日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Production of Clinical-Grade SARS-CoV-2 Spike Ferritin Nanoparticle Protein Immunogen by Transient Transfection

利用瞬时转染法生产临床级SARS-CoV-2刺突蛋白铁蛋白纳米颗粒免疫原

Hajduczki, Agnes; Chang, William C; De La Barrera, Rafael; Wood, James F; Chen, Wei-Hung; Martinez, Elizabeth J; Jensen, Jaime L; Sankhala, Rajeshwer S; Smith, Clayton; Anderson, Alexander; Morrison, Elaine B; Peterson, Caroline E; Rees, Phyllis A; Soman, Sandrine; Kuklis, Caitlin; Ahmed, Aslaa; King, Jocelyn; Nasar, Farooq; Corbitt, Courtney; Choe, Misook; Thomas, Paul V; Zemil, Michelle; Wieczorek, Lindsay; Polonis, Victoria R; Dooley, Helen M; Mascola, John R; de Val, Natalie; Matyas, Gary R; Rao, Mangala; Gromowski, Gregory D; Modjarrad, Kayvon; Vasan, Sandhya; Froude, Jeffrey W; Michael, Nelson L; Joyce, M Gordon; Zarling, Stasya

Antibody targeting of conserved sites of vulnerability on the SARS-CoV-2 spike receptor-binding domain.

针对SARS-CoV-2刺突蛋白受体结合域上保守易感位点的抗体

Sankhala Rajeshwer S, Dussupt Vincent, Chen Wei-Hung, Bai Hongjun, Martinez Elizabeth J, Jensen Jaime L, Rees Phyllis A, Hajduczki Agnes, Chang William C, Choe Misook, Yan Lianying, Sterling Spencer L, Swafford Isabella, Kuklis Caitlin, Soman Sandrine, King Jocelyn, Corbitt Courtney, Zemil Michelle, Peterson Caroline E, Mendez-Rivera Letzibeth, Townsley Samantha M, Donofrio Gina C, Lal Kerri G, Tran Ursula, Green Ethan C, Smith Clayton, de Val Natalia, Laing Eric D, Broder Christopher C, Currier Jeffrey R, Gromowski Gregory D, Wieczorek Lindsay, Rolland Morgane, Paquin-Proulx Dominic, van Dyk Dewald, Britton Zachary, Rajan Saravanan, Loo Yueh Ming, McTamney Patrick M, Esser Mark T, Polonis Victoria R, Michael Nelson L, Krebs Shelly J, Modjarrad Kayvon, Joyce M Gordon

Structure-guided design of direct-acting antivirals that exploit the gem-dimethyl effect and potently inhibit 3CL proteases of severe acute respiratory syndrome Coronavirus-2 (SARS-CoV-2) and middle east respiratory syndrome coronavirus (MERS-CoV)

利用结构引导设计直接作用的抗病毒药物,利用二甲基效应有效抑制严重急性呼吸综合征冠状病毒 2 (SARS-CoV-2) 和中东呼吸综合征冠状病毒 (MERS-CoV) 的 3CL 蛋白酶

Chamandi S Dampalla, Matthew J Miller, Yunjeong Kim, Alexandria Zabiegala, Harry Nhat Nguyen, Trent K Madden, Hayden A Thurman, Alexandra J Machen, Anne Cooper, Lijun Liu, Kevin P Battaile, Scott Lovell, Kyeong-Ok Chang, William C Groutas

Structure-Guided Design of Potent Spirocyclic Inhibitors of Severe Acute Respiratory Syndrome Coronavirus-2 3C-like Protease

严重急性呼吸综合征冠状病毒-2 3C 样蛋白酶强效螺环抑制剂的结构指导设计

Chamandi S Dampalla, Athri D Rathnayake, Anushka C Galasiti Kankanamalage, Yunjeong Kim, Krishani Dinali Perera, Harry Nhat Nguyen, Matthew J Miller, Trent K Madden, Hunter R Picard, Hayden A Thurman, Maithri M Kashipathy, Lijun Liu, Kevin P Battaile, Scott Lovell, Kyeong-Ok Chang, William C Groutas

Broad-Spectrum Cyclopropane-Based Inhibitors of Coronavirus 3C-like Proteases: Biochemical, Structural, and Virological Studies

基于环丙烷的广谱冠状病毒 3C 样蛋白酶抑制剂:生化、结构和病毒学研究

Chamandi S Dampalla, Harry Nhat Nguyen, Athri D Rathnayake, Yunjeong Kim, Krishani Dinali Perera, Trent K Madden, Hayden A Thurman, Alexandra J Machen, Maithri M Kashipathy, Lijun Liu, Kevin P Battaile, Scott Lovell, Kyeong-Ok Chang, William C Groutas

Structure-Guided Design of Conformationally Constrained Cyclohexane Inhibitors of Severe Acute Respiratory Syndrome Coronavirus-2 3CL Protease

严重急性呼吸综合征冠状病毒-2 3CL 蛋白酶的构象约束环己烷抑制剂的结构引导设计

Chamandi S Dampalla, Yunjeong Kim, Naemi Bickmeier, Athri D Rathnayake, Harry Nhat Nguyen, Jian Zheng, Maithri M Kashipathy, Matthew A Baird, Kevin P Battaile, Scott Lovell, Stanley Perlman, Kyeong-Ok Chang, William C Groutas

Efficacy of a Broadly Neutralizing SARS-CoV-2 Ferritin Nanoparticle Vaccine in Nonhuman Primates

广谱中和SARS-CoV-2铁蛋白纳米颗粒疫苗在非人灵长类动物中的疗效

Joyce, Michael G; King, Hannah A D; Naouar, Ines Elakhal; Ahmed, Aslaa; Peachman, Kristina K; Cincotta, Camila Macedo; Subra, Caroline; Chen, Rita E; Thomas, Paul V; Chen, Wei-Hung; Sankhala, Rajeshwer S; Hajduczki, Agnes; Martinez, Elizabeth J; Peterson, Caroline E; Chang, William C; Choe, Misook; Smith, Clayton; Lee, Parker J; Headley, Jarrett A; Taddese, Mekdi G; Elyard, Hanne A; Cook, Anthony; Anderson, Alexander; McGuckin-Wuertz, Kathryn; Dong, Ming; Swafford, Isabella; Case, James B; Currier, Jeffrey R; Lal, Kerri G; O'Connell, Robert J; Molnar, Sebastian; Nair, Manoj S; Dussupt, Vincent; Daye, Sharon P; Zeng, Xiankun; Barkei, Erica K; Staples, Hilary M; Alfson, Kendra; Carrion, Ricardo; Krebs, Shelly J; Paquin-Proulx, Dominic; Karasavva, Nicos; Polonis, Victoria R; Jagodzinski, Linda L; Amare, Mihret F; Vasan, Sandhya; Scott, Paul T; Huang, Yaoxing; Ho, David D; de Val, Natalia; Diamond, Michael S; Lewis, Mark G; Rao, Mangala; Matyas, Gary R; Gromowski, Gregory D; Peel, Sheila A; Michael, Nelson L; Bolton, Diane L; Modjarrad, Kayvon

Comparative Analysis of Thrombin Calibration Algorithms and Correction for Thrombin-α2macroglobulin Activity

凝血酶校准算法的比较分析及凝血酶-α2巨球蛋白活性校正

Chang, William C; Jackson, Joseph W; Machlus, Kellie R; Wolberg, Alisa S; Ovanesov, Mikhail V

Efficient RNA drug delivery using red blood cell extracellular vesicles

利用红细胞胞外囊泡高效递送RNA药物

Waqas Muhammad Usman ,Tin Chanh Pham ,Yuk Yan Kwok ,Luyen Tien Vu ,Victor Ma ,Boya Peng ,Yuen San Chan ,Likun Wei ,Siew Mei Chin ,Ajijur Azad ,Alex Bai-Liang He ,Anskar Y H Leung ,Mengsu Yang ,Ng Shyh-Chang ,William C Cho ,Jiahai Shi ,Minh T N Le

Structure-guided design of potent and permeable inhibitors of MERS coronavirus 3CL protease that utilize a piperidine moiety as a novel design element

利用哌啶部分作为新型设计元素,以结构为指导设计 MERS 冠状病毒 3CL 蛋白酶的强效、渗透性抑制剂

Anushka C Galasiti Kankanamalage, Yunjeong Kim, Vishnu C Damalanka, Athri D Rathnayake, Anthony R Fehr, Nurjahan Mehzabeen, Kevin P Battaile, Scott Lovell, Gerald H Lushington, Stanley Perlman, Kyeong-Ok Chang, William C Groutas