日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fragment-Based Drug Discovery of Novel High-affinity, Selective, and Anti-inflammatory Inhibitors of the Keap1-Nrf2 Protein-Protein Interaction

基于片段的新型高亲和力、选择性抗炎抑制剂在Keap1-Nrf2蛋白-蛋白相互作用中的应用

Lin, Chunyu; Narayanan, Dilip; Barreca, Marilia; Poulsen, Cecilie; da Costa, Leandro Silva; Chen, Xiangrong; Wichman, Kendall G; Charley, Cherisse A; Lindsay, Jaslin L; Dezfouli, Mahya; Vlissari, Dimitra; Mortensen, Thomas S; Chan, Camilla B; Wang, Jingyi; Richardson, William; Manning, Charlotte E; Chen, Zhuoyao; Zang, Jie; Käck, Helena; Gajhede, Michael; Bullock, Alex N; Blake, David J; Olagnier, David; Bach, Anders

A functional map of phosphoprotein phosphatase regulation identifies an evolutionary conserved reductase for the catalytic metal ions.

磷蛋白磷酸酶调控的功能图谱确定了一种进化上保守的催化金属离子还原酶

Meeusen Bob, Ambjørn Sara M, Veis Jiri, Riley Rachel C, Vit Gianmatteo, Brauer Brooke L, Møller Mads H, Greiner Elora C, Chan Camilla B, Weisser Melanie B, Garvanska Dimitriya H, Zhu Hao, Davey Norman E, Kettenbach Arminja N, Ogris Egon, Nilsson Jakob