日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Low-Efficacy Mu Opioid Agonists as Candidate Analgesics: Effects of Novel C-9 Substituted Phenylmorphans on Pain-Depressed Behavior in Mice.

低效μ阿片受体激动剂作为候选镇痛药：新型C-9取代苯基吗啡烷对小鼠疼痛抑制行为的影响

期刊:Journal of Pharmacology and Experimental Therapeutics
影响因子:3.8
doi:10.1124/jpet.124.002153
Santos Edna J, Akbarali Hamid I, Bow Eric W, Chambers Dana R, Gutman Eugene S, Jacobson Arthur E, Kang Minho, Lee Young K, Lutz Joshua A, Rice Kenner C, Sulima Agnieszka, Negus S Stevens
信号转导
发表日期：2024
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A MOR Antagonist with High Potency and Antagonist Efficacy among Diastereomeric C9-Alkyl-Substituted N-Phenethyl-5-(3-hydroxy)phenylmorphans

在非对映异构体 C9-烷基取代的 N-苯乙基-5-(3-羟基)苯基吗啡烷中，一种具有高活性和拮抗功效的 MOR 拮抗剂

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules28145411
Chambers, Dana R; Sulima, Agnieszka; Luo, Dan; Prisinzano, Thomas E; Jacobson, Arthur E; Rice, Kenner C
发表日期：2023
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A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists

非对映异构体空间之旅：新型高效非对映异构体MOR激动剂和拮抗剂的设计、合成、体外和体内药理活性及分子建模

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules27196455
Chambers, Dana R; Sulima, Agnieszka; Luo, Dan; Prisinzano, Thomas E; Goldberg, Alexander; Xie, Bing; Shi, Lei; Paronis, Carol A; Bergman, Jack; Nassehi, Nima; Selley, Dana E; Imler, Gregory H; Jacobson, Arthur E; Rice, Kenner C
发表日期：2022
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