日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dual function of Zika virus NS2B-NS3 protease

寨卡病毒 NS2B-NS3 蛋白酶的双重功能

Sergey A Shiryaev, Piotr Cieplak, Anton Cheltsov, Robert C Liddington, Alexey V Terskikh

Allosteric inhibitor of β-catenin selectively targets oncogenic Wnt signaling in colon cancer

β-catenin 的变构抑制剂选择性靶向结肠癌中的致癌 Wnt 信号

Anton Cheltsov, Natsuko Nomura, Venkata M Yenugonda, Jatin Roper, Rajesh Mukthavaram, Pengfei Jiang, Nam-Gu Her, Ivan Babic, Santosh Kesari, Elmar Nurmemmedov

Multi-Omics Studies towards Novel Modulators of Influenza A Virus-Host Interaction

针对甲型流感病毒-宿主相互作用新型调节因子的多组学研究

Söderholm, Sandra; Fu, Yu; Gaelings, Lana; Belanov, Sergey; Yetukuri, Laxman; Berlinkov, Mikhail; Cheltsov, Anton V; Anders, Simon; Aittokallio, Tero; Nyman, Tuula A; Matikainen, Sampsa; Kainov, Denis E

NSC-640358 acts as RXRα ligand to promote TNFα-mediated apoptosis of cancer cell

NSC-640358 作为 RXRα 配体促进 TNFα 介导的癌细胞凋亡

Fan Chen #, Jiebo Chen #, Jiacheng Lin #, Anton V Cheltsov, Lin Xu, Ya Chen, Zhiping Zeng, Liqun Chen, Mingfeng Huang, Mengjie Hu, Xiaohong Ye, Yuqi Zhou, Guanghui Wang, Ying Su, Long Zhang, Fangfang Zhou, Xiao-Kun Zhang, Hu Zhou

TRAIL-Based High Throughput Screening Reveals a Link between TRAIL-Mediated Apoptosis and Glutathione Reductase, a Key Component of Oxidative Stress Response

基于 TRAIL 的高通量筛选揭示了 TRAIL 介导的细胞凋亡与氧化应激反应的关键成分谷胱甘肽还原酶之间的联系

Dmitri Rozanov, Anton Cheltsov, Eduard Sergienko, Stefan Vasile, Vladislav Golubkov, Alexander E Aleshin, Trevor Levin, Elie Traer, Byron Hann, Julia Freimuth, Nikita Alexeev, Max A Alekseyev, Sergey P Budko, Hans Peter Bächinger, Paul Spellman

RNF4 interacts with both SUMO and nucleosomes to promote the DNA damage response

RNF4 与 SUMO 和核小体相互作用,从而促进 DNA 损伤反应。

Groocock, Lynda M; Nie, Minghua; Prudden, John; Moiani, Davide; Wang, Tao; Cheltsov, Anton; Rambo, Robert P; Arvai, Andrew S; Hitomi, Chiharu; Tainer, John A; Luger, Karolin; Perry, J Jefferson P; Lazzerini-Denchi, Eros; Boddy, Michael N

Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes

通过同时对人和小鼠同工酶进行超高通量筛选,鉴定出一种小鼠肠道碱性磷酸酶选择性抑制剂(ML260)。

Ardecky, Robert J; Bobkova, Ekaterina V; Kiffer-Moreira, Tina; Brown, Brock; Ganji, Santhi; Zou, Jiwen; Pass, Ian; Narisawa, Sonoko; Iano, Flávia Godoy; Rosenstein, Craig; Cheltsov, Anton; Rascon, Justin; Hedrick, Michael; Gasior, Carlton; Forster, Anita; Shi, Shenghua; Dahl, Russell; Vasile, Stefan; Su, Ying; Sergienko, Eduard; Chung, Thomas D Y; Kaunitz, Jonathan; Hoylaerts, Marc F; Pinkerton, Anthony B; Millán, José Luis

Novel MT1-MMP small-molecule inhibitors based on insights into hemopexin domain function in tumor growth

基于对血红素结合蛋白结构域在肿瘤生长中功能的洞察,研发新型 MT1-MMP 小分子抑制剂

Albert G Remacle, Vladislav S Golubkov, Sergey A Shiryaev, Russell Dahl, John L Stebbins, Andrei V Chernov, Anton V Cheltsov, Maurizio Pellecchia, Alex Y Strongin

Virtual ligand screening of the National Cancer Institute (NCI) compound library leads to the allosteric inhibitory scaffolds of the West Nile Virus NS3 proteinase

利用美国国家癌症研究所 (NCI) 化合物库进行虚拟配体筛选,获得了西尼罗河病毒 NS3 蛋白酶的变构抑制剂骨架。

Shiryaev, Sergey A; Cheltsov, Anton V; Gawlik, Katarzyna; Ratnikov, Boris I; Strongin, Alex Y

Refined structures of placental alkaline phosphatase show a consistent pattern of interactions at the peripheral site

胎盘碱性磷酸酶的精细结构显示其外周部位存在一致的相互作用模式。

Stec, Boguslaw; Cheltsov, Anton; Millán, José Luis