日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Origin and bioactivities of thiosulfinated FK228.

硫代亚磺酸酯化FK228的来源和生物活性

Liu Xiangyang, Currens Grant C, Xue Liang, Cheng Yi-Qiang

Chromobacterium spp. mediate their anti-Plasmodium activity through secretion of the histone deacetylase inhibitor romidepsin.

色杆菌属通过分泌组蛋白去乙酰化酶抑制剂罗米地辛来发挥其抗疟原虫活性

Saraiva Raúl G, Huitt-Roehl Callie R, Tripathi Abhai, Cheng Yi-Qiang, Bosch Jürgen, Townsend Craig A, Dimopoulos George

Histone deacetylase inhibitor thailandepsin-A activates Notch signaling and suppresses neuroendocrine cancer cell growth in vivo

组蛋白去乙酰化酶抑制剂泰国素A激活Notch信号通路并抑制体内神经内分泌癌细胞的生长

Jang, Samuel; Janssen, Andrew; Aburjania, Zviadi; Robers, Matthew B; Harrison, April; Dammalapati, Ajitha; Cheng, Yi-Qiang; Chen, Herbert; Jaskula-Sztul, Renata

Minimum Information about a Biosynthetic Gene cluster

生物合成基因簇的最低信息

Medema, Marnix H; Kottmann, Renzo; Yilmaz, Pelin; Cummings, Matthew; Biggins, John B; Blin, Kai; de Bruijn, Irene; Chooi, Yit Heng; Claesen, Jan; Coates, R Cameron; Cruz-Morales, Pablo; Duddela, Srikanth; Düsterhus, Stephanie; Edwards, Daniel J; Fewer, David P; Garg, Neha; Geiger, Christoph; Gomez-Escribano, Juan Pablo; Greule, Anja; Hadjithomas, Michalis; Haines, Anthony S; Helfrich, Eric J N; Hillwig, Matthew L; Ishida, Keishi; Jones, Adam C; Jones, Carla S; Jungmann, Katrin; Kegler, Carsten; Kim, Hyun Uk; Kötter, Peter; Krug, Daniel; Masschelein, Joleen; Melnik, Alexey V; Mantovani, Simone M; Monroe, Emily A; Moore, Marcus; Moss, Nathan; Nützmann, Hans-Wilhelm; Pan, Guohui; Pati, Amrita; Petras, Daniel; Reen, F Jerry; Rosconi, Federico; Rui, Zhe; Tian, Zhenhua; Tobias, Nicholas J; Tsunematsu, Yuta; Wiemann, Philipp; Wyckoff, Elizabeth; Yan, Xiaohui; Yim, Grace; Yu, Fengan; Xie, Yunchang; Aigle, Bertrand; Apel, Alexander K; Balibar, Carl J; Balskus, Emily P; Barona-Gómez, Francisco; Bechthold, Andreas; Bode, Helge B; Borriss, Rainer; Brady, Sean F; Brakhage, Axel A; Caffrey, Patrick; Cheng, Yi-Qiang; Clardy, Jon; Cox, Russell J; De Mot, René; Donadio, Stefano; Donia, Mohamed S; van der Donk, Wilfred A; Dorrestein, Pieter C; Doyle, Sean; Driessen, Arnold J M; Ehling-Schulz, Monika; Entian, Karl-Dieter; Fischbach, Michael A; Gerwick, Lena; Gerwick, William H; Gross, Harald; Gust, Bertolt; Hertweck, Christian; Höfte, Monica; Jensen, Susan E; Ju, Jianhua; Katz, Leonard; Kaysser, Leonard; Klassen, Jonathan L; Keller, Nancy P; Kormanec, Jan; Kuipers, Oscar P; Kuzuyama, Tomohisa; Kyrpides, Nikos C; Kwon, Hyung-Jin; Lautru, Sylvie; Lavigne, Rob; Lee, Chia Y; Linquan, Bai; Liu, Xinyu; Liu, Wen; Luzhetskyy, Andriy; Mahmud, Taifo; Mast, Yvonne; Méndez, Carmen; Metsä-Ketelä, Mikko; Micklefield, Jason; Mitchell, Douglas A; Moore, Bradley S; Moreira, Leonilde M; Müller, Rolf; Neilan, Brett A; Nett, Markus; Nielsen, Jens; O'Gara, Fergal; Oikawa, Hideaki; Osbourn, Anne; Osburne, Marcia S; Ostash, Bohdan; Payne, Shelley M; Pernodet, Jean-Luc; Petricek, Miroslav; Piel, Jörn; Ploux, Olivier; Raaijmakers, Jos M; Salas, José A; Schmitt, Esther K; Scott, Barry; Seipke, Ryan F; Shen, Ben; Sherman, David H; Sivonen, Kaarina; Smanski, Michael J; Sosio, Margherita; Stegmann, Evi; Süssmuth, Roderich D; Tahlan, Kapil; Thomas, Christopher M; Tang, Yi; Truman, Andrew W; Viaud, Muriel; Walton, Jonathan D; Walsh, Christopher T; Weber, Tilmann; van Wezel, Gilles P; Wilkinson, Barrie; Willey, Joanne M; Wohlleben, Wolfgang; Wright, Gerard D; Ziemert, Nadine; Zhang, Changsheng; Zotchev, Sergey B; Breitling, Rainer; Takano, Eriko; Glöckner, Frank Oliver

Identification and characterization of the spiruchostatin biosynthetic gene cluster enable yield improvement by overexpressing a transcriptional activator.

通过过表达转录激活因子,可以鉴定和表征螺旋菌素生物合成基因簇,从而提高产量

Potharla Vishwakanth Y, Wang Cheng, Cheng Yi-Qiang

The novel histone deacetylase inhibitor thailandepsin A inhibits anaplastic thyroid cancer growth

新型组蛋白去乙酰化酶抑制剂泰国肽A可抑制未分化甲状腺癌的生长

Weinlander, Eric; Somnay, Yash; Harrison, April D; Wang, Cheng; Cheng, Yi-Qiang; Jaskula-Sztul, Renata; Yu, Xiao-Min; Chen, Herbert

Thailandepsins are new small molecule class I HDAC inhibitors with potent cytotoxic activity in ovarian cancer cells: a preclinical study of epigenetic ovarian cancer therapy

Thailandepsins 是一种新型小分子 I 类 HDAC 抑制剂,对卵巢癌细胞具有强效细胞毒活性:一项表观遗传卵巢癌治疗的临床前研究

Wilson, Andrew J; Cheng, Yi-Qiang; Khabele, Dineo

New insights into the genetic organization of the FK228 biosynthetic gene cluster in Chromobacterium violaceum no. 968

对紫色色杆菌968号菌株中FK228生物合成基因簇的遗传组织有了新的认识

Potharla, Vishwakanth Y; Wesener, Shane R; Cheng, Yi-Qiang

Acyldepsipeptide antibiotics induce the formation of a structured axial channel in ClpP: A model for the ClpX/ClpA-bound state of ClpP.

酰基缩肽类抗生素诱导 ClpP 中形成结构化的轴向通道:ClpP 与 ClpX/ClpA 结合状态的模型

Li Dominic Him Shun, Chung Yu Seon, Gloyd Melanie, Joseph Ebenezer, Ghirlando Rodolfo, Wright Gerard D, Cheng Yi-Qiang, Maurizi Michael R, Guarné Alba, Ortega Joaquin

Novel features of the polysaccharide-digesting gliding bacterium Flavobacterium johnsoniae as revealed by genome sequence analysis

基因组序列分析揭示了消化多糖的滑行细菌约翰逊黄杆菌的新特征

McBride, Mark J; Xie, Gary; Martens, Eric C; Lapidus, Alla; Henrissat, Bernard; Rhodes, Ryan G; Goltsman, Eugene; Wang, Wei; Xu, Jian; Hunnicutt, David W; Staroscik, Andrew M; Hoover, Timothy R; Cheng, Yi-Qiang; Stein, Jennifer L