日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

FlowMol3: flow matching for 3D de novo small-molecule generation

FlowMol3:用于三维从头小分子生成的流动匹配

Moumad, Aziz; Bouhaoui, Abderrazzak; Eddahmi, Mohammed; Catto, Marco; Bouissane, Latifa; Dunn, Ian; Koes, David R

Investigating Amphoteric 3,4'-Biscoumarin-Based ortho-[(Dialkylamino)methyl]phenols as Dual MAO and ChE Inhibitors

研究两性3,4'-双香豆素基邻-[(二烷基氨基)甲基]苯酚作为MAO和ChE双重抑制剂

Petrou, Anthi; Deruvo, Caterina; Purgatorio, Rosa; Lichitsky, Boris; Komogortsev, Andrey N; Kartsev, Victor G; de Candia, Modesto; Catto, Marco; Altomare, Cosimo D; Geronikaki, Athina

miRNAs as neuro-oncologic therapeutics: A narrative review

miRNA作为神经肿瘤治疗药物:综述

Pisani, Leonardo; Farina, Roberta; Soto-Otero, Ramon; Denora, Nunzio; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio; Mendez-Alvarez, Estefania; Altomare, Cosimo Damiano; Catto, Marco; Carotti, Angelo; Das, Nikita; Bhat, Samar; Fugo, Perrin; Dhawan, Andrew

Exploring pyrazolidinone and pyrazolidinedione scaffolds for Alzheimer's therapy: multitarget COX-2 inhibitors with anti-amyloid β, anti-tau, antioxidant, and neuroprotective activities

探索吡唑烷酮和吡唑烷二酮骨架在阿尔茨海默病治疗中的应用:具有抗β-淀粉样蛋白、抗tau蛋白、抗氧化和神经保护活性的多靶点COX-2抑制剂

Emad, Michael; Waheed, Reham; Mostafa, Zeinab; Darwish, Sarah S; Purgatorio, Rosa; Miniero, Daniela Valeria; De Palma, Annalisa; Cheng, Tzu-Peng; Chen, Yu-Cheng; Gabr, Moustafa; El Kerdawy, Ahmed M; Catto, Marco; Abadi, Ashraf H; Hwang, Tsong-Long; Abdel-Halim, Mohammad

Inflammaging and Immunosenescence in the Post-COVID Era: Small Molecules, Big Challenges

后新冠时代炎症衰老与免疫衰老:小分子,大挑战

Francavilla, Fabio; Intranuovo, Francesca; La Spada, Gabriella; Lacivita, Enza; Catto, Marco; Graps, Elisabetta Anna; Altomare, Cosimo Damiano

A Critical Appraisal of the Protective Activity of Polyphenolic Antioxidants against Iatrogenic Effects of Anticancer Chemotherapeutics

对多酚类抗氧化剂对抗癌化疗药物医源性损害的保护作用进行批判性评价

Purgatorio, Rosa; Boccarelli, Angelina; Pisani, Leonardo; de Candia, Modesto; Catto, Marco; Altomare, Cosimo D

Synthesis, Molecular Electron Density Theory Study, Molecular Docking, and Pharmacological Evaluation of New Coumarin-Sulfonamide-Nitroindazolyl-Triazole Hybrids as Monoamine Oxidase Inhibitors.

新型香豆素-磺酰胺-硝基吲唑基-三唑杂合物作为单胺氧化酶抑制剂的合成、分子电子密度理论研究、分子对接和药理学评价

Eddahmi Mohammed, La Spada Gabriella, Domingo Luis R, Vergoten Gérard, Bailly Christian, Catto Marco, Bouissane Latifa

Coumarin Derivative Hybrids: Novel Dual Inhibitors Targeting Acetylcholinesterase and Monoamine Oxidases for Alzheimer's Therapy.

香豆素衍生物杂合物:靶向乙酰胆碱酯酶和单胺氧化酶的新型双重抑制剂,用于阿尔茨海默病治疗

Żołek Teresa, Purgatorio Rosa, Kłopotowski Łukasz, Catto Marco, Ostrowska Kinga

Investigation on Novel E/Z 2-Benzylideneindan-1-One-Based Photoswitches with AChE and MAO-B Dual Inhibitory Activity.

对新型 E/Z 2-亚苄基茚满-1-酮基光开关及其 AChE 和 MAO-B 双重抑制活性的研究

Paolino Marco, de Candia Modesto, Purgatorio Rosa, Catto Marco, Saletti Mario, Tondo Anna Rita, Nicolotti Orazio, Cappelli Andrea, Brizzi Antonella, Mugnaini Claudia, Corelli Federico, Altomare Cosimo D

A twenty-year journey exploring coumarin-based derivatives as bioactive molecules

二十年来,我们一直在探索香豆素衍生物作为生物活性分子的研究历程

Pisani, Leonardo; Catto, Marco; Muncipinto, Giovanni; Nicolotti, Orazio; Carrieri, Antonio; Rullo, Mariagrazia; Stefanachi, Angela; Leonetti, Francesco; Altomare, Cosimo