Asymmetric Engagement of Dimeric CRL3 (KBTBD4) by the Molecular Glue UM171 Licenses Degradation of HDAC1/2 Complexes
分子胶UM171与二聚体CRL3(KBTBD4)的不对称结合促进HDAC1/2复合物的降解
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doi:10.1101/2024.05.14.593897
Yeo, Megan Jr; Zhang, Olivia; Xie, Xiaowen; Nam, Eunju; Payne, Neil Connor; Gosavi, Pallavi M; Kwok, Hui Si; Iram, Irtiza; Lee, Ceejay; Li, Jiaming; Chen, Nicholas J; Jiang, Hanjie; Wang, Zhipeng A; Lee, Kwangwoon; Mao, Haibin; Harry, Stefan A; Barakat, Idris A; Takahashi, Mariko; Waterbury, Amanda L; Barone, Marco; Mattevi, Andrea; Bar-Peled, Liron; Cole, Philip A; Mazitschek, Ralph; Liau, Brian B; Zheng, Ning