Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes
通过同时对人和小鼠同工酶进行超高通量筛选,鉴定出一种小鼠肠道碱性磷酸酶选择性抑制剂(ML260)。
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2013.12.043
Ardecky, Robert J; Bobkova, Ekaterina V; Kiffer-Moreira, Tina; Brown, Brock; Ganji, Santhi; Zou, Jiwen; Pass, Ian; Narisawa, Sonoko; Iano, Flávia Godoy; Rosenstein, Craig; Cheltsov, Anton; Rascon, Justin; Hedrick, Michael; Gasior, Carlton; Forster, Anita; Shi, Shenghua; Dahl, Russell; Vasile, Stefan; Su, Ying; Sergienko, Eduard; Chung, Thomas D Y; Kaunitz, Jonathan; Hoylaerts, Marc F; Pinkerton, Anthony B; Millán, José Luis