日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Flexibility-tuning of dual-display DNA-encoded chemical libraries facilitates cyclic peptide ligand discovery

双显示DNA编码化学库的灵活性调控促进了环肽配体的发现

Petrov, Dimitar; Plais, Louise; Schira, Kristina; Cai, Junyu; Keller, Michelle; Lessing, Alice; Bassi, Gabriele; Cazzamalli, Samuele; Neri, Dario; Gloger, Andreas; Scheuermann, Jörg

Phenylalanine-Based DNA-Encoded Chemical Libraries for the Discovery of Potent and Selective Small Organic Ligands Against Markers of Cancer and Immune Cells

基于苯丙氨酸的DNA编码化学库用于发现针对癌症和免疫细胞标志物的高效选择性小分子有机配体

Migliorini, Francesca; Ciamarone, Andrea; Dakhel Plaza, Sheila; Georgiev, Tony; Mascellani, Marta; Sabato, Emanuela; Vistoli, Giulio; Biancofiore, Ilaria; Favalli, Nicholas; Puca, Emanuele; Oehler, Sebastian; Neri, Dario; Cazzamalli, Samuele

Expression patterns of fibroblast activation protein and extra-domain B fibronectin in canine malignant tumors.

犬恶性肿瘤中成纤维细胞活化蛋白和外域B纤连蛋白的表达模式。

Dell'Aere Silvia, Gariboldi Elisa Maria, Ubiali Alessandra, Ferrari Roberta, Auletta Luigi, Bocci Matilde, Galbiati Andrea, Gilardoni Ettore, Rotta Giulia, Balbi Valentina, Bianchi Gaia Beatrice Maria, Verdi Alessandra, Neri Dario, Cazzamalli Samuele, Stefanello Damiano, Roccabianca Paola

DNA-encoded chemical libraries enable the discovery of potent PSMA-ligands with substantially reduced affinity towards the GCPIII anti-target

DNA编码的化学库能够发现对GCPIII反靶标亲和力显著降低的高效PSMA配体。

Lucaroni, Laura; Oehler, Sebastian; Georgiev, Tony; Müller, Marco; Bocci, Matilde; De Luca, Roberto; Favalli, Nicholas; Neri, Dario; Cazzamalli, Samuele; Prati, Luca

Impact of library input on the hit discovery rate in DNA-encoded chemical library selections

文库输入对DNA编码化学文库筛选中命中发现率的影响

Puglioli, Sara; Oehler, Sebastian; Prati, Luca; Scheuermann, Jörg; Bassi, Gabriele; Cazzamalli, Samuele; Neri, Dario; Favalli, Nicholas

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker

利用体外质谱法对带有蛋白酶可切割和酸不稳定连接子的抗体-瑞喹莫德偶联物进行生物分布分析

Bisbal Lopez, Lydia; Ravazza, Domenico; Bocci, Matilde; Zana, Aureliano; Principi, Lucrezia; Dakhel Plaza, Sheila; Galbiati, Andrea; Gilardoni, Ettore; Scheuermann, Jörg; Neri, Dario; Pignataro, Luca; Gennari, Cesare; Cazzamalli, Samuele; Dal Corso, Alberto

Tumor-Targeted Interleukin 2 Boosts the Anticancer Activity of FAP-Directed Radioligand Therapeutics

肿瘤靶向白细胞介素 2 可增强 FAP 靶向放射性配体疗法的抗癌活性

Galbiati, Andrea; Dorten, Paulina; Gilardoni, Ettore; Gierse, Florian; Bocci, Matilde; Zana, Aureliano; Mock, Jacqueline; Claesener, Michael; Cufe, Juela; Büther, Florian; Schäfers, Klaus; Hermann, Sven; Schäfers, Michael; Neri, Dario; Cazzamalli, Samuele; Backhaus, Philipp

Automated Radiosynthesis, Preliminary In Vitro/In Vivo Characterization of OncoFAP-Based Radiopharmaceuticals for Cancer Imaging and Therapy

基于OncoFAP的放射性药物在癌症成像和治疗中的自动化放射合成、初步体外/体内表征

Bartoli, Francesco; Elsinga, Philip; Nazario, Luiza Reali; Zana, Aureliano; Galbiati, Andrea; Millul, Jacopo; Migliorini, Francesca; Cazzamalli, Samuele; Neri, Dario; Slart, Riemer H J A; Erba, Paola Anna

A Dimeric FAP-Targeting Small-Molecule Radioconjugate with High and Prolonged Tumor Uptake

一种靶向FAP的二聚体小分子放射性偶联物,具有高且持久的肿瘤摄取

Galbiati, Andrea; Zana, Aureliano; Bocci, Matilde; Millul, Jacopo; Elsayed, Abdullah; Mock, Jacqueline; Neri, Dario; Cazzamalli, Samuele

Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications

立体选择性和区域选择性明确的DNA编码化学库能够实现高效的肿瘤靶向应用

Favalli, Nicholas; Bassi, Gabriele; Pellegrino, Christian; Millul, Jacopo; De Luca, Roberto; Cazzamalli, Samuele; Yang, Su; Trenner, Anika; Mozaffari, Nour L; Myburgh, Renier; Moroglu, Mustafa; Conway, Stuart J; Sartori, Alessandro A; Manz, Markus G; Lerner, Richard A; Vogt, Peter K; Scheuermann, Jörg; Neri, Dario