日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanistic insights into the therapeutic properties of delta opioid receptor

对δ阿片受体治疗特性的机制性见解

Bernhard, Sarah M; Roy Chowdhury, Susovan; Murata, Tsuyoshi; Reinl, Erin L; Ramos-Gonzalez, Nokomis; Denn, Elizabeth; Appourchaux, Kevin; Inoue, Asuka; England, Sarah K; Fay, Jonathan F; Majumdar, Susruta; Chanda, Baron; Che, Tao

Polar regions are critical in achieving global sustainable development goals

极地地区对于实现全球可持续发展目标至关重要

Li, Xin; Guo, Huadong; Cheng, Guodong; Song, Xiaoyu; Ran, Youhua; Feng, Min; Che, Tao; Li, Xinwu; Wang, Lei; Duan, Anmin; Shangguan, Donghui; Chen, Deliang; Jin, Rui; Deng, Jie; Su, Jianbin; Cao, Bin

Structure-guided design of partial agonists at an opioid receptor.

基于结构的阿片受体部分激动剂设计

Varga Balazs R, Bernhard Sarah M, El Daibani Amal, Zaidi Saheem A, Lam Jordy H, Aguilar Jhoan, Appourchaux Kevin, Nazarova Antonina L, Kouvelis Alexa, Shinouchi Ryosuke, Hammond Haylee R, Eans Shainnel O, Weinreb Violetta, Margolis Elyssa B, Fay Jonathan F, Huang Xi-Ping, Pradhan Amynah, Katritch Vsevolod, McLaughlin Jay P, Majumdar Susruta, Che Tao

Global carbon flux dataset generated by fusing remote sensing and multiple flux networks observation

融合遥感和多通量网络观测数据生成的全球碳通量数据集

Yuan, Qiwang; Wang, Xufeng; Che, Tao; Li, Jun

Searching for Synthetic Opioid Rescue Agents. 2: Identification of an Ultra-Potent Synthetic Opioid Rescue Agent

寻找合成阿片类药物解救剂。2:超强效合成阿片类药物解救剂的鉴定

Martin, Jocelyn; Onyameh, Edem; Luo, Dan; Powell, Joshua W; Trivedi, Riya R; Woloshin, Eric J; Zhang, Yating; Shaykin, Jakob D; Denehy, Emily D; Alsum, Alexia R; Prantzalos, Emily; Jiang, Qianru; Che, Tao; Alilain, Warren J; Turner, Jill R; Bardo, Michael T; Prisinzano, Thomas E

Macranthoside B Suppresses the Growth of Adenocarcinoma of Esophagogastric Junction by Regulating Iron Homeostasis and Ferroptosis through NRF2 Inhibition

大花苷B通过抑制NRF2调节铁稳态和铁死亡,从而抑制食管胃交界处腺癌的生长

Wang, Lingling; Pan, Guangzhao; Tian, Sichao; Zhang, Che; Tao, Fangfang; Qin, Jiang-Jiang

How Ligands Achieve Biased Signaling toward Arrestins

配体如何实现对阻遏蛋白的偏向性信号传导

Jiang, Qianru; Che, Tao

Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Michael Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Differential effects of sodium on agonist-induced conformational transitions and signaling at μ and κ opioid receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma M; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

A µ-opioid receptor modulator that works cooperatively with naloxone.

一种与纳洛酮协同作用的μ-阿片受体调节剂

O'Brien Evan S, Rangari Vipin Ashok, El Daibani Amal, Eans Shainnel O, Hammond Haylee R, White Elizabeth, Wang Haoqing, Shiimura Yuki, Krishna Kumar Kaavya, Jiang Qianru, Appourchaux Kevin, Huang Weijiao, Zhang Chensong, Kennedy Brandon J, Mathiesen Jesper M, Che Tao, McLaughlin Jay P, Majumdar Susruta, Kobilka Brian K