Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor
将二苯二氮卓类药物优化为有效且选择性的变构 PAK1 抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/acsmedchemlett.5b00102
Alexei S Karpov, Payman Amiri, Cornelia Bellamacina, Marie-Helene Bellance, Werner Breitenstein, Dylan Daniel, Regis Denay, Doriano Fabbro, Cesar Fernandez, Inga Galuba, Stephanie Guerro-Lagasse, Sascha Gutmann, Linda Hinh, Wolfgang Jahnke, Julia Klopp, Albert Lai, Mika K Lindvall, Sylvia Ma, Henrik
