日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: BET inhibitor-based combinations targeting novel dependencies in MECOM-rearranged (r) AML

更正:基于BET抑制剂的联合疗法靶向MECOM重排(r) AML中的新型依赖性

Birdwell, Christine E; Fiskus, Warren; Mill, Christopher P; Kadia, Tapan M; Daver, Naval; DiNardo, Courtney D; Sasaki, Koji; Davis, John A; Das, Kaberi; Hou, Hanxi; Jain, Antrix; Malovannaya, Anna; Flores, Lauren B; Pourebrahim, Rasoul; Yuan, Selina; Su, Xiaoping; Ceribelli, Michele; Bhalla, Kapil N

BET inhibitor-based combinations targeting novel dependencies in MECOM-rearranged (r) AML

基于BET抑制剂的联合疗法靶向MECOM重排(r) AML中的新型依赖性

Birdwell, Christine E; Fiskus, Warren; Mill, Christopher P; Kadia, Tapan M; Daver, Naval; DiNardo, Courtney D; Sasaki, Koji; Davis, John A; Das, Kaberi; Hou, Hanxi; Jain, Antrix; Malovannaya, Anna; Flores, Lauren B; Pourebrahim, Rasoul; Yuan, Selina; Su, Xiaoping; Ceribelli, Michele; Bhalla, Kapil N

Targeting of IRAK4 and GSPT1 enhances therapeutic efficacy in AML via c-Myc destabilization.

靶向 IRAK4 和 GSPT1 可通过 c-Myc 不稳定增强 AML 的治疗效果

Vick Eric J, Hassan Aishlin, Choi Kwangmin, Bennett Joshua, Muto Tomoya, Clough Courtnee A, Culver-Cochran Ashley E, Hueneman Kathleen, Bolanos Lyndsey C, Wunderlich Mark, Zhang Xiaohu, McKnight Crystal, Ceribelli Michele, Holland David, Klumpp-Thomas Carleen, Greis Kenneth D, Thomas Craig J, Starczynowski Daniel T

Discovery and Optimization of LATS1 and LATS2 Kinase Inhibitors for Use in Regenerative Medicine

LATS1和LATS2激酶抑制剂的发现和优化及其在再生医学中的应用

Morris, Patrick J; Duveau, Damien Y; Ceribelli, Michele; Tosto, Frances Anne; Love, Dara N; Scherer, Bridget S; Tao, Dingyin; Fang, Yuhong; Evsen, Lale; Kotler, Samuel A; LeClair, Christopher A; Rai, Ganesha; Thomas, Craig J; Hoyt, Scott B

Targeting NAD+ Metabolism Vulnerability in FH-Deficient Hereditary Leiomyomatosis and Renal Cell Carcinoma with the Novel NAMPT Inhibitor OT-82.

利用新型 NAMPT 抑制剂 OT-82 靶向 FH 缺陷型遗传性平滑肌瘤病和肾细胞癌中的 NAD+ 代谢脆弱性

Najera Susana S, Ricketts Christopher J, Schmidt Laura S, Medina Julia I, Saito Keita, Ileva Lilia, Brender Jeffrey R, James Amy M, Peer Cody J, Gouker Brad, Karim Baktiar O, Chernova Olga, Wells Catherine, Wei Ming-Hui, Yang Youfeng, Zhang Xiaohu, Klumpp-Thomas Carleen, Travers Jameson, Chen Lu, Wilson Kelli M, Issaq Sameer H, Figg William D, Difilippantonio Simone, Kalen Joseph D, Krishna Murali C, Thomas Craig J, Ceribelli Michele, Heske Christine M, Crooks Daniel R, Meier Jordan L

An Assessment of Kinase Selectivity, Enzyme Inhibition Kinetics and in Vitro Activity for Several Bruton Tyrosine Kinase (BTK) Inhibitors

对几种布鲁顿酪氨酸激酶(BTK)抑制剂的激酶选择性、酶抑制动力学和体外活性进行评估

Corrionero, Ana; Zhang, Xiaohu; Alfonso, Patricia; Morris, Patrick J; Klumpp-Thomas, Carleen; Melani, Christopher; McKnight, Crystal; Phelan, James D; Holland, David; Wilson, Kelli; Hoyt, Scott B; Roschewski, Mark; Tonge, Peter J; Wilson, Wyndham; Ceribelli, Michele; Staudt, Louis M; Thomas, Craig J

Direct Co-Targeting of Bcl-xL and Mcl-1 Exhibits Synergistic Effects in AR-V7-Expressing CRPC Models.

Bcl-xL 和 Mcl-1 的直接共同靶向在 AR-V7 表达的 CRPC 模型中表现出协同效应

Brim Benjamin C, Leon Andres F, Beatson Erica L, Kindrick Jessica D, Bhadresha Kinjal, Zhang Xiaohu, Napoli Giulia C, Risdon Emily N, Schmidt Keith T, Wilson Kelli M, McKnight Crystal, Beck Erin, Klumpp-Thomas Carleen, Ceribelli Michele, Yin JuanJuan, Sowalsky Adam G, Price Douglas K, Chau Cindy H, Thomas Craig J, Figg William D

Multiple Epigenetic Mechanisms Functionally Cooperate to Silence Expression of Somatostatin Receptor Type 2 in Pancreatic Neuroendocrine Tumors

多种表观遗传机制协同作用,抑制胰腺神经内分泌肿瘤中生长抑素受体2型的表达

Madigan, James P; Andrews, Stephen G; Farrell, Rivka B; Forsythe, Steven D; Sharma, Rupali; Ceribelli, Michele; Thomas, Craig J; Shamsian, Kimia N; Lin, Shinjen; Cheng, Ken Chih-Chien; Sadowski, Samira M

Combination Targeted Therapy in Relapsed Diffuse Large B-Cell Lymphoma

复发性弥漫性大B细胞淋巴瘤的联合靶向治疗

Melani, Christopher; Lakhotia, Rahul; Pittaluga, Stefania; Phelan, James D; Huang, Da Wei; Wright, George; Simard, Jillian; Muppidi, Jagan; Thomas, Craig J; Ceribelli, Michele; Tosto, Frances A; Yang, Yandan; Xu, Weihong; Davies-Hill, Theresa; Pack, Svetlana D; Peer, Cody J; Arisa, Oluwatobi; Mena, Esther; Lindenberg, Liza; Bergvall, Ethan; Portell, Craig A; Farah, Rafic J; Lee, Seung Tae; Pradhan, Amynah; Morrison, Candis; Tadese, Atekelt; Juanitez, Anna Marie; Lu, Crystal; Jacob, Allison; Simmons, Heidi; Figg, William D; Steinberg, Seth M; Jaffe, Elaine S; Roschewski, Mark; Staudt, Louis M; Wilson, Wyndham H

CellMinerCDB: NCATS Is a Web-Based Portal Integrating Public Cancer Cell Line Databases for Pharmacogenomic Explorations

CellMinerCDB:NCATS 是一个基于网络的门户网站,整合了用于药物基因组学探索的公共癌症细胞系数据库。

Reinhold, William C; Wilson, Kelli; Elloumi, Fathi; Bradwell, Katie R; Ceribelli, Michele; Varma, Sudhir; Wang, Yanghsin; Duveau, Damien; Menon, Nikhil; Trepel, Jane; Zhang, Xiaohu; Klumpp-Thomas, Carleen; Micheal, Samuel; Shinn, Paul; Luna, Augustin; Thomas, Craig; Pommier, Yves