Fragment-Based Drug Discovery of Novel High-affinity, Selective, and Anti-inflammatory Inhibitors of the Keap1-Nrf2 Protein-Protein Interaction
基于片段的新型高亲和力、选择性抗炎抑制剂在Keap1-Nrf2蛋白-蛋白相互作用中的应用
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.202508121
Lin, Chunyu; Narayanan, Dilip; Barreca, Marilia; Poulsen, Cecilie; da Costa, Leandro Silva; Chen, Xiangrong; Wichman, Kendall G; Charley, Cherisse A; Lindsay, Jaslin L; Dezfouli, Mahya; Vlissari, Dimitra; Mortensen, Thomas S; Chan, Camilla B; Wang, Jingyi; Richardson, William; Manning, Charlotte E; Chen, Zhuoyao; Zang, Jie; Käck, Helena; Gajhede, Michael; Bullock, Alex N; Blake, David J; Olagnier, David; Bach, Anders