日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PI3Kα Inhibitor and Degrader Inavolisib Can Co-opt FGFR2 to Enhance Responses in Patients with PIK3CA-Mutated Solid Tumors and in Preclinical Models.

PI3Kα抑制剂和降解剂Inavolisib可利用FGFR2增强PIK3CA突变实体瘤患者和临床前模型的疗效。

Juric Dejan, Song Kyung, Johnson Radia M, Accordino Melissa K, Bedard Philippe L, Cervantes Andrés, Gambardella Valentina, Hamilton Erika, Italiano Antoine, Kalinsky Kevin, Krop Ian E, Oliveira Mafalda, Saura Cristina, Schmid Peter, Turner Nicholas C, Varga Andreea, Gendreau Steven, Hwang Michael S, Kuang Zheng, Lau Jeffrey T, Lin Eva, Pham Trang, Maddalo Danilo, Rees Matthew G, Ronan Melissa M, Roth Jennifer A, Martin Scott, Sodir Nicole M, Sokol Ethan S, Whitfield Zachary J, Wong Alice, Yauch Robert L, Aimi Junko, Cheeti Sravanthi, Fredrickson Jill, Hilz Stephanie, Hafner Marc, Hutchinson Katherine E, Jin Yanling, Peters Ubong, Zingg Daniel, Royer-Joo Stephanie, Shankar Noopur, Schutzman Jennifer L, Jhaveri Komal L, Dey Anwesha

An IQ Consortium Perspective on the FDA Guidance for Assessment of Pharmacokinetics in Participants With Impaired Renal Function

IQ联盟对FDA关于肾功能受损患者药代动力学评估指南的看法

Jin, Yan; Sharma, Ashish; Ahmed, Mariam A; Cheeti, Sravanthi; Ou, Ying; Devineni, Damayanthi; Chen, Yizhe; Kanodia, Jitendra S; Abouelhassan, Yasmeen; Noormohamed, Nadia; Zhou, Jin; Marroum, Patrick; Sahasrabudhe, Vaishali; Younis, Islam R

Identifying lung cancer in Emergency Department patients outside national lung cancer screening guidelines

在国家肺癌筛查指南之外,识别急诊科患者的肺癌

Wang, Hao; Cheeti, Radhika; Murray, Miles; Muirheid, Timothy A; McDowell, Jasmine; Sambamoorthi, Usha

Phase I/Ib Trial of Inavolisib Plus Palbociclib and Endocrine Therapy for PIK3CA-Mutated, Hormone Receptor-Positive, Human Epidermal Growth Factor Receptor 2-Negative Advanced or Metastatic Breast Cancer

Inavolisib联合Palbociclib和内分泌疗法治疗PIK3CA突变、激素受体阳性、人表皮生长因子受体2阴性晚期或转移性乳腺癌的I/Ib期临床试验

Jhaveri, Komal L; Accordino, Melissa K; Bedard, Philippe L; Cervantes, Andrés; Gambardella, Valentina; Hamilton, Erika; Italiano, Antoine; Kalinsky, Kevin; Krop, Ian E; Oliveira, Mafalda; Schmid, Peter; Saura, Cristina; Turner, Nicholas C; Varga, Andrea; Cheeti, Sravanthi; Hilz, Stephanie; Hutchinson, Katherine E; Jin, Yanling; Royer-Joo, Stephanie; Peters, Ubong; Shankar, Noopur; Schutzman, Jennifer L; Juric, Dejan

Exploring the Impact of Hepatic Impairment on Pralsetinib Pharmacokinetics

探讨肝功能损害对普拉替尼药代动力学的影响

Cheung, Kit Wun Kathy; Tang, Yang; Anders, Doreen; Barata, Teresa; Scalori, Astrid; Agarwal, Priya; Sane, Rucha; Cheeti, Sravanthi

Predicting overall survival from tumor dynamics metrics using parametric statistical and machine learning models: application to patients with RET-altered solid tumors

利用参数统计和机器学习模型,根据肿瘤动力学指标预测总生存期:应用于RET基因改变的实体瘤患者

Velasquez, Erick; Kassir, Nastya; Cheeti, Sravanthi; Kuruvilla, Denison; Sane, Rucha; Dang, Steve; Miles, Dale; Lu, James

Understanding CYP3A4 and P-gp mediated drug-drug interactions through PBPK modeling - Case example of pralsetinib

通过PBPK模型了解CYP3A4和P-gp介导的药物相互作用——以普拉替尼为例

Bowman, Christine; Dolton, Michael; Ma, Fang; Cheeti, Sravanthi; Kuruvilla, Denison; Sane, Rucha; Kassir, Nastya; Chen, Yuan

An Open-label Phase I Study of GDC-0927 in Postmenopausal Women with Locally Advanced or Metastatic Estrogen Receptor-Positive Breast Cancer

一项针对绝经后局部晚期或转移性雌激素受体阳性乳腺癌女性患者的GDC-0927开放标签I期研究

Chandarlapaty, Sarat; Dickler, Maura N; Perez Fidalgo, Jose Alejandro; Villanueva-Vázquez, Rafael; Giltnane, Jennifer; Gates, Mary; Chang, Ching-Wei; Cheeti, Sravanthi; Fredrickson, Jill; Wang, Xiaojing; Collier, Ann; Moore, Heather M; Metcalfe, Ciara; Lauchle, Jennifer; Humke, Eric W; Bardia, Aditya

The oral selective estrogen receptor degrader GDC-0810 (ARN-810) in postmenopausal women with hormone receptor-positive HER2-negative (HR + /HER2 -) advanced/metastatic breast cancer

口服选择性雌激素受体降解剂 GDC-0810 (ARN-810) 用于治疗绝经后激素受体阳性/HER2阴性 (HR+/HER2-) 晚期/转移性乳腺癌

Bardia, Aditya; Mayer, Ingrid; Winer, Eric; Linden, Hannah M; Ma, Cynthia X; Parker, Barbara A; Bellet, Meritxell; Arteaga, Carlos L; Cheeti, Sravanthi; Gates, Mary; Chang, Ching-Wei; Fredrickson, Jill; Spoerke, Jill M; Moore, Heather M; Giltnane, Jennifer; Friedman, Lori S; Chow Maneval, Edna; Chan, Iris; Jhaveri, Komal

Diagnostic implications of neuroimaging in epilepsy and other seizure disorders

神经影像学在癫痫和其他癫痫发作性疾病诊断中的应用

Nieto-Salazar, Maria A; Velasquez-Botero, Felipe; Toro-Velandia, Adriana C; Saldana-Rodriguez, Ericka A; Rodriguez-Rodriguez, Miguel E; Gupta, Aditi; Cheeti, Srinidhi; Huerta-Rengifo, Claudia; Pavón-Enamorado, Fredy R; Rodezno, Carmen M C; Medina, Patrick S D; De-Sario-Velasquez, Gioacchino D M S; Sah, Biki K; Shaheen, Fatima; Shree, Anagha; Sah, Rajan K