日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Arginase Inhibitors: An Overview

精氨酸酶抑制剂的合成:概述

Molaro, Maria Cristina; Battisegola, Chiara; Schiano, Marica Erminia; Failla, Mariacristina; Rimoli, Maria Grazia; Lazzarato, Loretta; Chegaev, Konstantin; Sodano, Federica

Special Issue "Development and Synthesis of Biologically Active Compounds"

特刊“生物活性化合物的开发与合成”

Gazieva, Galina A; Chegaev, Konstantin

Use of Enzymatically Activated Carbon Monoxide Donors for Sensitizing Drug-Resistant Tumor Cells

使用酶活化的一氧化碳供体来增强耐药肿瘤细胞的敏感性

Federica Sodano, Barbara Rolando, Loretta Lazzarato, Costanzo Costamagna, Mariacristina Failla, Chiara Riganti, Konstantin Chegaev

Multitarget Antioxidant NO-Donor Organic Nitrates: A Novel Approach to Overcome Nitrates Tolerance, an Ex Vivo Study

多靶点抗氧化剂NO供体有机硝酸盐:克服硝酸盐耐受性的新方法——一项离体研究

Marini, Elisabetta; Giorgis, Marta; Leporati, Marta; Rolando, Barbara; Chegaev, Konstantin; Lazzarato, Loretta; Bertinaria, Massimo; Vincenti, Marco; Di Stilo, Antonella

A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors

对 Sdox(一种有前景的 H2S 释放阿霉素,可用于治疗化疗耐药性肿瘤)的全面评估

Petko Alov, Merilin Al Sharif, Denitsa Aluani, Konstantin Chegaev, Jelena Dinic, Aleksandra Divac Rankov, Miguel X Fernandes, Fabio Fusi, Alfonso T García-Sosa, Risto Juvonen, Magdalena Kondeva-Burdina, José M Padrón, Ilza Pajeva, Tania Pencheva, Adrián Puerta, Hannu Raunio, Chiara Riganti, Ivanka T

Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts

含有释放 H2S 的阿霉素的透明质酸化脂质体对 P-糖蛋白阳性/阿霉素耐药的骨肉瘤细胞和异种移植有效

Elena Gazzano, Ilaria Buondonno, Alessandro Marengo, Barbara Rolando, Konstantin Chegaev, Joanna Kopecka, Simona Saponara, Matteo Sorge, Claudia Maria Hattinger, Alberto Gasco, Roberta Fruttero, Mara Brancaccio, Massimo Serra, Barbara Stella, Elias Fattal, Silvia Arpicco, Chiara Riganti

Endoplasmic reticulum-targeting doxorubicin: a new tool effective against doxorubicin-resistant osteosarcoma

内质网靶向阿霉素:一种有效治疗阿霉素耐药性骨肉瘤的新工具

Ilaria Buondonno, Elena Gazzano, Elisa Tavanti, Konstantin Chegaev, Joanna Kopecka, Marilù Fanelli, Barbara Rolando, Roberta Fruttero, Alberto Gasco, Claudia Hattinger, Massimo Serra, Chiara Riganti

Discovery of phenylsulfonylfuroxan derivatives as gamma globin inducers by histone acetylation

通过组蛋白乙酰化发现苯磺酰基呋喃酮衍生物作为γ珠蛋白诱导剂

Thais Regina Ferreira de Melo, Chutima Kumkhaek, Guilherme Felipe Dos Santos Fernandes, Maria Elisa Lopes Pires, Rafael Consolin Chelucci, Karina Pereira Barbieri, Fernanda Coelho, Ticiana Sidorenko de Oliveira Capote, Carolina Lanaro, Iracilda Zeppone Carlos, Sisi Marcondes, Konstantin Chegaev, Ste

New tetrahydroisoquinoline-based P-glycoprotein modulators: decoration of the biphenyl core gives selective ligands

新型四氢异喹啉基P-糖蛋白调节剂:联苯核心的修饰可得到选择性配体

Contino, Marialessandra; Guglielmo, Stefano; Perrone, Maria Grazia; Giampietro, Roberta; Rolando, Barbara; Carrieri, Antonio; Zaccaria, Daniele; Chegaev, Konstantin; Borio, Vanessa; Riganti, Chiara; Zabielska-Koczywąs, Katarzyna; Colabufo, Nicola A; Fruttero, Roberta

Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity

设计、合成和表征具有体内杀菌抗结核活性的含N-氧化物杂环化合物

Dos Santos Fernandes, Guilherme Felipe; de Souza, Paula Carolina; Moreno-Viguri, Elsa; Santivañez-Veliz, Mery; Paucar, Rocio; Pérez-Silanes, Silvia; Chegaev, Konstantin; Guglielmo, Stefano; Lazzarato, Loretta; Fruttero, Roberta; Man Chin, Chung; da Silva, Patricia Bento; Chorilli, Marlus; Solcia, Mariana Cristina; Ribeiro, Camila Maríngolo; Silva, Caio Sander Paiva; Marino, Leonardo Biancolino; Bosquesi, Priscila Longhin; Hunt, Debbie M; de Carvalho, Luiz Pedro S; de Souza Costa, Carlos Alberto; Cho, Sang Hyun; Wang, Yuehong; Franzblau, Scott Gary; Pavan, Fernando Rogério; Dos Santos, Jean Leandro