日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure basis of ligand recognition and activation of GPR55

GPR55配体识别和激活的结构基础

Chang, Hao; Li, Xiaoting; Shen, Ling; Ge, Xuanrui; Hao, Shuming; Wu, Lijie; Liu, Shenhui; Liu, Junlin; Cherezov, Vadim; Hua, Tian

Novel fold and wing structure of Forkhead transcription factor facilitate DNA binding

叉头转录因子的新型折叠和翼状结构促进其与DNA的结合

George L Wang,Yibei Jiang,Yuying Sun,Fariborz Nasertorabi,Jesse A Weller,Raktim Mitra,Alexander Batyuk,Oscar M Aparicio,Vadim Cherezov,Remo Rohs

Structural insights into the mechanism of activation and inhibition of the prostaglandin D2 receptor 1.

前列腺素D2受体1激活和抑制机制的结构性见解

Davoudinasab Behnaz, Raskovalov Aleksey, Lee Woojin, Kim Donggyun, Kim Heesoo, Lam Jordy Homing, Han Gye Won, Katritch Vsevolod, Cherezov Vadim

Opportunistic use of artificial intelligence with X-ray imaging for diagnosis of HIV status in tuberculosis patients in Uganda and Tanzania

在乌干达和坦桑尼亚,利用人工智能和X射线成像技术对结核病患者进行艾滋病毒感染状况诊断的机会性应用

Cherezov, Dmitrii; Dam, Tanmoy; Najjingo, Irene; Mbabazi, Margaret; Kisembo, Harriet; Kirenga, Bruce; Soka, Grace; Ngadaya, Esther; Mfinanga, Sayoki; Madabhushi, Anant

Unlocking GPCR-ligand interactions: Measuring binding affinities with thermal shift assay

揭示GPCR-配体相互作用:利用热位移分析法测定结合亲和力

Dashevskii, Dmitrii; Luginina, Aleksandra; Maslov, Ivan; Shevelyova, Marina; Khorn, Polina; Dmitrieva, Daria; Kapranov, Ivan; Belousov, Anatolii; Permyakov, Sergei; Cherezov, Vadim; Borshchevskiy, Valentin; Mishin, Alexey

Nicotinamide Riboside and CD38: Covalent Inhibition and Live-Cell Labeling.

烟酰胺核苷和 CD38:共价抑制和活细胞标记

Kao Guoyun, Zhang Xiao-Nan, Nasertorabi Fariborz, Katz Benjamin B, Li Zeyang, Dai Zhefu, Zhang Zeyu, Zhang Lei, Louie Stan G, Cherezov Vadim, Zhang Yong

Structural insights into the high basal activity and inverse agonism of the orphan receptor GPR6 implicated in Parkinson's disease.

帕金森病中孤儿受体 GPR6 的高基础活性和反向激动作用的结构见解

Barekatain Mahta, Johansson Linda C, Lam Jordy H, Chang Hao, Sadybekov Anastasiia V, Han Gye Won, Russo Joseph, Bliesath Joshua, Brice Nicola L, Carlton Mark B L, Saikatendu Kumar S, Sun Hukai, Murphy Sean T, Monenschein Holger, Schiffer Hans H, Popov Petr, Lutomski Corinne A, Robinson Carol V, Liu Zhi-Jie, Hua Tian, Katritch Vsevolod, Cherezov Vadim

Insulator-based dielectrophoresis-assisted separation of insulin secretory vesicles

基于绝缘体的介电泳辅助分离胰岛素分泌囊泡

Mahta Barekatain #, Yameng Liu #, Ashley Archambeau, Vadim Cherezov, Scott Fraser, Kate L White, Mark A Hayes

Monitoring GPCR conformation with GFP-inspired dyes

利用GFP类似染料监测GPCR构象

Anatoliy Belousov ,Ivan Maslov ,Philipp Orekhov ,Polina Khorn ,Pavel Kuzmichev ,Nadezhda Baleeva ,Vladislav Motov ,Andrey Bogorodskiy ,Svetlana Krasnova ,Konstantin Mineev ,Dmitry Zinchenko ,Evgeni Zernii ,Valentin Ivanovich ,Sergei Permyakov ,Johan Hofkens ,Jelle Hendrix ,Vadim Cherezov ,Thomas Gensch ,Alexander Mishin ,Mikhail Baranov ,Alexey Mishin ,Valentin Borshchevskiy

Native mass spectrometry prescreening of G protein-coupled receptor complexes for cryo-EM structure determination.

利用天然质谱法对 G 蛋白偶联受体复合物进行预筛选,以进行冷冻电镜结构测定

Kim Donggyun, Liu Weijing, Viner Rosa, Cherezov Vadim