller Jenna, Wang Chengqi, Casandra Debora, Zhang Min, Chawla Jyotsna, Adapa Swamy Rakesh, Otto Thomas D, Ferdig Michael T, Rayner Julian C, Jiang Rays H Y, Adams John H

A novel Modulator of Ring Stage Translation (MRST) gene alters artemisinin sensitivity in Plasmodium falciparum

一种新型的环状期翻译调节因子(MRST)基因改变了恶性疟原虫对青蒿素的敏感性

Simmons, Caroline; Gibbons, Justin; Wang, Chengqi; Pires, Camilla Valente; Zhang, Min; Siddiqui, Faiza; Oberstaller, Jenna; Casandra, Debora; Seyfang, Andreas; Cui, Liwang; Otto, Thomas D; Adams, John H

Structure-activity and structure-property relationship studies of spirocyclic chromanes with antimalarial activity

螺环色满类化合物抗疟活性的构效关系和构性关系研究

Iyamu, Iredia D; Zhao, Yingzhao; Parvatkar, Prakash T; Roberts, Bracken F; Casandra, Debora R; Wojtas, Lukasz; Kyle, Dennis E; Chakrabarti, Debopam; Manetsch, Roman

Design and Synthesis of Orally Bioavailable Piperazine Substituted 4(1H)-Quinolones with Potent Antimalarial Activity: Structure-Activity and Structure-Property Relationship Studies

口服生物利用度高的哌嗪取代的4(1H)-喹诺酮类化合物的设计与合成及其强效抗疟活性:构效关系和构性关系研究

Neelarapu, Raghupathi; Maignan, Jordany R; Lichorowic, Cynthia L; Monastyrskyi, Andrii; Mutka, Tina S; LaCrue, Alexis N; Blake, Lynn D; Casandra, Debora; Mashkouri, Sherwin; Burrows, Jeremy N; Willis, Paul A; Kyle, Dennis E; Manetsch, Roman

Artemisinin-resistant Plasmodium falciparum parasites exhibit altered patterns of development in infected erythrocytes

对青蒿素产生耐药性的恶性疟原虫在感染的红细胞中表现出发育模式的改变。

Hott, Amanda; Casandra, Debora; Sparks, Kansas N; Morton, Lindsay C; Castanares, Geocel-Grace; Rutter, Amanda; Kyle, Dennis E

Development of a pediatric formulation for treatment of P. falciparum malaria: Coartem(®) (artemether-lumefantrine) Dispersible

开发用于治疗恶性疟原虫疟疾的儿科制剂:Coartem®(蒿甲醚-苯芴醇)分散片

Lehmann, Tovi; Dao, Adama; Yaro, Alpha S; Huestis, Diana L; Diallo, Moussa; Timbiné, Seydou; Kassogué, Yaya; Adamou, Alpha; Traoré, Adama I; Samaké, Djibril; Howes, Rosalind; Weatherall, David; Douglas, Ross; Ester, Miriam; Hellmann, Janina; Frischknecht, Friedrich; Bello, Ibrahim S; Elusiyan, Jerome B; Awokola, Babatunde I; Ogundokun, Akinjide O; Omisore, Bridget; Oyegbade, Olanrewaju; Olowookere, Samuel Anu; Abioye-Kuteyi, Emmanuel Akintunde; Elujoba, Joseph O; Adeogun, Adedapo O; Popoola, Kehinde OK; Koekemoer, Lizette L; Brooke, Basil D; Oduola5, Adedayo O; Awolola, Samson T; Feachem, Richard; Arango, Eliana; Carmona, Jaime; Maestre, Amanda; Deobagkar, Deepti; Ozarkar, Aarti; Gupta, Shipra; Agrawal, Megha; Deobagkar, Dileep; Birth, Dominic; Kao, Wei-chun; Hunte, Carola; Etim, Susan; Ogbeche, Jude; Pothin, Emilie; Briët, Olivier; Kesteman, Thomas; Randrianarivelojosia, Milijaona; Rogier, Christophe; Smith, Thomas; Willcox, Merlin; Diallo, Drissa; Diakité, Chiaka; Daou, Pierre; Bamba, Drissa; Dembélé, Eugene; Harnden, Anthony; Mant, David; Biagini, Giancarlo; Billingsley, Peter; Sim, B Kim Lee; Bijker, Else; Roestenberg, Meta; Lyke, Kirsten; Laurens, Matthew; Mordmueller, Benjamin; Gomez, Patricia; Shekalaghe, Seif; Hodgson, Susanne; Hill, Adrian; Juma, Elizabeth; Ogutu, Bernhards; Lell, Bertrand; Alonso, Pedro; Abdullah, Salim; Kremsner, Peter; Tanner, Marcel; Sauerwein, Robert; Hoffman, Stephen; Bliss, Carly M; Salman, Ahmed M; Longley, Rhea J; Khan, Shahid M; Janse, Chris J; Hill, Adrian VS; Ewer, Katie J; Birkholtz, Lyn-Marie; LeRoy, Didier; Reader, Janette; Botha, Mariette; Mancama, Dalu; Coetzer, Theresa L; Bowyer, Georgina; Afolabi, Muhammed O; Bliss, Carly M; Tiono, Alfred B; Drammeh, Abdoulie; Nébié, Issa; Jagne, Ya Jankey; Yaro, Jean Baptiste; Imoukhuede, Egeruan B; Flanagan, Katie L; Kampman, Beate; Viebig, Nicola; Sirima, Sodiomon B; Bojang, Kalifa; Hill, Adrian VS; Ewer, Katie J; Bouyou-Akotet, Marielle Karine; Mawili-Mboumba, DP; Ndong, R Nikiema; Kendjo, E; Charron, Brigitte; Lameyre, Valérie; Kombila, Maryvonne; Adams, John H; George, Miriam T; Ntumngia, Francis B; Schloegel, Jesse; Barnes, Samantha J; McHenry, Amy M; Schuldt, Kathrin; Evans, Jennifer; Lenzen, Julia; Ehmen, Christa; Muntau, Birgit; Sievertsen, Jurgen; Enuameh, Yeetey; Osei-Kwakye, Kingsley; Opoku, Ernest Cudjoe; Browne, Edmund NL; Horstmann, Rolf; Timmann, Christian; Wampfler, Rahel; Robinson, Leanne; Hofmann, Natalie; Waltmann, Andreea; Betuela, Inoni; Silkey, Mariabeth; Siba, Peter; Smith, Tom; Mueller, Ivo; Felger, Ingrid; Kyle, Dennis E; Zhang, Rou; Lee, Wenn-Chyau; Malleret, Benoit; Suwanarusk, Rossarin; Dao, Ming; Chu, Cindy; Lim, Chwee Teck; Renia, Laurent; Nosten, Francois; Russell, Bruce; Eisele, Thomas; Steketee, Richard W; Hill, Adrian VS; Biswas, Sumi; Draper, Simon; Rampling, Thomas; Reyes-Sandoval, Arturo; Bhatt, Samir; Gething, Peter; Sauerwein, Robert; Hodgson, Susanne; Juma, Elizabeth; Salim, Amina; Magiri, Charles; Kimani, Domtila; Njenga, Daniel; Muia, Alfred; Cole, Andrew; Ogwang, Caroline; Billingsley, Peter; James, Eric; Sim, Kim Lee; Rampling, Thomas; Hill, Adrian; Osier, Faith; Draper, Simon; Bejon, Philip; Hoffman, Stephen; Ogutu, Bernhards; Marsh, Kevin; Shanks, Dennis; Billingsley, Peter; Sim, B Kim Lee; James, Eric; Richie, Thomas; Shekalaghe, Seif; Healy, Sara; Sissoko, Mahamadou; Mordmueller, Benjamin; Ledgerwood, Julie; Graham, Barney; Duffy, Patrick; Seder, Robert; Lyke, Kirsten; Epstein, Judith; Alonso, Pedro; Abdullah, Salim; Duombo, Ogobara; Kremsner, Peter; Tanner, Marcel; Hoffman, Stephen; Dabiré, Roch; Sawadogo, Simon; Diabaté, Abdoulaye; Toé, Hyacinthe; Kengne, Pierre; Ouari, Ali; Costantini, Carlo; Gouagna, Clement; Pennetier, Cedric; Simard, Frederic; Baldet, Thierry; Lehman, Tovi; Gibson, Gabriella; Leong, Joel; Li, Ruobing; Jain, Jay Prakash; Lefèvre, Gilbert; Magnusson, Baldur; Diagana, Thierry; Pertel, Peter; Ariey, Frédéric; Gomez, Daniela Zaffalon; Dussan, Andrés Olarte; Espinel, Vladimir Corredor; Morales, Hernando Diaz; Chan, Ernest; Menard, Didier; Barnwell, John; Zimmerman, Peter; Serre, David; Hopp, Christine; Sinnis, Photini; Kesteman, Thomas; Randrianarivelojosia, Milijaona; Piola, Patrice; Rogier, Christophe; Cunha, Janaiara A; Bianco-Junior, Cesare; Machado, Marcelo P; Druilhe, Pierre; Carvalho, Leonardo JM; Daniel-Ribeiro, Cláudio T; Dhimal, Meghnath; Ahrens, Bodo; Kuch, Ulrich; Deressa, Wakgari; Loha, Eskindir; Balkew, Meshesha; Desalegne, Alemayehu; Gari, Taye; Gebremichael, Teshome; Kenea, Oljira; Jima, Daddi; Robberstad, Bjarne; Overgaard, Hans J; Lindtjørn, Bernt; Dahal, Prabin; Eckhoff, Philip; Wenger, Edward; Endo, Akira; Nishiura, Hiroshi; Elias, Sean; Milne, Kathryn; Chui, Cecilia; Hodgson, Susanne; Borrow, Persephone; Draper, Simon; Ewer, Katie; Muller, Julius; Haks, Marielle; Loembe, Marguerite Massinga; Yazdanbakhsh, Maria; Matsumiya, Magali; Quinten, Edwin; Ottenhoff, Tom; Kremsner, Peter; Hill, Adrian; Smits, Hermelijn; Adegnika, Akim; Ajibaye, Olusola; Osuntoki, Akiniyi; Orok, Bassey; Iwalokun, Bamidele; Egbuna, Nneka; Olukosi, Yetunde; Aina, Olugbenga; Okoh, Hilary; Agomo, Chimere; Enya, Vera; Faneye, Oladayo; Akindele, Samuel; Akinnibosun, Olutope; Oyebola, Kolapo; Adenekan, Sunday; Ebuehi, Albert; Riccio, Evelyn Kety Pratt; Totino, Paulo Renato Rivas; Soares, Irene Silva; Rodrigues, Maurício Martins; Ribeiro, Cláudio Tadeu Daniel; de Fátima Ferreira da Cruz, Maria; Fabrigar, Danica; Penman, Bridget; Gupta, Sunetra; Weatherall, David; Galactionova, Katya; Tediosi, Fabrizio; de Savigny, Don; Smith, Thomas; Kahn, Maria; LaRue, Nicole; Wellhausen, Jeffrey; Pal, Sampa; Domingo, Gonzalo J; Fletcher, Sabine; Avery, Vicky; Kern, Steven E; McKenzie, F Ellis; Pemberton-Ross, Peter; Galactionova, Katya; Smith, Tom; Penny, Melissa; Krishna, Sanjeev; Wenger, Edward; Proctor, Joshua; Eckhoff, Philip; Sutherland, Colin; Braga de Oliveira, Alaide; Cristina de Paula, Renata; Dolabela, Maria Fani; Rocha, Fabiola; Gomes, Fabiana; Garavito, Giovanny; Brandão, Geraldo Célio; Mendes, Fúlvio; Tabach, Ricardo; Mourao, Luiza; Pucci, Maira; Almeida, Zelia; Pereira, Rosiane; Fontes, Cor Jesus; Lacerda, Marcus; Bemquerer, Marcelo; Braga, Erika; Ahmed, Rukhsana; Asih, Puji PB; Noviyanti, Rintis; Rozy, Ismail EP; Triyanti, Leily; Marleta, Rita; ter Kuile, Feiko; Syafruddin, Din; Bretscher, Michael T; Griffin, Jamie T; Hugo, Pierre; Baker, Mark; Ghani, Azra; Okell, Lucy; Chen, Ingrid; Drakeley, Chris; Poirot, Eugenie; Hwang, Jimee; Gosling, Roly; Burton, Robert; Tietje, Kathy; Ebels, Kelly; LaBarre, Paul; Andrade-Pacheco, Ricardo; Mubangizi, Martin; Quinn, John; Lawrence, Neil D; Kano, Flora S; Souza-Silva, Flávia A; Sousa, Taís N; Alves, Jéssica RS; Tang, Michaelis L; Rocha, Roberto S; Brito, Cristiana FA; Sell, Ana Maria; Carvalho, Luzia H; Kaneko, Akira; Chan, Chim; Taleo, George; Watanabe, Noriko; Kalkoa, Morris; Iamar, Sam; Chaves, Luis F; Junker, Klara; Cook, Jackie; Isozumi, Rie; Kimura, Masatsugu; Drakeley, Chris; Killeen, Gerry; Kano, Flora S; Lima, Barbara AS; Tang, Michaelis L; Costa, Pedro AC; Fontes, Cor JF; Sanchez, Bruno M; Rocha, Roberto S; Soares, Irene S; Brito, Cristiana FA; Antonelli, Lis; Carvalho, Luzia H; Uthaipibull, Chairat; Saengratwatchara, Patcharaporn; Boonbangyang, Manon; Prommana, Parichat; Kamchonwongpaisan, Sumalee; Srichiratanakool, Somdet; Walker, Andrew; Gupta, Sunetra; Bello, Ibrahim S; Rehal, Satwinder; Wimberly, Michael; Bayabil, Estifanos; Beyene, Belay; Henebry, Geoffrey; Liu, Yi; Mihretie, Abere; Senay, Gabriel; Keough, Dianne; Špaček, Petr; Hocková, Dana; Tichý, Tomáš; Vrbková, Silvie; Slavětínská, Lenka; Janeba, Zlatko; Naesens, Lieve; Edstein, Michael; Chavchich, Marina; Wang, Tzu; de Jersey, John; Guddat, Luke; Yamana, Teresa; Eltahir, Elfatih; Mensah, Victorine; Wright, Danny; Ewer, Katie; Edwards, Nick; Ndiaye, Magatte; Bejon, Phillip; Viebig, Nicola; Faye, Babacar; Hill, Adrian; Cisse, Badara; Tompkins, Adrian M; Di Giuseppe, Francesca; Colon-Gonzalez, Felipe; Chirombo, James; Bizimana, Jean Pierre; Namanya, Didacus; Homan, Tobias; Hiscox, Alexandra; di Pasquale, Aurelio; Kiche, Ibrahim; Mweresa, Collins; Mukabana, Wolfgang; Smith, Thomas; Takken, Willem; Maire, Nicolas; Zuccala, Elizabeth; Satchwell, Timothy; Angrisano, Fiona; Marapana, Danushka; Tan, Yan-Hong; Toye, Ashley; Baum, Jake; Valizadeh, Vahideh; Zakeri, Sedigheh; Mehrizi, Akram Abouei; Djadid, Navid Dinparast; Hott, Amanda; Casandra, Debora; Sparks, Kansas; Castarnes, Geocel; Rutter, Amanda; Kyle, Dennis; Humphreys, Georgina; Wondji, Charles; Paine, Mark; Miranda, Jacob; Ibrahim, Sulaiman; Hustedt, John; Canavati, Sara; Rang, Chandary; Uth, Sophal; Ly, Po; Sovannaroth, Siv; Ashton, Ruth; Meek, Sylvia; Felter, Arantxa Roca; Kalnoky, Michael; Kahn, Maria; Pal, Sampa; LaRue, Nicole; Leader, Brandon; Bancone, Germana; Nosten, Francois; Domingo, Gonzalo J; Kabir, Mohammad Moktadir; Naher, Shamsun; Islam, Akramul; Karim, Abdul; Rasid, Mohammad Harun-Or; Laskar, Shahidul Islam; Kajla, Mithilesh; Kakani, Parik; Choudhary, Tania Pal; Gupta, Kuldeep; Dhawan, Rini; Gakhar, SK; Gupta, Lalita; Kumar, Sanjeev; Peyton, David; Poirot, Eugenie; Stergachis, Andy; ter Kuile, Feiko; Guerin, Philippe J; Chen, Ingrid; Gosling, Roland; Alam, Mohammed Shafiul; Mohon, Abu Naser; Bayih, Abebe; Folefoc, Asongna; Pillai, Dylan; Machado, Patrícia; Vaz, Tiago R; Nogueira, Fátima; Rodrigues, João; Manco, Licínio; Ribeiro, Letícia; Bergstrom, Ed; Ashford, David; Vitorino, Rui; Thomas-Oates, Jane; Thomas, Jerry; Arez, Ana P; Khadjavi, Amina; Valente, Elena; Giribaldi, Giuliana; Prato, Mauro; Raeisi, Ahmad; Mirkhani, Vahid; Alkaran, Fatemeh Nikpour; Jalali, Bita Paktinat; Faraji, Leila; Keykhah, Mansour Ranjbar; Tabatabie, Seyed Mahdi; Makanga, Michael; Minzi, Omary; Maige, Sylivester; Sasi, Philip; Ngasala, Billy; Mappin, Bonnie; Dalrymple, Ursula; Cameron, Ewan; Bhatt, Samir; Weiss, Daniel J; Gething, Peter W; Nardella, Flore; Collot, Valérie; Stiebing, Sylvia; Kaiser, Marcel; Scmitt, Martine; Candolfi, Ermanno; Vonthron-Sénécheau, Catherine; Mørch, Kristine; Vivek, Rosario; Xena, Depeeka; Chandy, Sara; Manoharan, Anand; Haanshuus, Christel; Langeland, Nina; Blomberg, Bjørn; Mathai, Dilip; Palacpac, Nirianne MQ; Yagi, Masanori; Ntege, Edward; Balikagala, Betty; Yeka, Adoke; Shirai, Hiroki; Suzuki, Nahoko; Okada, Takuya; Kanoi, Bernard; Nobuko, Arisue; Tougan, Takahiro; Ishii, Ken J; Egwang, Thomas G; Horii, Toshihiro; Paganotti, Giacomo Maria; Gallo, Baba Christiane; Verra, Federica; Sirima, Bienvenu Sodiomon; Nebie’, Issa; Diarra, Amidou; Coluzzi, Mario; Modiano, David; Pett, Helmi; Drakeley, Chris; Eziefula, Chi; Neuvonen, Mikko; Lanke, Kjerstin; Sauerwein, Robert; Niemi, Mikko; Bousema, Teun; Reyes-Sandoval, Arturo; Khan, Shahid; Janse, Chris; Bachmann, Martin; Hill, Adrian; Rees-Channer, Roxanne; Cunningham, Jane; Chiodini, Peter; Barnwell, John; Glenn, Jeffery; Gonzalez, Iveth; Bell, David; Incardona, Sandra; Sanz, Laura; Lafuente, Maria Jose; Prats, Sara; Neria, Fernando; Roncalés, María; de Cózar, Cristina; Rodríguez, Ane; Gómez, María; Gamo, Francisco Javier; Santhanam, Jayanthi; Raberg, Lars; Read, Andrew; Savill, Nick; Sibanda, Mthokozisi; Focke, Walter; Ghidelli-Disse, Sonja; Lafuente-Monasterio, Maria Jose; Waterson, David; Witty, Michael; Younis, Yassir; Paquet, Tanya; Street, Leslie J; Chibale, Kelly; Gamo-Benito, Francisco Javier; Bantscheff, Marcus; Drewes, Gerard; Simão-Gurge, Raquel; Cricco, Julia; Wunderlich, Gerhard; Kimura, Emilia; Cirulli, Brenda; Katzin, Alejandro; Siegel, Sasha; Rivero, Andrea; Kyle, Dennis; Alves, Eduardo; Salman, Ahmed; Janse, Chris; Khan, Shahid; Hill, Adrian; Reyes-Sandoval, Arturo; Haanshuus, Christel Gill; Mohn, Stein Christian; Spencer, Alexandra; Longley, Rhea; Gola, Anita; Lambe, Teresa; Hill, Adrian; Srichairatanakool, Somdet; Thipubol, Supalerk; Tipsuwan, Wachiraporn; Uthaipibull, Chairat; Hiscox, Alexandra; Homan, Tobias; Vreugdenhil, Corné; Otieno, Bruno; Kibet, Anthony; Mweresa, Collins K; van Lammeren, Ron; Mukabana, Wolfgang R; Takken, Willem; Stresman, Gillian H; Baidjoe, Amrish; Stevenson, Jennifer; Odongo, Wycliffe; Owaga, Chrispin; Marube, Elizabeth; Osoti, Victor; Makori, Euniah; Shagari, Shehu; Drakeley, Chris; Cox, Jonathan; Bousema, Teun; Haanshuus, Christel Gill; Vivek, Rosario; Xena, Deepika; Chandy, Sara; Mathai, Dilip; Manoharan, Anand; Langeland, Nina; Blomberg, Bjørn; Mørch, Kristine; Stein, Daniel S; Jain, Jay Prakash; Lickliter, Jason; Kangas, Michael; Machineni, Surendra; Griffin, Paul; Lefevre, Gilbert; Tsoka-Gwegweni, Joyce; Okafor, Uchenna; Golassa, Lemu; Enweji, Nizar; Swedberg, Göte; Kamugisha, Erasmus; Choy, Angel; Hockham, Carinna; Penman, Bridget; Piel, Frédéric; Gupta, Sunetra; Leisewitz, Andrew; Turner, Gareth; Clift, Sarah; Pardini, Anne; Lafuente, Maria Jose; Guidelli-Disse, Sonja; Selenski, Carolyn; Lelievre, Joel; Willson, Timothy; Gamo, Francisco Javier; Drewes, Gerard; Vandal, Omar; Ballell-Pages, Luis; Littrell, Megan; Sudoi, Raymond; Archer, Julie; Ngigi, Julius; Ujuju, Chinazo; Mpanya, Godéfroid; Vasireddy, Vamsi; Poyer, Stephen; Bilak, Hana; Lindtjørn, Bernt; Loha, Eskindir; Deressa, Wakgari; Balkew, Meshesha; Gebremichael, Teshome; Sorteberg, Asgeir; Woyessa, Adugna; Animut, Abebe; Diriba, Korecha; Massebo, Fekadu; Viste, Ellen; Lunde, Torleif Markussen; Tesfahun, Dereje; Md Idris, Zulkarnain; Chim, Wai Chan; Chang, Sheng Deng; Masatsugu, Kimura; Isao, Teramoto; Ahmediin, Omar; Willis, Akhwale; James, Kongere; Akira, Kaneko; Ordanovich, Dariya; Tatem, Andrew; Penny, Melissa; Galactionova, Katya; Smith, Thomas; Bassat, Quique; Ogutu, Bernhards; DJimde, Abdoulaye; Stricker, Kirstin; Hamed, Kamal