日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Different chemical scaffolds bind to L-phe site in Mycobacterium tuberculosis Phe-tRNA synthetase

不同的化学支架与结核分枝杆菌Phe-tRNA合成酶中的L-phe位点结合。

Gade, Priyanka; Chang, Changsoo; Pryde, Denise S; Fletcher, Daniel; Niven, Sarah; Magalhaes, Luma Godoy; Robinson, David; Saini, Jagmohan; Ibrahim, Peter E G F; Forte, Barbara; Wower, Jacek; Bodkin, Michael J; Baragaña, Beatriz; Gilbert, Ian H; Michalska, Karolina; Joachimiak, Andrzej

Structural genomics of bacterial drug targets: Application of a high-throughput pipeline to solve 58 protein structures from pathogenic and related bacteria

细菌药物靶点的结构基因组学:应用高通量流程解析致病菌及相关细菌的58个蛋白质结构

Inniss, Nicole L; Minasov, George; Chang, Changsoo; Tan, Kemin; Kim, Youngchang; Maltseva, Natalia; Stogios, Peter; Filippova, Ekaterina; Michalska, Karolina; Osipiuk, Jerzy; Jaroszewki, Lukasz; Godzik, Adam; Savchenko, Alexei; Joachimiak, Andrzej; Anderson, Wayne F; Satchell, Karla J F

Cofactorless oxygenases guide anthraquinone-fused enediyne biosynthesis

无辅因子加氧酶指导蒽醌稠合烯二炔的生物合成

Gui, Chun; Kalkreuter, Edward; Liu, Yu-Chen; Li, Gengnan; Steele, Andrew D; Yang, Dong; Chang, Changsoo; Shen, Ben

Solvent organization in the ultrahigh-resolution crystal structure of crambin at room temperature

室温下克拉宾超高分辨率晶体结构中的溶剂组织

Chen, Julian C H; Gilski, Miroslaw; Chang, Changsoo; Borek, Dominika; Rosenbaum, Gerd; Lavens, Alex; Otwinowski, Zbyszek; Kubicki, Maciej; Dauter, Zbigniew; Jaskolski, Mariusz; Joachimiak, Andrzej

Intramolecular C-C Bond Formation Links Anthraquinone and Enediyne Scaffolds in Tiancimycin Biosynthesis

分子内C-C键的形成连接天西霉素生物合成中的蒽醌和烯二炔骨架。

Gui, Chun; Kalkreuter, Edward; Liu, Yu-Chen; Adhikari, Ajeeth; Teijaro, Christiana N; Yang, Dong; Chang, Changsoo; Shen, Ben

Docking study of transmembrane serine protease type 2 inhibitors for the treatment of COVID-19

跨膜丝氨酸蛋白酶2型抑制剂治疗COVID-19的分子对接研究

Mercado, Jonathan M; Lee, Sukyeong; Chang, Changsoo; Sung, Nuri; Soong, Lynn; Catic, Andre; Tsai, Francis T F; Solanki, Naishadh

Mycobacterium tuberculosis Phe-tRNA synthetase: structural insights into tRNA recognition and aminoacylation

结核分枝杆菌Phe-tRNA合成酶:tRNA识别和氨酰化的结构解析

Michalska, Karolina; Jedrzejczak, Robert; Wower, Jacek; Chang, Changsoo; Baragaña, Beatriz; Gilbert, Ian H; Forte, Barbara; Joachimiak, Andrzej

Tipiracil binds to uridine site and inhibits Nsp15 endoribonuclease NendoU from SARS-CoV-2

替吡嘧啶与尿苷结合位点,抑制SARS-CoV-2的Nsp15核糖核酸内切酶NendoU。

Kim, Youngchang; Wower, Jacek; Maltseva, Natalia; Chang, Changsoo; Jedrzejczak, Robert; Wilamowski, Mateusz; Kang, Soowon; Nicolaescu, Vlad; Randall, Glenn; Michalska, Karolina; Joachimiak, Andrzej

Allosteric inhibitors of Mycobacterium tuberculosis tryptophan synthase

结核分枝杆菌色氨酸合成酶的变构抑制剂

Michalska, Karolina; Chang, Changsoo; Maltseva, Natalia I; Jedrzejczak, Robert; Robertson, Gregory T; Gusovsky, Fabian; McCarren, Patrick; Schreiber, Stuart L; Nag, Partha P; Joachimiak, Andrzej

Characterization and Crystal Structure of a Nonheme Diiron Monooxygenase Involved in Platensimycin and Platencin Biosynthesis

参与普拉替霉素和普拉替霉素生物合成的非血红素双铁单加氧酶的表征和晶体结构

Dong, Liao-Bin; Liu, Yu-Chen; Cepeda, Alexis J; Kalkreuter, Edward; Deng, Ming-Rong; Rudolf, Jeffrey D; Chang, Changsoo; Joachimiak, Andrzej; Phillips, George N Jr; Shen, Ben