Drugging the catalytically inactive state of RET kinase in RET-rearranged tumors
针对RET重排肿瘤中RET激酶催化失活状态的药物治疗
期刊:Science Translational Medicine
影响因子:14.6
doi:10.1126/scitranslmed.aah6144
Plenker, Dennis; Riedel, Maximilian; Brägelmann, Johannes; Dammert, Marcel A; Chauhan, Rakhee; Knowles, Phillip P; Lorenz, Carina; Keul, Marina; Bührmann, Mike; Pagel, Oliver; Tischler, Verena; Scheel, Andreas H; Schütte, Daniel; Song, Yanrui; Stark, Justina; Mrugalla, Florian; Alber, Yannic; Richters, André; Engel, Julian; Leenders, Frauke; Heuckmann, Johannes M; Wolf, Jürgen; Diebold, Joachim; Pall, Georg; Peifer, Martin; Aerts, Maarten; Gevaert, Kris; Zahedi, René P; Buettner, Reinhard; Shokat, Kevan M; McDonald, Neil Q; Kast, Stefan M; Gautschi, Oliver; Thomas, Roman K; Sos, Martin L