Identification of N-(quinolin-8-yl)benzenesulfonamides as agents capable of down-regulating NFkappaB activity within two separate high-throughput screens of NFkappaB activation
在两项独立的高通量NF-κB激活筛选中,鉴定出N-(喹啉-8-基)苯磺酰胺类化合物能够下调NF-κB活性。
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2007.10.100
Xie, Yuli; Deng, ShiXian; Thomas, Craig J; Liu, Yidong; Zhang, Ya-Qin; Rinderspacher, Alison; Huang, Wenwei; Gong, Gangli; Wyler, Michael; Cayanis, Efithia; Aulner, Nathalie; Többen, Udo; Chung, Caty; Pampou, Sergey; Southall, Noel; Vidović, Dusica; Schürer, Stephan; Branden, Lars; Davis, R Eric; Staudt, Louis M; Inglese, James; Austin, Christopher P; Landry, Donald W; Smith, Deborah H; Auld, Douglas S