日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural Mechanism of an Efficacy Photoswitch Targeting the β(2)-adrenergic Receptor

靶向β(2)-肾上腺素能受体的高效光开关的结构机制

Stipp, Robin; Bertrand, Quentin; Trabuco, Matilde; Duran-Corbera, Anna; Ignazzitto, Maria Tindara; Glover, Hannah; Stierli, Fabienne; Catena, Juanlo; Carrillo, Melissa; Hartmann, Sina; Seidel, Hans-Peter; Mulder, Matthias; Mason, Thomas; Kondo, Yasushi; Wranik, Maximillian; Appleby, Martin; Sager, Christoph; Sierra, Raymond; Gate, Gregory; Schleissner, Pamela; Cheng, Xinxin; Weinert, Tobias; Cheng, Robert; Mous, Sandra; Beale, John H; Kepa, Michal; Llebaria, Amadeu; Hennig, Michael; Rovira, Xavier; Standfuss, Joerg

Elevated tumor NOS2/COX2 promotes immunosuppressive phenotypes associated with poor survival in ER- breast cancer

肿瘤NOS2/COX2水平升高会促进与ER阴性乳腺癌患者预后不良相关的免疫抑制表型。

Ridnour, Lisa A; Cheng, Robert Ys; Heinz, William F; Pore, Milind; Gonzalez, Ana L; Femino, Elise L; Moffat, Rebecca L; Wink, Adelaide L; Imtiaz, Fatima; Coutinho, Leandro L; Butcher, Donna; Edmondson, Elijah F; Rangel, M Cristina; Wong, Stephen Tc; Lipkowitz, Stanley; Glynn, Sharon A; Vitek, Michael P; McVicar, Daniel W; Li, Xiaoxian; Anderson, Stephen K; Paolocci, Nazareno; Hewitt, Stephen M; Ambs, Stefan; Billiar, Timothy R; Chang, Jenny C; Lockett, Stephen J; Wink, David A

Apo-state structure of the metabotropic glutamate receptor 5 transmembrane domain obtained using a photoswitchable ligand.

利用光开关配体获得的代谢型谷氨酸受体5跨膜结构域的无配体状态结构

Kondo Yasushi, Hatton Caitlin, Cheng Robert, Trabuco Matilde, Glover Hannah, Bertrand Quentin, Stierli Fabienne, Seidel Hans-Peter, Mason Thomas, Sarma Sivathmika, Tellkamp Friedjof, Kepa Michal, Dworkowski Florian, Mehrabi Pedram, Hennig Michael, Standfuss Joerg

RETRACTED: Waheed et al. Nitric Oxide Donor DETA/NO Inhibits the Growth of Endometrial Cancer Cells by Upregulating the Expression of RASSF1 and CDKN1A. Molecules 2019, 24, 3722

撤稿:Waheed 等人,《一氧化氮供体 DETA/NO 通过上调 RASSF1 和 CDKN1A 的表达抑制子宫内膜癌细胞的生长》,Molecules 2019, 24, 3722

Waheed, Sana; Cheng, Robert Ys; Casablanca, Yovanni; Maxwell, G Larry; Wink, David A; Syed, Viqar

Photoswitch dissociation from a G protein-coupled receptor resolved by time-resolved serial crystallography

利用时间分辨连续晶体学解析光开关从G蛋白偶联受体上的解离

Glover, Hannah; Saßmannshausen, Torben; Bertrand, Quentin; Trabuco, Matilde; Slavov, Chavdar; Bacchin, Arianna; Andres, Fabio; Kondo, Yasushi; Stipp, Robin; Wranik, Maximilian; Khusainov, Georgii; Carrillo, Melissa; Kekilli, Demet; Nan, Jie; Gonzalez, Ana; Cheng, Robert; Neidhart, Werner; Weinert, Tobias; Leonarski, Filip; Dworkowski, Florian; Kepa, Michal; Wachtveitl, Josef; Hennig, Michael; Standfuss, Joerg

UBR5 promotes antiviral immunity by disengaging the transcriptional brake on RIG-I like receptors

UBR5通过解除RIG-I样受体的转录抑制来促进抗病毒免疫。

Duomeng Yang ,Tingting Geng ,Andrew G Harrison ,Jason G Cahoon ,Jian Xing ,Baihai Jiao ,Mark Wang ,Chao Cheng ,Robert E Hill ,Huadong Wang ,Anthony T Vella ,Gong Cheng ,Yanlin Wang ,Penghua Wang

Macrophage depletion protects against cisplatin-induced ototoxicity and nephrotoxicity

巨噬细胞耗竭可预防顺铂引起的耳毒性和肾毒性

Cathy Yea Won Sung ,Naoki Hayase ,Peter S T Yuen ,John Lee ,Katharine Fernandez ,Xuzhen Hu ,Hui Cheng ,Robert A Star ,Mark E Warchol ,Lisa L Cunningham

Comprehensive Integration of Multiple Single-Cell Transcriptomic Data Sets Defines Distinct Cell Populations and Their Phenotypic Changes in Murine Atherosclerosis

综合整合多个单细胞转录组数据集定义小鼠动脉粥样硬化中的不同细胞群及其表型变化

Disha Sharma, Matthew D Worssam, Albert J Pedroza, Alex R Dalal, Haizea Alemany, Hyun-Jung Kim, Ramendra Kundu, Michael P Fischbein, Paul Cheng #, Robert Wirka #, Thomas Quertermous #

Impacts of CACNB4 overexpression on dendritic spine density in both sexes and relevance to schizophrenia

CACNB4 过表达对两性树突棘密度的影响及其与精神分裂症的相关性

Emily M Parker, Nathan L Kindja, Rebecca A DeGiosio, Ryan B Salisbury, Josh M Krivinko, Claire E J Cheetham, Matthew L MacDonald, Weijia Fan, Bin Cheng, Robert A Sweet

NOS2 and COX-2 Co-Expression Promotes Cancer Progression: A Potential Target for Developing Agents to Prevent or Treat Highly Aggressive Breast Cancer

NOS2 和 COX-2 共表达促进癌症进展:开发预防或治疗高侵袭性乳腺癌药物的潜在靶点

Coutinho, Leandro L; Femino, Elise L; Gonzalez, Ana L; Moffat, Rebecca L; Heinz, William F; Cheng, Robert Y S; Lockett, Stephen J; Rangel, M Cristina; Ridnour, Lisa A; Wink, David A