日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Reversible male contraception by targeted inhibition of serine/threonine kinase 33

通过靶向抑制丝氨酸/苏氨酸激酶33实现可逆性男性避孕

Ku, Angela F; Sharma, Kiran L; Ta, Hai Minh; Sutton, Courtney M; Bohren, Kurt M; Wang, Yong; Chamakuri, Srinivas; Chen, Ruihong; Hakenjos, John M; Jimmidi, Ravikumar; Kent, Katarzyna; Li, Feng; Li, Jian-Yuan; Ma, Lang; Madasu, Chandrashekhar; Palaniappan, Murugesan; Palmer, Stephen S; Qin, Xuan; Robers, Matthew B; Sankaran, Banumathi; Tan, Zhi; Vasquez, Yasmin M; Wang, Jian; Wilkinson, Jennifer; Yu, Zhifeng; Ye, Qiuji; Young, Damian W; Teng, Mingxing; Kim, Choel; Matzuk, Martin M

Discovery of highly potent and ALK2/ALK1 selective kinase inhibitors using DNA-encoded chemistry technology.

利用DNA编码化学技术发现高效且对ALK2/ALK1具有选择性的激酶抑制剂

Jimmidi Ravikumar, Monsivais Diana, Ta Hai Minh, Sharma Kiran L, Bohren Kurt M, Chamakuri Srinivas, Liao Zian, Li Feng, Hakenjos John M, Li Jian-Yuan, Mishina Yuji, Pan Haichun, Qin Xuan, Robers Matthew B, Sankaran Banumathi, Tan Zhi, Tang Suni, Vasquez Yasmin M, Wilkinson Jennifer, Young Damian W, Palmer Stephen S, MacKenzie Kevin R, Kim Choel, Matzuk Martin M

Expanding Complex Morpholines Using Systematic Chemical Diversity

利用系统化学多样性扩展复杂吗啉

Tang, Sunny Ann; Fults, Afton; Boyd, Shelton R; Gattu, Nikhil; Tran, Kevin A; Fan, Jiayi; MacKenzie, Kevin R; Palzkill, Timothy; Young, Damian W; Chamakuri, Srinivas

Chemical Catalysis Guides Structural Identification for the Major In Vivo Metabolite of the BET Inhibitor JQ1

化学催化指导BET抑制剂JQ1主要体内代谢物的结构鉴定

Holmes, Secondra; Jain, Prashi; Rodriguez, Kenneth Guzman; Williams, Jade; Yu, Zhifeng; Cerda-Smith, Christian; Samuel, Errol L G; Campbell, James; Hakenjos, John Michael; Monsivais, Diana; Li, Feng; Chamakuri, Srinivas; Matzuk, Martin M; Santini, Conrad; MacKenzie, Kevin R; Young, Damian W

Synthesis and Optimization of Small Molecule Inhibitors of Prostate Specific Antigen

前列腺特异性抗原小分子抑制剂的合成与优化

Erickson, Jeffery A; Jimmidi, Ravikumar; Anamthathmakula, Prashanth; Qin, Xuan; Wang, Jian; Gong, Leyi; Park, Jaehyeon; Koolpe, Gary; Tan, Caitlin; Matzuk, Martin M; Li, Feng; Chamakuri, Srinivas; Winuthayanon, Wipawee

Awareness, attitudes and cost among patients for dental implants in teeth replacement

患者对牙齿种植的认知、态度和费用

Kaur, Maninderjit; Chamakuri, Kirithana; Parashar, Pranav; Hiten Shah, Charmee; Singh, Pargat; Touchan, Layal

DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors

DNA 编码化学库产生非共价和非肽类 SARS-CoV-2 主要蛋白酶抑制剂

Ravikumar Jimmidi #, Srinivas Chamakuri #, Shuo Lu #, Melek Nihan Ucisik, Peng-Jen Chen, Kurt M Bohren, Seyed Arad Moghadasi, Leroy Versteeg, Christina Nnabuife, Jian-Yuan Li, Xuan Qin, Ying-Chu Chen, John C Faver, Pranavanand Nyshadham, Kiran L Sharma, Banumathi Sankaran, Allison Judge, Zhifeng Yu,

Heterocyclic Merging of Stereochemically Diverse Chiral Piperazines and Morpholines with Indazoles

立体化学结构多样的手性哌嗪和吗啉与吲唑的杂环融合

Viveki, Amol B; Mansfield, Timothy M; Tran, Kevin A; Lenkeit, Evan; MacKenzie, Kevin R; Young, Damian W; Chamakuri, Srinivas

Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 Mpro/3CLpro in Living Cells

信号增益分析探测活细胞中 SARS-CoV-2 Mpro/3CLpro 的抑制情况

Seyed Arad Moghadasi, Morgan A Esler, Yuka Otsuka, Jordan T Becker, Sofia N Moraes, Constance B Anderson, Srinivas Chamakuri, Christopher Belica, Chloe Wick, Daniel A Harki, Damian W Young, Louis Scampavia, Timothy P Spicer, Ke Shi, Hideki Aihara, William L Brown, Reuben S Harris

The iTHRIV Commons: a cross-institution information and health research data sharing architecture and web application

iTHRIV Commons:一个跨机构的信息和健康研究数据共享架构和网络应用程序

Loomba, Johanna Jean; Wasson, Glenn S; Chamakuri, Ravi Kiran Reddy; Dash, Pabitra Kumar; Patterson, Stephen G; Potter, Mary M A; Krisch, Jason Edward; Tenzer, Martha M; Johnston, Karen C; Brown, Don E