日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Alternative splicing in the DBD linker region of p63 modulates binding to DNA and iASPP in vitro.

p63 的 DBD 连接区中的选择性剪接可调节其在体外与 DNA 和 iASPP 的结合

Lotz Rebecca, Osterburg Christian, Chaikuad Apirat, Weber Sabrina, Akutsu Masato, Machel Anne Christin, Beyer Ulrike, Gebel Jakob, Löhr Frank, Knapp Stefan, Dobbelstein Matthias, Lu Xin, Dötsch Volker

Structural analysis of TRIM family PRYSPRY domains and its implications for E3-ligand design

TRIM家族PRYSPRY结构域的结构分析及其对E3配体设计的影响

Zhubi, Rezart; Chaikuad, Apirat; Muñoz Sosa, Christian J; Joerger, Andreas C; Knapp, Stefan

A twist in the tale: shifting from covalent targeting of a tyrosine in JAK3 to a lysine in MK2

剧情出现转折:从JAK3中酪氨酸的共价靶向转变为MK2中赖氨酸的共价靶向。

Hillebrand, Laura; Wang, Guiqun; Rasch, Alexander; Masberg, Benedikt; Chaikuad, Apirat; Kronenberger, Thales; Günther, Ellen; Forster, Michael; Poso, Antti; Lämmerhofer, Michael; Laufer, Stefan A; Knapp, Stefan; Gehringer, Matthias

Synthesis and Characterization of ULK1/2 Kinase Inhibitors that Inhibit Autophagy and Upregulate Expression of Major Histocompatibility Complex I for the Treatment of Non-Small Cell Lung Cancer

合成和表征抑制自噬并上调主要组织相容性复合体I表达的ULK1/2激酶抑制剂,用于治疗非小细胞肺癌

Layng, Fabiana Izidro A L; Ren, Huiyu; Bakas, Nicole A; Panickar, Dhanya R; Lambert, Lester J; Celeridad, Maria; Wu, Jiaqian; De Backer, Laurent; Chandrachud, Preeti; Limpert, Allison S; Vamos, Mitchell; Chaikuad, Apirat; Verdugo, Betsaida B; Hagan, Patrick M; Brun, Sonja N; Tautz, Lutz; Knapp, Stefan; Shaw, Reuben J; Salvesen, Guy S; Sheffler, Douglas J; Cosford, Nicholas D P

Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation

靶向替代维生素E代谢物结合位点可实现非经典PPARγ调节

Arifi, Silvia; Marschner, Julian A; Pollinger, Julius; Isigkeit, Laura; Heitel, Pascal; Kaiser, Astrid; Obeser, Lennart; Höfner, Georg; Proschak, Ewgenij; Knapp, Stefan; Chaikuad, Apirat; Heering, Jan; Merk, Daniel

Structural insights into a regulatory mechanism of FIR RRM1-FUSE interaction

FIR RRM1-FUSE相互作用调控机制的结构解析

Ni, Xiaomin; Joerger, Andreas C; Chaikuad, Apirat; Knapp, Stefan

Image-Based Annotation of Chemogenomic Libraries for Phenotypic Screening

基于图像的化学基因组文库表型筛选注释

Tjaden, Amelie; Chaikuad, Apirat; Kowarz, Eric; Marschalek, Rolf; Knapp, Stefan; Schröder, Martin; Müller, Susanne

Target 2035 - update on the quest for a probe for every protein

2035年目标——为每种蛋白质寻找探针的最新进展

Müller, Susanne; Ackloo, Suzanne; Al Chawaf, Arij; Al-Lazikani, Bissan; Antolin, Albert; Baell, Jonathan B; Beck, Hartmut; Beedie, Shaunna; Betz, Ulrich A K; Bezerra, Gustavo Arruda; Brennan, Paul E; Brown, David; Brown, Peter J; Bullock, Alex N; Carter, Adrian J; Chaikuad, Apirat; Chaineau, Mathilde; Ciulli, Alessio; Collins, Ian; Dreher, Jan; Drewry, David; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Frye, Stephen V; Fuchs, Stephen M; Hall, Matthew D; Hartung, Ingo V; Hillisch, Alexander; Hitchcock, Stephen H; Homan, Evert; Kannan, Natarajan; Kiefer, James R; Knapp, Stefan; Kostic, Milka; Kubicek, Stefan; Leach, Andrew R; Lindemann, Sven; Marsden, Brian D; Matsui, Hisanori; Meier, Jordan L; Merk, Daniel; Michel, Maurice; Morgan, Maxwell R; Mueller-Fahrnow, Anke; Owen, Dafydd R; Perry, Benjamin G; Rosenberg, Saul H; Saikatendu, Kumar Singh; Schapira, Matthieu; Scholten, Cora; Sharma, Sujata; Simeonov, Anton; Sundström, Michael; Superti-Furga, Giulio; Todd, Matthew H; Tredup, Claudia; Vedadi, Masoud; von Delft, Frank; Willson, Timothy M; Winter, Georg E; Workman, Paul; Arrowsmith, Cheryl H

Comparative structural analyses of the NHL domains from the human E3 ligase TRIM-NHL family

人类E3连接酶TRIM-NHL家族NHL结构域的比较结构分析

Chaikuad, Apirat; Zhubi, Rezart; Tredup, Claudia; Knapp, Stefan

Controlling the Covalent Reactivity of a Kinase Inhibitor with Light

利用光控制激酶抑制剂的共价反应性

Reynders, Martin; Chaikuad, Apirat; Berger, Benedict-Tilman; Bauer, Katharina; Koch, Pierre; Laufer, Stefan; Knapp, Stefan; Trauner, Dirk