日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploiting the Cryptic αD Pocket of Casein Kinase 2α (CK2α) to Deliver Highly Potent and Selective Type 1 Inhibitors.

利用酪蛋白激酶 2α (CK2α) 的隐蔽 αD 口袋递送高效选择性 1 型抑制剂。

Glossop Paul A, Brear Paul, Wright Susanne, Flanagan Neil, Glossop Melanie S, Lane Charlotte A L, Butt Richard P, Spring David R, Hyvönen Marko, Cawkill Darren

Preclinical trial of a MAP4K4 inhibitor to reduce infarct size in the pig: does cardioprotection in human stem cell-derived myocytes predict success in large mammals?

MAP4K4 抑制剂减少猪梗塞面积的临床前试验:人类干细胞衍生的心肌细胞中的心脏保护作用是否可以预示大型哺乳动物的成功?

Maaike Te Lintel Hekkert #, Gary Newton #, Kathryn Chapman, Rehan Aqil, Robert Downham, Robert Yan, Daphne Merkus, Gavin Whitlock, Charlotte A L Lane, Darren Cawkill, Trevor Perrior, Dirk J Duncker #, Michael D Schneider #

Author Correction: Exploring use of unsupervised clustering to associate signaling profiles of GPCR ligands to clinical response

作者更正:探索使用无监督聚类将GPCR配体的信号谱与临床反应关联起来

Benredjem, Besma; Gallion, Jonathan; Pelletier, Dennis; Dallaire, Paul; Charbonneau, Johanie; Cawkill, Darren; Nagi, Karim; Gosink, Mark; Lukasheva, Viktoryia; Jenkinson, Stephen; Ren, Yong; Somps, Christopher; Murat, Brigitte; Van Der Westhuizen, Emma; Le Gouill, Christian; Lichtarge, Olivier; Schmidt, Anne; Bouvier, Michel; Pineyro, Graciela

Exploring use of unsupervised clustering to associate signaling profiles of GPCR ligands to clinical response

探索使用无监督聚类将 GPCR 配体的信号传导特征与临床反应关联起来

Besma Benredjem, Jonathan Gallion, Dennis Pelletier, Paul Dallaire, Johanie Charbonneau, Darren Cawkill, Karim Nagi, Mark Gosink, Viktoryia Lukasheva, Stephen Jenkinson, Yong Ren, Christopher Somps, Brigitte Murat, Emma Van Der Westhuizen, Christian Le Gouill, Olivier Lichtarge, Anne Schmidt, Michel

Dementia, post-traumatic stress disorder and major depressive disorder: a review of the mental health risk factors for dementia in the military veteran population

痴呆症、创伤后应激障碍和重度抑郁症:退伍军人群体痴呆症心理健康风险因素综述

Rafferty, L A; Cawkill, P E; Stevelink, S A M; Greenberg, K; Greenberg, N

Plate-Based Phenotypic Screening for Pain Using Human iPSC-Derived Sensory Neurons

使用人类 iPSC 衍生的感觉神经元进行基于培养板的疼痛表型筛选

Peter Stacey, Anne Mai Wassermann, Laura Kammonen, Emma Impey, Anna Wilbrey, Darren Cawkill

Synergistic malaria vaccine combinations identified by systematic antigen screening

通过系统抗原筛选确定协同疟疾疫苗组合

Leyla Y Bustamante, Gareth T Powell, Yen-Chun Lin, Michael D Macklin, Nadia Cross, Alison Kemp, Paula Cawkill, Theo Sanderson, Cecile Crosnier, Nicole Muller-Sienerth, Ogobara K Doumbo, Boubacar Traore, Peter D Crompton, Pietro Cicuta, Tuan M Tran, Gavin J Wright, Julian C Rayner

Biased ligand quantification in drug discovery: from theory to high throughput screening to identify new biased μ opioid receptor agonists

药物发现中的偏向性配体定量:从理论到高通量筛选以鉴定新的偏向性μ阿片受体激动剂

Winpenny, David; Clark, Mellissa; Cawkill, Darren