日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents

首创的双重PDGFR/碳酸酐酶IX/XII抑制剂:6,7-二甲氧基喹啉磺酰胺类药物作为有前景的抗白血病药物

Roshdy, Eslam; Řezníčková, Eva; Elbadawi, Mostafa M; Celik, Ismail; Giovannuzzi, Simone; Veselá, Denisa; Vojáčková, Veronika; Krňávková, Petra; Nocentini, Alessio; Supuran, Claudiu T; Kryštof, Vladimír; Eldehna, Wagdy M; Abe, Manabu

Evaluation of oxadiazole-N-phenylacetamide conjugates as VEGFR-2 inhibitors and apoptosis inducers: design, synthesis, anti-proliferative assessment, molecular docking, and dynamics studies

评价恶二唑-N-苯基乙酰胺缀合物作为VEGFR-2抑制剂和细胞凋亡诱导剂的活性:设计、合成、抗增殖活性评估、分子对接和动力学研究

Otify, Islam I; Ayyad, Rezk R A; Celik, Ismail; Sakr, Helmy; Elwan, Alaa

Immunoinformatics-driven multi-epitope vaccine design targeting PSMA, STEAP1, and B7H3 for prostate cancer

免疫信息学驱动的多表位疫苗设计,靶向PSMA、STEAP1和B7H3,用于治疗前列腺癌

Runtunuwu, Stefanus Vicky Bernhard Elisa; Tallei, Trina Ekawati; Kim, Hyo Jeong; Park, Moon Nyeo; Celik, Ismail; Kirilmaz, Burak; Turalaki, Grace Lendawati Amelia; Fatimawali, Fatimawali; Tendean, Lydia Estelina Naomi; Kaseke, Martha Marie; Makawaehe, Dionisius Rafael; Rambi, Elne Vieke; Kim, Bonglee

Design, Synthesis, and Biological Evaluation of BODIPY-Caged Resiquimod as a Dual-Acting Phototherapeutic.

BODIPY笼状瑞喹莫特作为双效光疗剂的设计、合成和生物学评价

Roshdy Eslam, Taniguchi Haruto, Nakamura Yoki, Takahashi Haruko, Kikuchi Yutaka, Celik Ismail, Mohammed Elsayed S I, Ishihara Yasuhiro, Morioka Norimitsu, Abe Manabu

Synthesis of Thiazole-methylsulfonyl Derivatives, X-ray Study, and Investigation of Their Carbonic Anhydrase Activities: In Vitro and In Silico Potentials

噻唑甲基磺酰衍生物的合成、X射线研究及其碳酸酐酶活性研究:体外和计算机模拟潜力

Maryam, Zahra; Işık, Ayşen; Bağcı, Emine Rana; Yıldız, Maksut; Ünver, Hakan; Kocyigit, Ümit M; Kırılmaz, Burak; Celik, Ismail; Acar Çevik, Ulviye; Özkay, Yusuf; Kaplancıklı, Zafer Asım

Ternary Complex Modeling, Induced Fit Docking and Molecular Dynamics Simulations as a Successful Approach for the Design of VHL-Mediated PROTACs Targeting the Kinase FLT3

三元复合物建模、诱导契合对接和分子动力学模拟是设计靶向激酶FLT3的VHL介导的PROTAC的成功方法

Nassar, Husam; Sarnow, Anne-Christin; Celik, Ismail; Abdelsalam, Mohamed; Robaa, Dina; Sippl, Wolfgang

Molecular mechanisms of phytoconstituents from selected Egyptian plants against non-small cell lung cancer using integrated in vitro network pharmacology and molecular docking approach

利用整合体外网络药理学和分子对接方法,研究埃及部分植物成分抗非小细胞肺癌的分子机制

Shaala, Lamiaa A; Youssef, Diaa T A; Ramadan, Mahmoud A; Khalifa, Azza A; Ibrahim, Reham S; Valeriote, Fred; Celik, Ismail; Dawood, Hend M

Investigating Potential Cancer Therapeutics: Insight into Histone Deacetylases (HDACs) Inhibitions

探索潜在的癌症治疗方法:深入了解组蛋白去乙酰化酶(HDACs)抑制剂

Ahmad, Basharat; Saeed, Aamir; Al-Amery, Ahmed; Celik, Ismail; Ahmed, Iraj; Yaseen, Muhammad; Khan, Imran Ahmad; Al-Fahad, Dhurgham; Bhat, Mashooq Ahmad

A network pharmacology approach to elucidate the anti-inflammatory and antioxidant effects of bitter leaf (Vernonia amygdalina Del.)

利用网络药理学方法阐明苦叶(Vernonia amygdalina Del.)的抗炎和抗氧化作用

Sailah, Illah; Tallei, Trina E; Safitri, Linda; Tamala, Yulianida; Halimatushadyah, Ernie; Ekatanti, Dewi; Maulydia, Nur B; Celik, Ismail

Epigallocatechin-3-Gallate Therapeutic Potential in Cancer: Mechanism of Action and Clinical Implications

表没食子儿茶素-3-没食子酸酯在癌症治疗中的潜力:作用机制和临床意义

Kciuk, Mateusz; Alam, Manzar; Ali, Nemat; Rashid, Summya; Głowacka, Pola; Sundaraj, Rajamanikandan; Celik, Ismail; Yahya, Esam Bashir; Dubey, Amit; Zerroug, Enfale; Kontek, Renata