日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of small-molecule binding sites of a ubiquitin-conjugating enzyme-UBE2T through fragment-based screening

通过基于片段的筛选鉴定泛素结合酶UBE2T的小分子结合位点

Loh, Yong Yao; Anantharajan, Jothi; Huang, Qiwei; Xu, Weijun; Fulwood, Justina; Ng, Hui Qi; Ng, Elizabeth Yihui; Gea, Chong Yu; Choong, Meng Ling; Tan, Qian Wen; Koh, Xiaoying; Lim, Wan Hsin; Nacro, Kassoum; Cherian, Joseph; Baburajendran, Nithya; Ke, Zhiyuan; Kang, CongBao

Hybrid Polystyrene-Plasmonic Systems as High Binding Density Biosensing Platforms

混合聚苯乙烯-等离子体系统作为高结合密度生物传感平台

Darr, Charles M; Hasan, Juiena; Mathai, Cherian Joseph; Gangopadhyay, Keshab; Gangopadhyay, Shubhra; Bok, Sangho

Fragment-based Discovery of a Small-Molecule Protein Kinase C-iota Inhibitor Binding Post-kinase Domain Residues

基于片段的发现小分子蛋白激酶C-ι抑制剂结合激酶后结构域残基

Kwiatkowski, Jacek; Baburajendran, Nithya; Poulsen, Anders; Liu, Boping; Tee, Doris Hui Ying; Wong, Yun Xuan; Poh, Zhi Ying; Ong, Esther Hq; Dinie, Nurul; Cherian, Joseph; Jansson, Anna Elisabet; Hill, Jeffrey; Keller, Thomas H; Hung, Alvin W

Small Molecules Targeting the Inactive Form of the Mnk1/2 Kinases

靶向Mnk1/2激酶非活性形式的小分子

Kannan, Srinivasaraghavan; Pradhan, Mohan R; Cherian, Joseph; Joseph, Thomas L; Poh, Zhi Ying; Hai Yan, Yang; Melvyn, Ho; Boping, Liu; Jeffrey, Hill; Nacro, Kassoum; Verma, Chandra S

Pharmacokinetics-pharmacodynamics analysis of bicyclic 4-nitroimidazole analogs in a murine model of tuberculosis

在结核病小鼠模型中对双环4-硝基咪唑类似物进行药代动力学-药效学分析

Lakshminarayana, Suresh B; Boshoff, Helena I M; Cherian, Joseph; Ravindran, Sindhu; Goh, Anne; Jiricek, Jan; Nanjundappa, Mahesh; Nayyar, Amit; Gurumurthy, Meera; Singh, Ramandeep; Dick, Thomas; Blasco, Francesca; Barry, Clifton E 3rd; Ho, Paul C; Manjunatha, Ujjini H

Structure of Ddn, the deazaflavin-dependent nitroreductase from Mycobacterium tuberculosis involved in bioreductive activation of PA-824

结核分枝杆菌中参与 PA-824 生物还原活化的脱氮黄素依赖性硝基还原酶 Ddn 的结构

Cellitti, Susan E; Shaffer, Jennifer; Jones, David H; Mukherjee, Tathagata; Gurumurthy, Meera; Bursulaya, Badry; Boshoff, Helena I; Choi, Inhee; Nayyar, Amit; Lee, Yong Sok; Cherian, Joseph; Niyomrattanakit, Pornwaratt; Dick, Thomas; Manjunatha, Ujjini H; Barry, Clifton E 3rd; Spraggon, Glen; Geierstanger, Bernhard H

Substrate specificity of the deazaflavin-dependent nitroreductase from Mycobacterium tuberculosis responsible for the bioreductive activation of bicyclic nitroimidazoles.

结核分枝杆菌脱氮黄素依赖性硝基还原酶的底物特异性,该酶负责双环硝基咪唑的生物还原活化

Gurumurthy Meera, Mukherjee Tathagata, Dowd Cynthia S, Singh Ramandeep, Niyomrattanakit Pornwaratt, Tay Jo Ann, Nayyar Amit, Lee Yong Sok, Cherian Joseph, Boshoff Helena I, Dick Thomas, Barry Clifton E 3rd, Manjunatha Ujjini H

Selective killing of nonreplicating mycobacteria

选择性杀灭非复制型分枝杆菌

Bryk, Ruslana; Gold, Benjamin; Venugopal, Aditya; Singh, Jasbir; Samy, Raghu; Pupek, Krzysztof; Cao, Hua; Popescu, Carmen; Gurney, Mark; Hotha, Srinivas; Cherian, Joseph; Rhee, Kyu; Ly, Lan; Converse, Paul J; Ehrt, Sabine; Vandal, Omar; Jiang, Xiuju; Schneider, Jean; Lin, Gang; Nathan, Carl