日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Decarbonylative Strategy to Enhance Efficiency and Regioselectivity in Photocatalyzed Hydrogen Atom Transfer

脱羰策略提高光催化氢原子转移的效率和区域选择性

Cassera, Elena; Martini, Vittoria; Morlacci, Valerio; Abrami, Serena; Della Ca', Nicola; Ravelli, Davide; Fagnoni, Maurizio; Capaldo, Luca

Aldehydes as CO Releasing Molecules: In Situ and Ex Situ Giese Reactions and Palladium-Catalyzed Aminocarbonylations

醛类作为CO释放分子:原位和非原位Giese反应以及钯催化氨基羰基化反应

Cassera, Elena; Fagnoni, Maurizio

Characterization of β-Carboline Derivatives Reveals a High Barrier to Resistance and Potent Activity against Ring-Stage and DHA-Induced Dormant Plasmodium falciparum

β-咔啉衍生物的表征揭示了其对环状体和DHA诱导的休眠期恶性疟原虫具有高抗药性屏障和强效活性。

Haney, Reagan S; Butler, Joshua H; Wardlaw, Lyric A; Merino, Emilio F; Mendiola, Victoria; Cooper, Caitlin A; Mathew, Jopaul; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Kyle, Dennis E; Rizopoulos, Zaira; Baud, Delphine; Brand, Stephen; Totrov, Maxim; Carlier, Paul R; Cassera, Maria Belen

Stereospecific Resistance to N2-Acyl Tetrahydro-β-carboline Antimalarials Is Mediated by a PfMDR1 Mutation That Confers Collateral Drug Sensitivity

对N2-酰基四氢-β-咔啉类抗疟药的立体特异性耐药性是由PfMDR1突变介导的,该突变赋予了药物的附带敏感性。

Bremers, Emily K; Butler, Joshua H; Do Amaral, Leticia S; Merino, Emilio F; Almolhim, Hanan; Zhou, Bo; Baptista, Rodrigo P; Totrov, Maxim; Carlier, Paul R; Cassera, Maria Belen

Benzo-ring modification on Malaria Box hit MMV008138: effects on antimalarial potency and microsomal stability

疟疾靶点 MMV008138 的苯并环修饰:对抗疟疾效力和微粒体稳定性的影响

Ghavami, Maryam; Li, Haibo; Liu, Lixuan; Butler, Joshua H; Ding, Sha; Butschek, Grant J; Haney, Reagan S; Council-Troche, R McAlister; Grams, R Justin; Merino, Emilio F; Davis, Jennifer M; Totrov, Maxim; Cassera, Maria B; Carlier, Paul R

Machine Learning-Based Predictive Maintenance at Smart Ports Using IoT Sensor Data

基于机器学习的智能港口预测性维护:利用物联网传感器数据

Aslam, Sheraz; Navarro, Alejandro; Aristotelous, Andreas; Garro Crevillen, Eduardo; Martınez-Romero, Alvaro; Martínez-Ceballos, Álvaro; Cassera, Alessandro; Orphanides, Kyriacos; Herodotou, Herodotos; Michaelides, Michalis P

β-Carboline-3-carboxamide Antimalarials: Structure-Activity Relationship, ADME-Tox Studies, and Resistance Profiling

β-咔啉-3-甲酰胺类抗疟药:构效关系、ADME-Tox研究及耐药性分析

Mathew, Jopaul; Zhou, Bo; Haney, Reagan S; Kunz, Kevin A; Do Amaral, Leticia S; Roy Chowdhury, Rudraneel; Butler, Joshua H; Li, Haibo; Chakraborty, Amarraj J; Tabassum, Anika; Bremers, Emily K; Merino, Emilio F; Coyle, Rachael; Lee, Marcus C S; Baud, Delphine; Brand, Stephen; Totrov, Maxim; Cassera, Maria Belen; Carlier, Paul R

Positive events in psychotherapy: What do adolescents and young adults say is helpful?

心理治疗中的积极事件:青少年和年轻人认为哪些因素有帮助?

Cassera, Luisa; Calabrò, Alessia; Filippo, Aschieri

Cripowellins Pause Plasmodium falciparum Intraerythrocytic Development at the Ring Stage

克里波韦林蛋白可暂停恶性疟原虫环状体红细胞内发育

Butler, Joshua H; Painter, Heather J; Bremers, Emily K; Krai, Priscilla; Llinás, Manuel; Cassera, Maria B

Aptamer-Based Imaging of Polyisoprenoids in the Malaria Parasite

基于适体的疟原虫聚异戊二烯类化合物成像

Flavia M Zimbres, Emilio F Merino, Grant J Butschek, Joshua H Butler, Frédéric Ducongé, Maria B Cassera