日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Allosteric inhibition of JAK2 with lysine-reactive compounds that bind the pseudokinase domain

利用与假激酶结构域结合的赖氨酸反应性化合物对JAK2进行变构抑制

Primi, Marina C; Tavares, Maurício T; Hatcher, John M; Kang, Hyelim; Kresina, Tomás A C; Chakraborty, Sayan; Leroy, Emilie; Schmoker, Anna M; Jeon, Hyesung; Weisberg, Ellen L; Akatsu, Taisei; Griffin, James D; Scott, David A; Eck, Michael J

Discovery of Pan-TEAD Inhibitors That Disrupt YAP-TEAD Interaction as a Potential Therapy for Gastric Cancers and Mutant KRAS and EGFR Lung Cancers

发现可破坏YAP-TEAD相互作用的泛TEAD抑制剂,有望成为胃癌以及KRAS和EGFR突变型肺癌的潜在疗法

Kumar, Ramesh; Thian, Joanne; Toh, Joel D W; Farzana, Noorul; Sun, Jialin; Kang, CongBao; Low, Suet Mei Crystal; Wee, Sheena; Lim, Zijie; Gunaratne, Jayantha; Loh, Hui Mun; Kannan, Srinivasaraghavan; Verma, Chandra S; Chakraborty, Sayan; Hong, Wanjin

Structure and function of the human apoptotic scramblase Xkr4

人类凋亡调控酶Xkr4的结构和功能

Chakraborty, Sayan; Feng, Zhang; Lee, Sangyun; Alvarenga, Omar E; Panda, Aniruddha; Zhang, Shuming; Bruni, Renato; Khelashvili, George; Gupta, Kallol; Accardi, Alessio

An Agrin-YAP/TAZ Rigidity Sensing Module Drives EGFR-Addicted Lung Tumorigenesis.

Agrin-YAP/TAZ 刚性传感模块驱动 EGFR 依赖性肺肿瘤发生

Mokhtari Reza Bayat, Sampath Divyaleka, Eversole Paige, Yu Lin Melissa Ong, Bosykh Dmitriy A, Boopathy Gandhi T K, Sivakumar Aravind, Wang Cheng-Chun, Kumar Ramesh, Sheng Joe Yeong Poh, Karasik Ellen, Foster Barbara A, Yu Han, Ling Xiang, Wu Wenjie, Li Fengzhi, Ohler Zoë Weaver, Brainson Christine F, Goodrich David W, Hong Wanjin, Chakraborty Sayan

A Comprehensive Oncological Biomarker Framework Guiding Precision Medicine

指导精准医疗的综合肿瘤生物标志物框架

Mokhtari, Reza Bayat; Sambi, Manpreet; Shekari, Faezeh; Satari, Kosar; Ghafoury, Roya; Ashayeri, Neda; Eversole, Paige; Baluch, Narges; Harless, William W; Muscarella, Lucia Anna; Yeger, Herman; Das, Bikul; Szewczuk, Myron R; Chakraborty, Sayan

HER2-Low Breast Cancer at the Interface of Pathology and Technology: Toward Precision Management

HER2低表达乳腺癌:病理学与技术交叉领域的研究进展——迈向精准治疗

Shekari, Faezeh; Bayat Mokhtari, Reza; Salahandish, Razieh; Sambi, Manpreet; Tarrahi, Roshanak; Salehi, Mahsa; Ashayeri, Neda; Eversole, Paige; Szewczuk, Myron R; Chakraborty, Sayan; Baluch, Narges

RAF isoform selectivity of MEK inhibitors and rational design of a covalent ARAF-MEK inhibitor

MEK抑制剂的RAF亚型选择性及共价ARAF-MEK抑制剂的合理设计

Chakraborty, Sayan; Jiang, Jie; Camallonga, Javier Vinals; Gazgalis, Dimitris; Gero, Thomas W; Tavares, Maurício T; Dittemore, Georgia; Tkacik, Emre; Jang, Dong Man; Ha, Byung Hak; Gottlieb, Felix H; Levitz, Talya; Metivier, Rebecca J; Schmoker, Anna M; Scott, David A; Jeon, Hyesung; Jänne, Pasi A; Eck, Michael J

Secrets of DNA-PKcs beyond DNA repair

DNA-PKcs 修复之外的秘密

Camfield, Sydney; Chakraborty, Sayan; Dwivedi, Shailendra Kumar Dhar; Pramanik, Pijush Kanti; Mukherjee, Priyabrata; Bhattacharya, Resham

Circulatory Agrin Serves as a Prognostic Indicator for Hepatocellular Carcinoma

循环Agrin可作为肝细胞癌的预后指标

Kapoor, Ankita; Bayat Mokhtari, Reza; Sonti, Sahithi Savithri; Patel, Riya; George, Anthony; Attwood, Kristopher; Iyer, Renuka; Chakraborty, Sayan

In or out of the groove? Mechanisms of lipid scrambling by TMEM16 proteins

位于沟槽内还是沟槽外?TMEM16蛋白介导的脂质重排机制

Feng, Zhang; Di Zanni, Eleonora; Alvarenga, Omar; Chakraborty, Sayan; Rychlik, Nicole; Accardi, Alessio