日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Thioquinazolinones as Antituberculosis Agents Targeting Phosphopantetheinyl Transferase

硫代喹唑啉酮类化合物作为靶向磷酸泛酰巯基转移酶的抗结核药物

Singh, Amrita; Zwerneman, Logan T; Planck, Kyle; Kaneko, Takushi; Perkowski, Andrew J; Suh, Christine M; Alex, Alexander; Bean, James; Burns-Huang, Kristin; Zhang, David; Boshoff, Helena I M; Roubert, Christine; Krieger, Inna; Gardner, Mark; Cautain, Bastien; Cooper, Christopher B; Tanvir, Zaid; Sacchettini, James; Gold, Ben S; Rhee, Kyu Y; Fotouhi, Nader; Nathan, Carl F; Aubé, Jeffrey

Acetylenic Fatty Acids and Stilbene Glycosides Isolated from Santalum yasi Collected from the Fiji Islands.

从斐济群岛采集的檀香树中分离得到的乙炔脂肪酸和芪类糖苷。

Maqbali Khalid Al, Vuiyasawa Miriama, Gube-Ibrahim Mercy Ayinya, Sewariya Shubham, Balat Clément, Helland Kirsti, Garcia-Sorribes Tamar, Cruz Mercedes de la, Cautain Bastien, Andersen Jeanette Hammer, Reyes Fernando, Tabudravu Jioji N

Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.

将 raltitrexed 从癌细胞胸苷酸合成酶重定向到结核分枝杆菌磷酸泛酰巯基转移酶

Singh Amrita, Ottavi Samantha, Krieger Inna, Planck Kyle, Perkowski Andrew, Kaneko Takushi, Davis Andrew M, Suh Christine, Zhang David, Goullieux Laurent, Alex Alexander, Roubert Christine, Gardner Mark, Preston Marian, Smith Dave M, Ling Yan, Roberts Julia, Cautain Bastien, Upton Anna, Cooper Christopher B, Serbina Natalya, Tanvir Zaid, Mosior John, Ouerfelli Ouathek, Yang Guangli, Gold Ben S, Rhee Kyu Y, Sacchettini James C, Fotouhi Nader, Aubé Jeffrey, Nathan Carl

Small Molecule Inhibitors of CRM1

CRM1的小分子抑制剂

Ferreira, Bibiana I; Cautain, Bastien; Grenho, Inês; Link, Wolfgang

Structural Elucidation of Antibiotic TKR2999, an Antifungal Lipodepsipeptide Isolated from the Fungus Foliophoma fallens

从落叶孢霉中分离得到的抗真菌脂肽类抗生素TKR2999的结构解析

Crespo, Gloria; Pérez-Victoria, Ignacio; Ortiz-López, Francisco Javier; González-Menéndez, Víctor; de la Cruz, Mercedes; Cautain, Bastien; Sánchez, Pilar; Vicente, Francisca; Genilloud, Olga; Reyes, Fernando

First evidence of anticancer and antimicrobial activity in Mediterranean mesopelagic species

首次发现地中海中层鱼类具有抗癌和抗菌活性

Lauritano, Chiara; Martínez, Kevin A; Battaglia, Pietro; Granata, Antonia; de la Cruz, Mercedes; Cautain, Bastien; Martín, Jesús; Reyes, Fernando; Ianora, Adrianna; Guglielmo, Letterio

Amphidinol 22, a New Cytotoxic and Antifungal Amphidinol from the Dinoflagellate Amphidinium carterae

Amphidinol 22,一种来自甲藻 Amphidinium carterae 的新型细胞毒性和抗真菌 Amphidinol 化合物

Martínez, Kevin A; Lauritano, Chiara; Druka, Dana; Romano, Giovanna; Grohmann, Teresa; Jaspars, Marcel; Martín, Jesús; Díaz, Caridad; Cautain, Bastien; de la Cruz, Mercedes; Ianora, Adrianna; Reyes, Fernando

Cytotoxic Furanoditerpenes from the Sponge Spongia tubulifera Collected in the Mexican Caribbean

从墨西哥加勒比海地区采集的管状海绵(Spongia tubulifera)中提取的细胞毒性呋喃二萜类化合物

Pech-Puch, Dawrin; Rodríguez, Jaime; Cautain, Bastien; Sandoval-Castro, Carlos Alfredo; Jiménez, Carlos

New Napyradiomycin Analogues from Streptomyces sp. Strain CA-271078

来自链霉菌属 CA-271078 菌株的新型萘吡啶霉素类似物

Carretero-Molina, Daniel; Ortiz-López, Francisco Javier; Martín, Jesús; Oves-Costales, Daniel; Díaz, Caridad; de la Cruz, Mercedes; Cautain, Bastien; Vicente, Francisca; Genilloud, Olga; Reyes, Fernando

Bioactivities and Extract Dereplication of Actinomycetales Isolated From Marine Sponges

从海洋海绵中分离的放线菌的生物活性和提取物去重复性

Santos, José D; Vitorino, Inês; De la Cruz, Mercedes; Díaz, Caridad; Cautain, Bastien; Annang, Frederick; Pérez-Moreno, Guiomar; Gonzalez Martinez, Ignacio; Tormo, Jose R; Martín, Jesús M; Urbatzka, Ralph; Vicente, Francisca M; Lage, Olga M