日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fine-tuning 5-HT(7) receptor selectivity, inverse agonism, and metabolic stability of new (aryloxy)ethyl-piperidines toward antidepressant and pro-cognitive properties

通过微调新型(芳氧基)乙基哌啶类化合物的5-HT(7)受体选择性、反向激动作用和代谢稳定性,探索其抗抑郁和促认知特性。

Canale, Vittorio; Blicharz-Futera, Klaudia; Bijata, Monika; Cavalco, Natalie G; Partyka, Anna; Stefaniak, Matylda; Kamiński, Michał; Satała, Grzegorz; Warszycki, Dawid; Lanham, Janelle K; Gołębiowska, Joanna; Gawlik, Maciej; Smolik, Magdalena; Bijata, Krystian; Jastrzębska-Więsek, Magdalena; Kurczab, Rafał; Bojarski, Andrzej J; Walczak, Maria; McCorvy, John D; Włodarczyk, Jakub; Popik, Piotr; Zajdel, Paweł

Discovery of Highly Selective 5-HT(2A) Agonists Using Structure-Guided Design

利用结构导向设计发现高选择性5-HT(2A)激动剂

Fenske, Tyler G; McKee, John L; Cavalco, Natalie G; Schalk, Serena S; Bonniwell, Emma M; Lammers, Josie C; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D

Serotonin 5-HT(2C) Receptor Signaling Analysis Reveals Psychedelic Biased Agonism

血清素 5-HT(2C) 受体信号分析揭示迷幻剂偏向性激动作用

Bonniwell, Emma M; Alabdali, Rana; Hennessey, Joseph J; McKee, John L; Cavalco, Natalie G; Lammers, Josie C; Moore, Ethan J; Franchini, Luca; Orlandi, Cesare; McCorvy, John D

Functional profiling of the G protein-coupled receptor C3aR1 reveals ligand-mediated biased agonism

蛋白偶联受体 C3aR1 的功能分析揭示了配体介导的偏向激动作用

Pedro Rodriguez, Lauren J Laskowski, Jean Pierre Pallais, Hailey A Bock, Natalie G Cavalco, Emilie I Anderson, Maggie M Calkins, Maria Razzoli, Yuk Y Sham, John D McCorvy, Alessandro Bartolomucci

Serotonin 1A Receptors Modulate Serotonin 2A Receptor-Mediated Behavioral Effects of 5-Methoxy-N,N-dimethyltryptamine Analogs in Mice

血清素1A受体调节5-甲氧基-N,N-二甲基色胺类似物在小鼠体内的血清素2A受体介导的行为效应

Glatfelter, Grant C; Clark, Allison A; Cavalco, Natalie G; Landavazo, Antonio; Partilla, John S; Naeem, Marilyn; Golen, James A; Chadeayne, Andrew R; Manke, David R; Blough, Bruce E; McCorvy, John D; Baumann, Michael H

Gonadal hormones and sex chromosome complement differentially contribute to ethanol intake, preference, and relapse-like behaviour in four core genotypes mice

性腺激素和性染色体组成对四种核心基因型小鼠的乙醇摄入量、偏好和复发样行为的影响各不相同。

Sneddon, Elizabeth A; Rasizer, Lindsay N; Cavalco, Natalie G; Jaymes, Asa H; Ostlie, Noah J; Minshall, Brianna L; Masters, Brianna M; Hughes, Michael R; Hrncir, Haley; Arnold, Arthur P; Radke, Anna K